ECSP12012332A - Asociación de inhibidores de la xantina oxidasa y la instatina y su uso - Google Patents

Asociación de inhibidores de la xantina oxidasa y la instatina y su uso

Info

Publication number
ECSP12012332A
ECSP12012332A ECSP12012332A ECSP12012332A EC SP12012332 A ECSP12012332 A EC SP12012332A EC SP12012332 A ECSP12012332 A EC SP12012332A EC SP12012332 A ECSP12012332 A EC SP12012332A
Authority
EC
Ecuador
Prior art keywords
association
inhibitors
instatine
xantina
oxidase
Prior art date
Application number
Other languages
English (en)
Inventor
Sandro Giuliani
Carlo Alberto Maggi
Francesco Melani
Original Assignee
Menarini Int Operations Lu Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42753377&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP12012332(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Menarini Int Operations Lu Sa filed Critical Menarini Int Operations Lu Sa
Publication of ECSP12012332A publication Critical patent/ECSP12012332A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a la asociación de principios activos, a saber de un inhibidor de la xantina oxidasa con uno o más inhibidores de la HMG CoA reductasa, composiciones farmacéuticas que comprende dicho principio activo, para uso en el tratamiento terapéutico humano o veterinario, y métodos para su preparación.
ECSP12012332 2010-05-10 2012-12-10 Asociación de inhibidores de la xantina oxidasa y la instatina y su uso ECSP12012332A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITRM2010A000232A IT1400311B1 (it) 2010-05-10 2010-05-10 Associazione di inibitori della xantina ossidasi e antagonisti del recettore dell'angiotensina ii e loro uso.

Publications (1)

Publication Number Publication Date
ECSP12012332A true ECSP12012332A (es) 2013-02-28

Family

ID=42753377

Family Applications (2)

Application Number Title Priority Date Filing Date
ECSP12012332 ECSP12012332A (es) 2010-05-10 2012-12-10 Asociación de inhibidores de la xantina oxidasa y la instatina y su uso
ECSP12012331 ECSP12012331A (es) 2010-05-10 2012-12-10 Combinacion de inhibidores de xantina oxidasa y antagonistas del receptor de angiotensina ii y su uso

Family Applications After (1)

Application Number Title Priority Date Filing Date
ECSP12012331 ECSP12012331A (es) 2010-05-10 2012-12-10 Combinacion de inhibidores de xantina oxidasa y antagonistas del receptor de angiotensina ii y su uso

Country Status (24)

Country Link
US (1) US20130131128A1 (es)
EP (1) EP2568982B1 (es)
JP (1) JP2013526503A (es)
KR (1) KR20130101447A (es)
CN (1) CN103037861A (es)
AR (1) AR081376A1 (es)
AU (1) AU2011252151A1 (es)
BR (1) BR112012028887A2 (es)
CA (1) CA2798573A1 (es)
CL (1) CL2012003143A1 (es)
CO (1) CO6640306A2 (es)
EA (1) EA201201528A1 (es)
EC (2) ECSP12012332A (es)
IL (1) IL222927A0 (es)
IT (1) IT1400311B1 (es)
MA (1) MA34297B1 (es)
MX (1) MX2012013054A (es)
NZ (1) NZ603414A (es)
PE (1) PE20130812A1 (es)
PH (1) PH12012502198A1 (es)
SG (1) SG185474A1 (es)
TW (1) TW201206432A (es)
WO (1) WO2011141431A1 (es)
ZA (1) ZA201209295B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR3028371B1 (fr) * 2014-11-06 2016-11-18 Bull Sas Procede de surveillance et de controle deportes d'un cluster utilisant un reseau de communication de type infiniband et programme d'ordinateur mettant en oeuvre ce procede
JP2018135278A (ja) * 2017-02-20 2018-08-30 株式会社スタージェン 循環器疾患及び/又はミトコンドリア病の改善用医薬
KR102284764B1 (ko) 2020-07-08 2021-08-04 주식회사 우드메탈 멀티빔구조를 통한 부속의 결속이 용이한 칸막이

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE122008000051I1 (de) 1990-11-30 2009-02-05 Teijin Ltd 2-arylthiazolderivat sowie dieses enthaltendes arzneimittel
CA2229000C (en) 1991-02-21 2002-04-09 Sankyo Company, Limited 1-biphenylimidazole derivatives, their preparation and their therapeutic use
SK287928B6 (sk) 1998-06-19 2012-04-03 Teijin Pharma Limited Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4- methyl-5-thiazole-carboxylic acid and processes for the preparation thereof
PT1336407E (pt) 2000-11-21 2006-07-31 Sankyo Co Composicao contendo um antagonista do receptor de angiotensina e um diuretico e sua utilizacao para o tratamento da hipertensao
US20040122067A1 (en) 2002-12-20 2004-06-24 Lin Zhao Treatment of chronic heart failure
RS20050590A (sr) 2003-01-31 2007-09-21 Sankyo Company Limited, Lek za profilaksu i tretman arterioskleroze i hipertenzije
WO2005027887A2 (en) * 2003-09-17 2005-03-31 Cardimone Pharma Corporation Methods and compositions for improving endothelial function
JP5242393B2 (ja) * 2005-08-03 2013-07-24 タケダ ファーマシューティカルズ ユー.エス.エー. インコーポレイティド 高血圧症の治療方法
EP1957064A4 (en) 2005-11-21 2010-01-06 Tap Pharmaceutical Prod Inc TREATMENT OF QT INTERVAL EXTENSION AND RELEVANT DISEASES
EP2101761A4 (en) 2006-11-13 2010-01-27 Takeda Pharmaceuticals North A METHODS FOR PRESERVING RENAL FUNCTION USING XANTHINE OXYDOREDUCTASE INHIBITORS

Also Published As

Publication number Publication date
ZA201209295B (en) 2013-08-28
JP2013526503A (ja) 2013-06-24
KR20130101447A (ko) 2013-09-13
WO2011141431A1 (en) 2011-11-17
ECSP12012331A (es) 2013-02-28
NZ603414A (en) 2014-03-28
EP2568982A1 (en) 2013-03-20
IL222927A0 (en) 2012-12-31
MX2012013054A (es) 2013-03-05
BR112012028887A2 (pt) 2016-07-26
CA2798573A1 (en) 2011-11-17
AU2011252151A1 (en) 2012-11-29
CO6640306A2 (es) 2013-03-22
CL2012003143A1 (es) 2013-06-21
ITRM20100232A1 (it) 2011-11-11
EP2568982B1 (en) 2014-04-02
AR081376A1 (es) 2012-08-29
TW201206432A (en) 2012-02-16
SG185474A1 (en) 2012-12-28
CN103037861A (zh) 2013-04-10
PE20130812A1 (es) 2013-08-08
PH12012502198A1 (en) 2013-02-25
IT1400311B1 (it) 2013-05-24
EA201201528A1 (ru) 2013-04-30
US20130131128A1 (en) 2013-05-23
MA34297B1 (fr) 2013-06-01

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