ECSP099805A - NEW DERIVATIVES OF DICARBOXYL ACID AS AGONISTS OF S1P1 RECEPTORS - Google Patents
NEW DERIVATIVES OF DICARBOXYL ACID AS AGONISTS OF S1P1 RECEPTORSInfo
- Publication number
- ECSP099805A ECSP099805A ECSP099805A ECSP099805A EC SP099805 A ECSP099805 A EC SP099805A EC SP099805 A ECSP099805 A EC SP099805A EC SP099805 A ECSP099805 A EC SP099805A
- Authority
- EC
- Ecuador
- Prior art keywords
- receptors
- agonists
- new derivatives
- dicarboxyl acid
- compounds
- Prior art date
Links
- 239000000556 agonist Substances 0.000 title abstract 2
- 102100025750 Sphingosine 1-phosphate receptor 1 Human genes 0.000 title 1
- 101710155454 Sphingosine 1-phosphate receptor 1 Proteins 0.000 title 1
- 239000002253 acid Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- DUYSYHSSBDVJSM-KRWOKUGFSA-N sphingosine 1-phosphate Chemical compound CCCCCCCCCCCCC\C=C\[C@@H](O)[C@@H](N)COP(O)(O)=O DUYSYHSSBDVJSM-KRWOKUGFSA-N 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 1
- 229940125721 immunosuppressive agent Drugs 0.000 abstract 1
- 239000003018 immunosuppressive agent Substances 0.000 abstract 1
- 230000004968 inflammatory condition Effects 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención se refiere a nuevos compuestos de fórmula (I) que poseen actividad agonista con respecto a los receptores de esfingosina-1 -fosfato (S1P), a su procedimiento de preparación y su uso como agentes inmunosupresores. La invención también se refiere a composiciones farmacéuticas que contienen estos compuestos y al uso de estos compuestos para el tratamiento/la prevención de enfermedades y condiciones mediadas inmunológicamente y condiciones o enfermedades inflamatorias.The present invention relates to new compounds of formula (I) that possess agonist activity with respect to sphingosine-1-phosphate (S1P) receptors, their preparation process and their use as immunosuppressive agents. The invention also relates to pharmaceutical compositions containing these compounds and the use of these compounds for the treatment / prevention of immunologically mediated diseases and conditions and inflammatory conditions or diseases.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07290748A EP2014653A1 (en) | 2007-06-15 | 2007-06-15 | Novel dicarboxylic acid derivatives as S1P1 receptor agonists |
| EP08057571 | 2008-06-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP099805A true ECSP099805A (en) | 2010-04-30 |
Family
ID=42261381
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP099805 ECSP099805A (en) | 2007-06-15 | 2009-12-15 | NEW DERIVATIVES OF DICARBOXYL ACID AS AGONISTS OF S1P1 RECEPTORS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP099805A (en) |
-
2009
- 2009-12-15 EC ECSP099805 patent/ECSP099805A/en unknown
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