ECSP11010801A - Derivados de pirazolo-[5,1-b]-oxazol como antagonistas de crf1 - Google Patents
Derivados de pirazolo-[5,1-b]-oxazol como antagonistas de crf1Info
- Publication number
- ECSP11010801A ECSP11010801A EC2011010801A ECSP11010801A ECSP11010801A EC SP11010801 A ECSP11010801 A EC SP11010801A EC 2011010801 A EC2011010801 A EC 2011010801A EC SP11010801 A ECSP11010801 A EC SP11010801A EC SP11010801 A ECSP11010801 A EC SP11010801A
- Authority
- EC
- Ecuador
- Prior art keywords
- crf1
- derivatives
- antigonist
- pirazolo
- oxazol
- Prior art date
Links
- 102100038018 Corticotropin-releasing factor receptor 1 Human genes 0.000 title 1
- 101000878678 Homo sapiens Corticotropin-releasing factor receptor 1 Proteins 0.000 title 1
- 101000948733 Saccharomyces cerevisiae (strain ATCC 204508 / S288c) Probable phospholipid translocase non-catalytic subunit CRF1 Proteins 0.000 title 1
- 102400000739 Corticotropin Human genes 0.000 abstract 1
- 101800000414 Corticotropin Proteins 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- IDLFZVILOHSSID-OVLDLUHVSA-N corticotropin Chemical compound C([C@@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC=1NC=NC=1)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](C(C)C)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC=1C=CC=CC=1)C(O)=O)NC(=O)[C@@H](N)CO)C1=CC=C(O)C=C1 IDLFZVILOHSSID-OVLDLUHVSA-N 0.000 abstract 1
- 229960000258 corticotropin Drugs 0.000 abstract 1
- BKRKYGDGROPRDS-UHFFFAOYSA-N pyrazolo[5,1-b][1,3]oxazole Chemical class O1C=CN2N=CC=C21 BKRKYGDGROPRDS-UHFFFAOYSA-N 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/424—Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Virology (AREA)
- Addiction (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Endocrinology (AREA)
- Pulmonology (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Obesity (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Urology & Nephrology (AREA)
- Molecular Biology (AREA)
- Hematology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Anesthesiology (AREA)
- Cardiology (AREA)
- AIDS & HIV (AREA)
Abstract
Se describen derivados de pirazolo-[5.1-b]-oxazol de la estructura I útiles como antagonistas del receptor del factor de liberación de corticotropina (CRF1).
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08161930 | 2008-08-06 | ||
| US20509609P | 2009-01-14 | 2009-01-14 | |
| EP09150553 | 2009-01-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP11010801A true ECSP11010801A (es) | 2011-03-31 |
Family
ID=41653505
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2011010801A ECSP11010801A (es) | 2008-08-06 | 2011-02-02 | Derivados de pirazolo-[5,1-b]-oxazol como antagonistas de crf1 |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7994203B2 (es) |
| EP (1) | EP2328902A1 (es) |
| JP (1) | JP2011529943A (es) |
| KR (1) | KR20110051226A (es) |
| CN (1) | CN102171220A (es) |
| AR (1) | AR073262A1 (es) |
| AU (1) | AU2009279137A1 (es) |
| BR (1) | BRPI0917565A2 (es) |
| CA (1) | CA2733176A1 (es) |
| CO (1) | CO6351723A2 (es) |
| EA (1) | EA201100303A1 (es) |
| EC (1) | ECSP11010801A (es) |
| IL (1) | IL211030A0 (es) |
| MA (1) | MA32537B1 (es) |
| MX (1) | MX2011001392A (es) |
| TW (1) | TW201011039A (es) |
| UY (1) | UY32029A (es) |
| WO (1) | WO2010015628A1 (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0911659B8 (pt) | 2008-04-15 | 2021-05-25 | Eisai R&D Man Co Ltd | composto 3-fenilpirazolo[5,1-b]tiazol e composição farmacêutica compreendendo o mesmo |
| US8273900B2 (en) | 2008-08-07 | 2012-09-25 | Novartis Ag | Organic compounds |
| AR078521A1 (es) | 2009-10-08 | 2011-11-16 | Eisai R&D Man Co Ltd | Compuesto pirazolotiazol |
