ECSP10010152A - Uso de un gestágeno en combinación con un estrógeno y uno o varios excipientes/portadores farmacéuticamente aceptables para la anticoncepción oral sin lactosa - Google Patents
Uso de un gestágeno en combinación con un estrógeno y uno o varios excipientes/portadores farmacéuticamente aceptables para la anticoncepción oral sin lactosaInfo
- Publication number
- ECSP10010152A ECSP10010152A EC2010010152A ECSP10010152A ECSP10010152A EC SP10010152 A ECSP10010152 A EC SP10010152A EC 2010010152 A EC2010010152 A EC 2010010152A EC SP10010152 A ECSP10010152 A EC SP10010152A EC SP10010152 A ECSP10010152 A EC SP10010152A
- Authority
- EC
- Ecuador
- Prior art keywords
- pharmaceutically acceptable
- combination
- oract
- strategen
- gestagen
- Prior art date
Links
- 239000003937 drug carrier Substances 0.000 title abstract 2
- 239000000546 pharmaceutical excipient Substances 0.000 title abstract 2
- 239000000583 progesterone congener Substances 0.000 title abstract 2
- VOXZDWNPVJITMN-ZBRFXRBCSA-N 17β-estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 VOXZDWNPVJITMN-ZBRFXRBCSA-N 0.000 abstract 2
- 208000002705 Glucose Intolerance Diseases 0.000 abstract 2
- 206010018429 Glucose tolerance impaired Diseases 0.000 abstract 2
- BFPYWIDHMRZLRN-UHFFFAOYSA-N 17alpha-ethynyl estradiol Natural products OC1=CC=C2C3CCC(C)(C(CC4)(O)C#C)C4C3CCC2=C1 BFPYWIDHMRZLRN-UHFFFAOYSA-N 0.000 abstract 1
- QMBJSIBWORFWQT-DFXBJWIESA-N Chlormadinone acetate Chemical compound C1=C(Cl)C2=CC(=O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@@](C(C)=O)(OC(=O)C)[C@@]1(C)CC2 QMBJSIBWORFWQT-DFXBJWIESA-N 0.000 abstract 1
- RSEPBGGWRJCQGY-RBRWEJTLSA-N Estradiol valerate Chemical compound C1CC2=CC(O)=CC=C2[C@@H]2[C@@H]1[C@@H]1CC[C@H](OC(=O)CCCC)[C@@]1(C)CC2 RSEPBGGWRJCQGY-RBRWEJTLSA-N 0.000 abstract 1
- BFPYWIDHMRZLRN-SLHNCBLASA-N Ethinyl estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 BFPYWIDHMRZLRN-SLHNCBLASA-N 0.000 abstract 1
- GUBGYTABKSRVRQ-QKKXKWKRSA-N Lactose Natural products OC[C@H]1O[C@@H](O[C@H]2[C@H](O)[C@@H](O)C(O)O[C@@H]2CO)[C@H](O)[C@@H](O)[C@H]1O GUBGYTABKSRVRQ-QKKXKWKRSA-N 0.000 abstract 1
- 229960001616 chlormadinone acetate Drugs 0.000 abstract 1
- 229960003309 dienogest Drugs 0.000 abstract 1
- AZFLJNIPTRTECV-FUMNGEBKSA-N dienogest Chemical compound C1CC(=O)C=C2CC[C@@H]([C@H]3[C@@](C)([C@](CC3)(O)CC#N)CC3)C3=C21 AZFLJNIPTRTECV-FUMNGEBKSA-N 0.000 abstract 1
- 229960005309 estradiol Drugs 0.000 abstract 1
- 229960004766 estradiol valerate Drugs 0.000 abstract 1
- 239000000262 estrogen Substances 0.000 abstract 1
- 229940011871 estrogen Drugs 0.000 abstract 1
- 229960002568 ethinylestradiol Drugs 0.000 abstract 1
- 239000008101 lactose Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 230000002035 prolonged effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/14—Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Endocrinology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Reproductive Health (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
Abstract
