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Priority to ECSP10010663priorityCriticalpatent/ECSP10010663A/en
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Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Nitrogen Condensed Heterocyclic Rings
(AREA)
Abstract
Se describen nuevos compuestos de [1.2.4]triazol[1,5-a]pirazina e imidazo[1,2-a]pirazina que poseen una formula representada por las siguientes: Fórmula (Ia) o Fórmula (Ib)- Los compuestos se pueden preparar como composiciones farmacéuticas, y se pueden utilizar para la prevención y el tratamiento de una variedad de afecciones en mamíferos incluyendo los seres humanos, que incluye a modo de ejemplo no limitativo, dolor, inflamación, y otros.New compounds of [1.2.4] triazol [1,5-a] pyrazine and imidazo [1,2-a] pyrazine are described which have a formula represented by the following: Formula (Ia) or Formula (Ib) - The compounds they can be prepared as pharmaceutical compositions, and can be used for the prevention and treatment of a variety of conditions in mammals including humans, which includes by way of non-limiting example, pain, inflammation, and others.
ECSP100106632010-12-072010-12-07
USEFUL FUSIONED PIRAZINE COMPOUNDS FOR THE TREATMENT OF DEGENARATIVE AND INFLAMMATORY DISEASES
ECSP10010663A
(en)
2-Fluoro-N-Methyl-4- [7- (Quinolin-6-yl-Methyl) -imidazo [1,2-B] [1,2,4] triazine-2-yl] benzamide salts and their procedures WITH THE PREPARATION OF THESE
DERIVATIVES OF 2,3-DIHYDROIMIDAZO [1,2-C] QUINAZOLINA SUBSTITUTED WITH AMINOALCOHOLES THAT ARE USEFUL TO TREAT HYPERPROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS
DERIVATIVES OF PIRIDIN-2 (1H) -ONE USEFUL AS MEDICINES FOR THE TREATMENT OF MYELOPROLIFERATIVE DISORDERS, REJECTION OF TRANSPLANTS, DISEASES MEDIATED BY THE IMMUNE SYSTEM AND INFLAMMATORY DISEASES.
Compounds derived from pyrrole [3,4-b] pyridin-5-one, inhibitors of pi3k; pharmaceutical composition comprising them; and use for the treatment of diseases such as Alzheimer's, epilepsy, multiple sclerosis, Parkinson's, among others.
6,7-dihydro-5h-imidazo [1,2-alpha] imidazole-3-carboxylic acid amide derivative compounds; pharmaceutical composition comprising them; and uses in the treatment of an inflammatory condition.
ACID DERIVATIVES OF 1,2,4-OXADIAZOL CARBOXILIC CYCLBUTHANAMINE, A PHARMACEUTICAL COMPOSITION, COMPOSITE PREPARATION PROCESS AND ITS USE TO PREPARE MEDICATIONS
1,2,3,4-TETRAHYDROPYRROLO [1,2-A] PYRAZINE-6-CARBOXAMIDES AND 2,3,4,5-TETRAHYDROPYRROLO [1,2-A] [1,4] -DIAZEPINE-7 DERIVATIVES -CARBOXAMIDES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
Compounds derived from sulfonamide, inhibitors of beta amyloid production; Preparation method; pharmaceutical composition; pharmaceutical kit; and use in the treatment of diseases such as Alzheimer's, amyloid angiopathy, down syndrome, among others.