ECSP099692A - NEW VINYLLOID RECEIVER LINKS AND ITS USE OF THEM FOR THE PRODUCTION OF PHARMACEUTICAL SUBSTANCES - Google Patents
NEW VINYLLOID RECEIVER LINKS AND ITS USE OF THEM FOR THE PRODUCTION OF PHARMACEUTICAL SUBSTANCESInfo
- Publication number
- ECSP099692A ECSP099692A EC2009009692A ECSP099692A ECSP099692A EC SP099692 A ECSP099692 A EC SP099692A EC 2009009692 A EC2009009692 A EC 2009009692A EC SP099692 A ECSP099692 A EC SP099692A EC SP099692 A ECSP099692 A EC SP099692A
- Authority
- EC
- Ecuador
- Prior art keywords
- production
- pharmaceutical substances
- vinylloid
- new
- receiver links
- Prior art date
Links
- 239000000126 substance Substances 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 102000011040 TRPV Cation Channels Human genes 0.000 abstract 1
- 108010062740 TRPV Cation Channels Proteins 0.000 abstract 1
- 239000003446 ligand Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D215/14—Radicals substituted by oxygen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D241/40—Benzopyrazines
- C07D241/42—Benzopyrazines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
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Abstract
La presente invención se relaciona con ligandos de receptor vainilloide novedosos, un método para la producción de los mismos, sustancias farmacéuticas que contienen dichos compuestos y el uso de tales compuestos para la producción de sustancias farmacéuticas.The present invention relates to novel vanilloid receptor ligands, a method for the production thereof, pharmaceutical substances containing said compounds and the use of such compounds for the production of pharmaceutical substances.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102007018149A DE102007018149A1 (en) | 2007-04-16 | 2007-04-16 | Novel vanilloid receptor ligands and their use in the preparation of medicines |
| EP2008002997 | 2008-04-15 | ||
| US12/103,667 US8084484B2 (en) | 2007-04-16 | 2008-04-15 | Vanilloid receptor ligands, pharmaceutical compositions containing them, process for making them, and use thereof for treating pain and other conditions |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP099692A true ECSP099692A (en) | 2009-11-30 |
Family
ID=41360190
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2009009692A ECSP099692A (en) | 2007-04-16 | 2009-10-16 | NEW VINYLLOID RECEIVER LINKS AND ITS USE OF THEM FOR THE PRODUCTION OF PHARMACEUTICAL SUBSTANCES |
Country Status (14)
| Country | Link |
|---|---|
| JP (1) | JP2010523727A (en) |
| KR (1) | KR20100016593A (en) |
| CN (1) | CN101679370A (en) |
| AU (1) | AU2008238250B2 (en) |
| BR (1) | BRPI0810035A2 (en) |
| CA (1) | CA2683461A1 (en) |
| CO (1) | CO6241154A2 (en) |
| EC (1) | ECSP099692A (en) |
| IL (1) | IL201505A0 (en) |
| MX (1) | MX2009011149A (en) |
| NZ (1) | NZ580411A (en) |
| RU (1) | RU2498982C2 (en) |
| WO (1) | WO2008125342A2 (en) |
| ZA (1) | ZA200907099B (en) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102007018149A1 (en) | 2007-04-16 | 2008-10-23 | Grünenthal GmbH | Novel vanilloid receptor ligands and their use in the preparation of medicines |
| CN106243037A (en) * | 2009-05-07 | 2016-12-21 | 格吕伦塔尔有限公司 | The substituted phenylurea of part and phenyl amide as Rhizoma et radix valerianae compounds receptor |
| US8946204B2 (en) | 2009-05-07 | 2015-02-03 | Gruenenthal Gmbh | Substituted phenylureas and phenylamides as vanilloid receptor ligands |
| BR112014001908A2 (en) | 2011-07-26 | 2017-02-21 | Gruenenthal Gmbh | substituted heterocyclic aza derivatives |
| MX2014000963A (en) | 2011-07-26 | 2014-03-27 | Gruenenthal Gmbh | Substituted bicyclic aromatic carboxamide and urea derivatives as vanilloid receptor ligands. |
| CA2854935A1 (en) * | 2011-11-09 | 2013-05-16 | Grunenthal Gmbh | Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an n-containing group as vanilloid receptor ligands |
| AU2013230425B2 (en) * | 2012-03-05 | 2017-05-25 | Dr.Reddy's Laboratories Ltd. | Substituted heterocyclic acetamides as kappa opioid receptor (kor) agonists |
| MA39145B1 (en) * | 2013-12-20 | 2018-05-31 | Esteve Labor Dr | Piperazine derivatives having multimode activity against pain |