. Los gestágenos, con preferencia dienogest, acetato de clormadinona o levornogetrel en combinación con estrógenos tales como, por ejemplo, etinilestradiol, 17ß-estradiol o valerato de estradiol y uno o varios excipientes/portadores farmacéuticamente aceptables realizan una anticoncepción oral sin lactosa. Se da una posibilidad para mejorar la prevención de la intolerancia a la glucosa en un factor que eventualmente contribuye con la mejoría, incluso en cuanto a costosos ensayos de la intolerancia a la glucosa. La invención también es apropiada para un uso prolongado.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07021465A EP2055306A1 (de) | 2007-11-05 | 2007-11-05 | Verwendung eines Gestagens in Kombination mit einem Estrogen und einem oder mehreren pharmazeutisch annehmbaren hilfsstoffen/Trägern zur laktosefreien oralen Kontrazeption |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP10010152A true ECSP10010152A (es) | 2010-06-29 |
Family
ID=39016019
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2010010152A ECSP10010152A (es) | 2007-11-05 | 2010-05-05 | Uso de un gestágeno en combinación con un estrógeno y uno o varios excipientes/portadores farmacéuticamente aceptables para la anticoncepción oral sin lactosa |
Country Status (30)
| Country | Link |
|---|---|
| EP (3) | EP2055306A1 (es) |
| JP (1) | JP2011502136A (es) |
| KR (1) | KR20100103794A (es) |
| CN (1) | CN101848716B (es) |
| AR (1) | AR069195A1 (es) |
| AT (1) | AT12800U1 (es) |
| AU (1) | AU2008324549A1 (es) |
| BR (1) | BRPI0819189A2 (es) |
| CA (1) | CA2704523A1 (es) |
| CO (1) | CO6270329A2 (es) |
| CR (1) | CR11413A (es) |
| DE (1) | DE202007019049U1 (es) |
| DK (1) | DK2217243T3 (es) |
| DO (1) | DOP2010000130A (es) |
| EA (1) | EA201000749A1 (es) |
| EC (1) | ECSP10010152A (es) |
| ES (1) | ES2511841T3 (es) |
| HR (1) | HRP20140962T1 (es) |
| IL (1) | IL205349A0 (es) |
| MX (1) | MX2010004975A (es) |
| NZ (1) | NZ585065A (es) |
| PA (1) | PA8803001A1 (es) |
| PE (1) | PE20091020A1 (es) |
| PL (1) | PL2217243T3 (es) |
| PT (1) | PT2217243E (es) |
| SG (1) | SG188118A1 (es) |
| TW (1) | TW200936142A (es) |
| UY (1) | UY31454A1 (es) |
| WO (1) | WO2009059690A1 (es) |
| ZA (1) | ZA201004024B (es) |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0368373A1 (en) * | 1988-10-13 | 1990-05-16 | Akzo Nobel N.V. | Multi-phase contraceptive preparation |
| US5223268A (en) * | 1991-05-16 | 1993-06-29 | Sterling Drug, Inc. | Low solubility drug-coated bead compositions |
| DK95093D0 (da) * | 1993-08-20 | 1993-08-20 | Novo Nordisk As | Farmaceutisk formulering indeholdende et hormon |
| US5898032A (en) * | 1997-06-23 | 1999-04-27 | Medical College Of Hampton Roads | Ultra low dose oral contraceptives with less menstrual bleeding and sustained efficacy |
| JPH1171268A (ja) * | 1997-08-28 | 1999-03-16 | Kayaku:Kk | 性ホルモン含有錠剤 |
| CA2260673A1 (en) | 1999-02-04 | 2000-08-04 | Natrel Inc. | A process for making a lactose-free milk without negatively affecting the organoleptic properties thereof; and milk so processed |
| DE10043846A1 (de) * | 2000-09-04 | 2002-04-04 | Jenapharm Gmbh | 17-Methylensteroide, Verfahren zu deren Herstellung und diese Verbindung enthaltende pharmazeutische Zusammensetzungen |
| FR2832065B1 (fr) * | 2001-11-13 | 2004-11-05 | Besins Int Belgique | Composition pharmaceutique a base de progesterone micronisee son procede de preparation et ses utilisations |
| WO2005030176A1 (en) | 2003-09-29 | 2005-04-07 | Novo Nordisk Femcare Ag | Improved stability of progestogen formulations |
