ECSP11011535A - DERIVATIVES OF N- (HETERO) ARIL-PIRROLIDINA DE PIRAZOL-4-IL-PIRROLO [2,3-D] PIRIMIDINES AND PIRROL-3-IL-PIRROLO [2,3-D] PYRIMIDINS AS INHIBITORS OF THE JANUS KINASE - Google Patents

DERIVATIVES OF N- (HETERO) ARIL-PIRROLIDINA DE PIRAZOL-4-IL-PIRROLO [2,3-D] PIRIMIDINES AND PIRROL-3-IL-PIRROLO [2,3-D] PYRIMIDINS AS INHIBITORS OF THE JANUS KINASE

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Publication number
ECSP11011535A
ECSP11011535A ECSP11011535A ECSP11011535A EC SP11011535 A ECSP11011535 A EC SP11011535A EC SP11011535 A ECSP11011535 A EC SP11011535A EC SP11011535 A ECSP11011535 A EC SP11011535A
Authority
EC
Ecuador
Prior art keywords
pirrolo
inhibitors
hetero
derivatives
pirimidines
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Joseph Glenn
James D Rodgers
Stacey Shepard
Haisheng Wang
Argyrios G Arvanitis
Louis Storace
Wenyu Zhu
Beverly Folmer
Lixin Shao
Original Assignee
Incyte Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47780587&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP11011535(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Incyte Corp filed Critical Incyte Corp
Publication of ECSP11011535A publication Critical patent/ECSP11011535A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente invención se relaciona con derivados de N-(hetero)aril-pirrolidina de Fórmula I:que son inhibidores de JAK, tal como inhibidores selectivos de JAK1 , útiles en el tratamiento de enfermedades asociadas con JAK, entre las que se incluyen, por ejemplo, los trastornos inflamatorios y autoinmunes y también el cáncer.The present invention relates to N- (hetero) aryl-pyrrolidine derivatives of Formula I: which are JAK inhibitors, such as selective JAK1 inhibitors, useful in the treatment of diseases associated with JAK, which include, by example, inflammatory and autoimmune disorders and also cancer.

ECSP11011535 2009-05-22 2011-12-15 DERIVATIVES OF N- (HETERO) ARIL-PIRROLIDINA DE PIRAZOL-4-IL-PIRROLO [2,3-D] PIRIMIDINES AND PIRROL-3-IL-PIRROLO [2,3-D] PYRIMIDINS AS INHIBITORS OF THE JANUS KINASE ECSP11011535A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18062209P 2009-05-22 2009-05-22

Publications (1)

Publication Number Publication Date
ECSP11011535A true ECSP11011535A (en) 2012-01-31

Family

ID=47780587

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP11011535 ECSP11011535A (en) 2009-05-22 2011-12-15 DERIVATIVES OF N- (HETERO) ARIL-PIRROLIDINA DE PIRAZOL-4-IL-PIRROLO [2,3-D] PIRIMIDINES AND PIRROL-3-IL-PIRROLO [2,3-D] PYRIMIDINS AS INHIBITORS OF THE JANUS KINASE

Country Status (2)

Country Link
EC (1) ECSP11011535A (en)
UA (1) UA106617C2 (en)

Also Published As

Publication number Publication date
UA106617C2 (en) 2014-09-25

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