ECSP099692A - NEW VINYLLOID RECEIVER LINKS AND ITS USE OF THEM FOR THE PRODUCTION OF PHARMACEUTICAL SUBSTANCES - Google Patents

NEW VINYLLOID RECEIVER LINKS AND ITS USE OF THEM FOR THE PRODUCTION OF PHARMACEUTICAL SUBSTANCES

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Publication number
ECSP099692A
ECSP099692A EC2009009692A ECSP099692A ECSP099692A EC SP099692 A ECSP099692 A EC SP099692A EC 2009009692 A EC2009009692 A EC 2009009692A EC SP099692 A ECSP099692 A EC SP099692A EC SP099692 A ECSP099692 A EC SP099692A
Authority
EC
Ecuador
Prior art keywords
production
pharmaceutical substances
vinylloid
new
receiver links
Prior art date
Application number
EC2009009692A
Other languages
Spanish (es)
Inventor
Jee Woo Lee
Vry Jean Marie Victor De
Thomas Christoph
Robert Frank
Gregor Bahrenberg
Klaus Schiene
Derek John Sauders
Bernd Saudermann
Original Assignee
Gruenenthal Chemie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE102007018149A external-priority patent/DE102007018149A1/en
Application filed by Gruenenthal Chemie filed Critical Gruenenthal Chemie
Publication of ECSP099692A publication Critical patent/ECSP099692A/en

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14Radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
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    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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Abstract

La presente invención se relaciona con ligandos de receptor vainilloide novedosos, un método para la producción de los mismos, sustancias farmacéuticas que contienen dichos compuestos y el uso de tales compuestos para la producción de sustancias farmacéuticas.The present invention relates to novel vanilloid receptor ligands, a method for the production thereof, pharmaceutical substances containing said compounds and the use of such compounds for the production of pharmaceutical substances.

EC2009009692A 2007-04-16 2009-10-16 NEW VINYLLOID RECEIVER LINKS AND ITS USE OF THEM FOR THE PRODUCTION OF PHARMACEUTICAL SUBSTANCES ECSP099692A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102007018149A DE102007018149A1 (en) 2007-04-16 2007-04-16 Novel vanilloid receptor ligands and their use in the preparation of medicines
EP2008002997 2008-04-15
US12/103,667 US8084484B2 (en) 2007-04-16 2008-04-15 Vanilloid receptor ligands, pharmaceutical compositions containing them, process for making them, and use thereof for treating pain and other conditions

Publications (1)

Publication Number Publication Date
ECSP099692A true ECSP099692A (en) 2009-11-30

Family

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Application Number Title Priority Date Filing Date
EC2009009692A ECSP099692A (en) 2007-04-16 2009-10-16 NEW VINYLLOID RECEIVER LINKS AND ITS USE OF THEM FOR THE PRODUCTION OF PHARMACEUTICAL SUBSTANCES

Country Status (14)

Country Link
JP (1) JP2010523727A (en)
KR (1) KR20100016593A (en)
CN (1) CN101679370A (en)
AU (1) AU2008238250B2 (en)
BR (1) BRPI0810035A2 (en)
CA (1) CA2683461A1 (en)
CO (1) CO6241154A2 (en)
EC (1) ECSP099692A (en)
IL (1) IL201505A0 (en)
MX (1) MX2009011149A (en)
NZ (1) NZ580411A (en)
RU (1) RU2498982C2 (en)
WO (1) WO2008125342A2 (en)
ZA (1) ZA200907099B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102007018149A1 (en) 2007-04-16 2008-10-23 Grünenthal GmbH Novel vanilloid receptor ligands and their use in the preparation of medicines
CN106243037A (en) * 2009-05-07 2016-12-21 格吕伦塔尔有限公司 The substituted phenylurea of part and phenyl amide as Rhizoma et radix valerianae compounds receptor
US8946204B2 (en) 2009-05-07 2015-02-03 Gruenenthal Gmbh Substituted phenylureas and phenylamides as vanilloid receptor ligands
BR112014001908A2 (en) 2011-07-26 2017-02-21 Gruenenthal Gmbh substituted heterocyclic aza derivatives
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