| WO2005030175A1 (en) | 2003-09-29 | 2005-04-07 | Novo Nordisk Femcare Ag | Hrt formulations |
| CN1672685A (zh) * | 2004-03-26 | 2005-09-28 | 董可娟 | 一种新的避孕药物 |
| DE102004019406A1 (de) * | 2004-04-19 | 2005-11-03 | Schering Ag | 17α-Fluorsteroide |
| DE102004026670A1 (de) * | 2004-05-28 | 2005-12-15 | Grünenthal GmbH | Hormonales Kontrazeptivum enthaltend eine Kombination aus Ethinylestradiol und Chlormadinonacetat |
| DE102004026671A1 (de) * | 2004-05-28 | 2005-12-15 | Grünenthal GmbH | Darreichungsform zur hormonalen Kontrazeption |
| EP1690543A1 (de) * | 2005-02-15 | 2006-08-16 | Schering AG | Pharmazeutisches Präparat zur Kontrazeption |
| EP1774970A1 (de) * | 2005-10-13 | 2007-04-18 | Bayer Schering Pharma AG | Verfahren zur Herstellung eines einphasigen pharmazeutischen Präparates zur Therapie der dysfunktionellen uterinen Blutung, enthaltend Ethinylestradiol und Dienogest |
-
2007
- 2007-11-05 AT ATGM371/2010U patent/AT12800U1/de not_active IP Right Cessation
- 2007-11-05 DE DE202007019049U patent/DE202007019049U1/de not_active Expired - Lifetime
- 2007-11-05 EP EP07021465A patent/EP2055306A1/de not_active Withdrawn
-
2008
- 2008-10-22 EP EP14164080.5A patent/EP2774614A1/de not_active Withdrawn
- 2008-10-22 CA CA2704523A patent/CA2704523A1/en not_active Abandoned
- 2008-10-22 CN CN2008801148441A patent/CN101848716B/zh not_active Expired - Fee Related
- 2008-10-22 SG SG2013008883A patent/SG188118A1/en unknown
- 2008-10-22 MX MX2010004975A patent/MX2010004975A/es not_active Application Discontinuation
- 2008-10-22 KR KR1020107012376A patent/KR20100103794A/ko not_active Ceased
- 2008-10-22 ES ES08847408.5T patent/ES2511841T3/es active Active
- 2008-10-22 BR BRPI0819189-1A patent/BRPI0819189A2/pt not_active IP Right Cessation
- 2008-10-22 DK DK08847408.5T patent/DK2217243T3/da active
- 2008-10-22 EP EP08847408.5A patent/EP2217243B1/de active Active
- 2008-10-22 HR HRP20140962AT patent/HRP20140962T1/hr unknown
- 2008-10-22 NZ NZ585065A patent/NZ585065A/en not_active IP Right Cessation
- 2008-10-22 WO PCT/EP2008/008900 patent/WO2009059690A1/de not_active Ceased
- 2008-10-22 PL PL08847408T patent/PL2217243T3/pl unknown
- 2008-10-22 JP JP2010531446A patent/JP2011502136A/ja not_active Ceased
- 2008-10-22 EA EA201000749A patent/EA201000749A1/ru unknown
- 2008-10-22 AU AU2008324549A patent/AU2008324549A1/en not_active Abandoned
- 2008-10-22 PT PT88474085T patent/PT2217243E/pt unknown
- 2008-11-04 PE PE2008001887A patent/PE20091020A1/es not_active Application Discontinuation
- 2008-11-04 UY UY31454A patent/UY31454A1/es unknown
- 2008-11-05 AR ARP080104837A patent/AR069195A1/es unknown
- 2008-11-05 TW TW097142714A patent/TW200936142A/zh unknown
- 2008-11-06 PA PA20088803001A patent/PA8803001A1/es unknown
-
2010
- 2010-04-26 IL IL205349A patent/IL205349A0/en unknown
- 2010-05-05 DO DO2010000130A patent/DOP2010000130A/es unknown
- 2010-05-05 CR CR11413A patent/CR11413A/es not_active Application Discontinuation
- 2010-05-05 EC EC2010010152A patent/ECSP10010152A/es unknown
- 2010-05-05 CO CO10053517A patent/CO6270329A2/es not_active Application Discontinuation
- 2010-06-04 ZA ZA2010/04024A patent/ZA201004024B/en unknown
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