| CN107721919B (en) * | 2017-10-30 | 2020-12-08 | 中国药科大学 | Phenylquinoline TRPV1 antagonist and preparation method and application thereof |
| KR102334947B1 (en) * | 2020-04-22 | 2021-12-06 | 주식회사 제이맥켐 | Benzimidazolone based cinnamamide derivatives as TRPV1 antagonists and a pharmaceutical composition for treating or preventing pain containing the same as an active ingredient |
| RU2755206C1 (en) | 2020-05-20 | 2021-09-14 | Федеральное государственное бюджетное учреждение науки Тихоокеанский институт биоорганической химии им. Г.Б. Елякова Дальневосточного отделения Российской академии наук (ТИБОХ ДВО РАН) | Agent with prolonged analgesic action and medicinal product based thereon |
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| CA2468159A1 (en) * | 2001-11-27 | 2003-06-05 | Merck & Co., Inc. | 4-aminoquinoline compounds |
| CA2476936A1 (en) * | 2002-02-20 | 2003-08-28 | Chih-Hung Lee | Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor |
| GB0206876D0 (en) * | 2002-03-22 | 2002-05-01 | Merck Sharp & Dohme | Therapeutic agents |
| US6933311B2 (en) * | 2003-02-11 | 2005-08-23 | Abbott Laboratories | Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor |
| AU2004234611A1 (en) * | 2003-04-29 | 2004-11-11 | Century Technology Inc | Method of diagnosing a genetic susceptibility for bone damage |
| SE0301446D0 (en) * | 2003-05-16 | 2003-05-16 | Astrazeneca Ab | New Compounds |
| KR20060027338A (en) * | 2003-06-12 | 2006-03-27 | 아스텔라스세이야쿠 가부시키가이샤 | Benzamide derivatives or salts thereof |
| US20050113576A1 (en) * | 2003-08-05 | 2005-05-26 | Chih-Hung Lee | Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor |
| GB0322016D0 (en) * | 2003-09-19 | 2003-10-22 | Merck Sharp & Dohme | New compounds |
| EP1685112B1 (en) * | 2003-11-08 | 2011-07-20 | Bayer Schering Pharma Aktiengesellschaft | Tetrahydro-quinolinylurea derivatives as vr1 antagonists |
| US20050165015A1 (en) * | 2004-01-23 | 2005-07-28 | Ncube Mghele V. | Vanilloid receptor ligands and their use in treatments |
| DE102005023943A1 (en) * | 2005-05-20 | 2006-11-23 | Grünenthal GmbH | Pentafluorosulfanyl-substituted compound and its use for the preparation of medicaments |
| AU2006336504C9 (en) * | 2005-12-28 | 2015-05-14 | Vertex Pharmaceuticals Incorporated | 1-(benzo [D] [1,3] dioxol-5-yl) -N- (phenyl) cyclopropane- carboxamide derivatives and related compounds as modulators of ATP-Binding Cassette transporters for the treatment of Cystic Fibrosis |
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2008
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- 2008-04-16 KR KR1020097023887A patent/KR20100016593A/en not_active Ceased
- 2008-04-16 CN CN200880020483A patent/CN101679370A/en active Pending
- 2008-04-16 AU AU2008238250A patent/AU2008238250B2/en not_active Ceased
- 2008-04-16 WO PCT/EP2008/003027 patent/WO2008125342A2/en not_active Ceased
- 2008-04-16 NZ NZ580411A patent/NZ580411A/en not_active IP Right Cessation
- 2008-04-16 JP JP2010503397A patent/JP2010523727A/en not_active Ceased
- 2008-04-16 RU RU2009142023/04A patent/RU2498982C2/en not_active IP Right Cessation
- 2008-04-16 MX MX2009011149A patent/MX2009011149A/en active IP Right Grant
- 2008-04-16 CA CA002683461A patent/CA2683461A1/en not_active Abandoned
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2009
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- 2009-10-16 EC EC2009009692A patent/ECSP099692A/en unknown
- 2009-10-22 CO CO09118505A patent/CO6241154A2/en active IP Right Grant
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| IL201505A0 (en) | 2010-05-31 |
| RU2009142023A (en) | 2011-05-27 |
| BRPI0810035A2 (en) | 2016-07-26 |
| WO2008125342A2 (en) | 2008-10-23 |
| NZ580411A (en) | 2012-06-29 |
| AU2008238250B2 (en) | 2013-01-24 |
| ZA200907099B (en) | 2013-03-27 |
| CO6241154A2 (en) | 2011-01-20 |
| MX2009011149A (en) | 2009-10-30 |
| WO2008125342A3 (en) | 2009-01-15 |
| RU2498982C2 (en) | 2013-11-20 |
| CN101679370A (en) | 2010-03-24 |
| JP2010523727A (en) | 2010-07-15 |
| CA2683461A1 (en) | 2008-10-23 |
| AU2008238250A1 (en) | 2008-10-23 |
| KR20100016593A (en) | 2010-02-12 |
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