ECSP12011706A - PROCEDURE FOR MANUFACTURING ACID 2 - [(3,5-DIFLUORO-3'-METOXI-1,1'-BIFENIL-4-IL) AMINO] NICOTINIC - Google Patents
PROCEDURE FOR MANUFACTURING ACID 2 - [(3,5-DIFLUORO-3'-METOXI-1,1'-BIFENIL-4-IL) AMINO] NICOTINICInfo
- Publication number
- ECSP12011706A ECSP12011706A ECSP12011706A ECSP12011706A EC SP12011706 A ECSP12011706 A EC SP12011706A EC SP12011706 A ECSP12011706 A EC SP12011706A EC SP12011706 A ECSP12011706 A EC SP12011706A
- Authority
- EC
- Ecuador
- Prior art keywords
- difluoro
- amino
- nicotinic
- bifenil
- metoxi
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000002253 acid Substances 0.000 title 1
- BFAMMODYWZEGDM-UHFFFAOYSA-N 2,6-difluoro-4-(3-methoxyphenyl)aniline Chemical compound COC1=CC=CC(C=2C=C(F)C(N)=C(F)C=2)=C1 BFAMMODYWZEGDM-UHFFFAOYSA-N 0.000 abstract 3
- OMPATGZMNFWVOH-UHFFFAOYSA-N 2-[2,6-difluoro-4-(3-methoxyphenyl)anilino]pyridine-3-carboxylic acid Chemical compound COC1=CC=CC(C=2C=C(F)C(NC=3C(=CC=CN=3)C(O)=O)=C(F)C=2)=C1 OMPATGZMNFWVOH-UHFFFAOYSA-N 0.000 abstract 2
- -1 amine salt Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pyridine Compounds (AREA)
Abstract
Esta invención se refiere a un procedimiento para fabricar ácido 2-[(3,5-difluoro-3'-metoxi-1,1'-bifenil-4-il)amino]nicotínico, que comprende las etapas de:a) proporcionar 3,5-difluoro-3'-metoxibifenil-4-amina,b) proporcionar y aislar una sal de aminio de la 3,5-difluoro-3'-metoxibifenil-4-amina, yc) además hacer reaccionar la sal de aminio de 3,5-difluoro-3'-metoxibifenil-4-amina obtenida en b) para obtener ácido 2-[(3,5-difluoro-3'-metoxi-1,1'-bifenil-4-il)amino]nicotínico.This invention relates to a process for manufacturing 2 - [(3,5-difluoro-3'-methoxy-1,1'-biphenyl-4-yl) amino] nicotinic acid, comprising the steps of: a) providing 3 , 5-difluoro-3'-methoxybiphenyl-4-amine, b) provide and isolate an aminium salt of 3,5-difluoro-3'-methoxybiphenyl-4-amine, and c) further react the amine salt of 3,5-Difluoro-3'-methoxybiphenyl-4-amine obtained in b) to obtain 2 - [(3,5-difluoro-3'-methoxy-1,1'-biphenyl-4-yl) amino] nicotinic acid .
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP12011706 ECSP12011706A (en) | 2012-03-02 | 2012-03-02 | PROCEDURE FOR MANUFACTURING ACID 2 - [(3,5-DIFLUORO-3'-METOXI-1,1'-BIFENIL-4-IL) AMINO] NICOTINIC |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP12011706 ECSP12011706A (en) | 2012-03-02 | 2012-03-02 | PROCEDURE FOR MANUFACTURING ACID 2 - [(3,5-DIFLUORO-3'-METOXI-1,1'-BIFENIL-4-IL) AMINO] NICOTINIC |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP12011706A true ECSP12011706A (en) | 2012-04-30 |
Family
ID=52630131
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP12011706 ECSP12011706A (en) | 2012-03-02 | 2012-03-02 | PROCEDURE FOR MANUFACTURING ACID 2 - [(3,5-DIFLUORO-3'-METOXI-1,1'-BIFENIL-4-IL) AMINO] NICOTINIC |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP12011706A (en) |
-
2012
- 2012-03-02 EC ECSP12011706 patent/ECSP12011706A/en unknown
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