| JPWO2011043387A1 (ja) | 2009-10-08 | 2013-03-04 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ピラゾロオキサゾール化合物 |
| CN102762572A (zh) * | 2010-02-01 | 2012-10-31 | 诺瓦提斯公司 | 作为CRF-1受体拮抗剂的吡唑并[5,1b]*唑衍生物 |
| US8546416B2 (en) | 2011-05-27 | 2013-10-01 | Novartis Ag | 3-spirocyclic piperidine derivatives as ghrelin receptor agonists |
| EP2567959B1 (en) | 2011-09-12 | 2014-04-16 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| CA2867043A1 (en) | 2012-05-03 | 2013-11-07 | Novartis Ag | L-malate salt of 2,7-diaza-spiro[4.5]dec-7-yle derivatives and crystalline forms thereof as ghrelin receptor agonists |
| RU2718918C2 (ru) | 2014-01-21 | 2020-04-15 | Ньюрокрайн Байосайенсиз, Инк. | Антагонисты рецептора cfr1 для лечения врожденной гиперплазии коры надпочечников |
| KR20200035035A (ko) | 2017-07-31 | 2020-04-01 | 노파르티스 아게 | 코카인 사용 감소 또는 코카인 사용 재발 예방에 있어서 마보글루란트의 용도 |
| BR112021010847A2 (pt) | 2018-12-07 | 2021-09-08 | Neurocrine Biosciences Inc. | Antagonista de receptor de crf1, formulações farmacêuticas e formas sólidas das mesmas para o tratamento de hiperplasia adrenal congênita |
| US12383536B2 (en) | 2019-09-27 | 2025-08-12 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods of use |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU5426296A (en) * | 1995-04-04 | 1996-10-23 | E.I. Du Pont De Nemours And Company | Herbicidal heteroaryl-substituted anilides |
| HRP20030675A2 (en) * | 2001-01-26 | 2004-08-31 | Bristol Myers Squibb Co | Imidazolyl derivatives as corticotropin relasing factor inhibitors |
-
2009
- 2009-08-03 US US12/462,417 patent/US7994203B2/en not_active Expired - Fee Related
- 2009-08-04 WO PCT/EP2009/060094 patent/WO2010015628A1/en not_active Ceased
- 2009-08-04 EA EA201100303A patent/EA201100303A1/ru unknown
- 2009-08-04 CA CA2733176A patent/CA2733176A1/en not_active Abandoned
- 2009-08-04 MX MX2011001392A patent/MX2011001392A/es not_active Application Discontinuation
- 2009-08-04 EP EP09804561A patent/EP2328902A1/en not_active Withdrawn
- 2009-08-04 AU AU2009279137A patent/AU2009279137A1/en not_active Abandoned
- 2009-08-04 UY UY0001032029A patent/UY32029A/es not_active Application Discontinuation
- 2009-08-04 CN CN2009801394474A patent/CN102171220A/zh active Pending
- 2009-08-04 KR KR1020117005158A patent/KR20110051226A/ko not_active Withdrawn
- 2009-08-04 AR ARP090102986A patent/AR073262A1/es unknown
- 2009-08-04 JP JP2011521562A patent/JP2011529943A/ja not_active Withdrawn
- 2009-08-04 BR BRPI0917565A patent/BRPI0917565A2/pt not_active Application Discontinuation
- 2009-08-05 TW TW098126427A patent/TW201011039A/zh unknown
-
2011
- 2011-02-01 CO CO11011419A patent/CO6351723A2/es not_active Application Discontinuation
- 2011-02-02 EC EC2011010801A patent/ECSP11010801A/es unknown
- 2011-02-03 IL IL211030A patent/IL211030A0/en unknown
- 2011-02-03 MA MA33581A patent/MA32537B1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL211030A0 (en) | 2011-04-28 |
| CO6351723A2 (es) | 2011-12-20 |
| UY32029A (es) | 2010-03-26 |
| TW201011039A (en) | 2010-03-16 |
| CN102171220A (zh) | 2011-08-31 |
| EA201100303A1 (ru) | 2011-10-31 |
| AU2009279137A1 (en) | 2010-02-11 |
| EP2328902A1 (en) | 2011-06-08 |
| BRPI0917565A2 (pt) | 2015-11-17 |
| JP2011529943A (ja) | 2011-12-15 |
| CA2733176A1 (en) | 2010-02-11 |
| AU2009279137A8 (en) | 2011-03-03 |
| WO2010015628A1 (en) | 2010-02-11 |
| US20100035874A1 (en) | 2010-02-11 |
| MA32537B1 (fr) | 2011-08-01 |
| US7994203B2 (en) | 2011-08-09 |
| KR20110051226A (ko) | 2011-05-17 |
| AR073262A1 (es) | 2010-10-28 |
| MX2011001392A (es) | 2011-03-25 |
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