ECSP13012394A - Nuevas formas de dosificación de liberación modificada de un inhibidor de la xantina oxidorreductasa o de inhibidores de xantina oxidasa - Google Patents

Nuevas formas de dosificación de liberación modificada de un inhibidor de la xantina oxidorreductasa o de inhibidores de xantina oxidasa

Info

Publication number
ECSP13012394A
ECSP13012394A ECSP13012394A ECSP13012394A EC SP13012394 A ECSP13012394 A EC SP13012394A EC SP13012394 A ECSP13012394 A EC SP13012394A EC SP13012394 A ECSP13012394 A EC SP13012394A
Authority
EC
Ecuador
Prior art keywords
xantina
inhibitors
oxidorreductasa
oxidasa
inhibitor
Prior art date
Application number
Other languages
English (en)
Inventor
Rajneesh Taneja
Vijay Gupte
Majid Vakilynejad
Original Assignee
Takeda Pharmaceuticals Usa Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45328897&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP13012394(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceuticals Usa Inc filed Critical Takeda Pharmaceuticals Usa Inc
Publication of ECSP13012394A publication Critical patent/ECSP13012394A/es

Links

Classifications

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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
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    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
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    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Reproductive Health (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Nuevas formas de dosificación de inhibidores de la xantina oxidorreductasa.
ECSP13012394 2010-06-16 2013-01-16 Nuevas formas de dosificación de liberación modificada de un inhibidor de la xantina oxidorreductasa o de inhibidores de xantina oxidasa ECSP13012394A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US35516410P 2010-06-16 2010-06-16

Publications (1)

Publication Number Publication Date
ECSP13012394A true ECSP13012394A (es) 2013-04-30

Family

ID=45328897

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP13012394 ECSP13012394A (es) 2010-06-16 2013-01-16 Nuevas formas de dosificación de liberación modificada de un inhibidor de la xantina oxidorreductasa o de inhibidores de xantina oxidasa

Country Status (25)

Country Link
US (2) US9248119B2 (es)
EP (1) EP2582812B1 (es)
JP (2) JP5865904B2 (es)
KR (1) KR101872189B1 (es)
CN (1) CN103210084B (es)
AU (2) AU2011268445B2 (es)
BR (1) BR112012032033A2 (es)
CA (1) CA2801930A1 (es)
CL (1) CL2012003548A1 (es)
CO (1) CO6650415A2 (es)
EC (1) ECSP13012394A (es)
ES (1) ES2669184T3 (es)
IL (2) IL223455B (es)
JO (1) JO3450B1 (es)
MX (2) MX361138B (es)
MY (1) MY167126A (es)
NZ (1) NZ604646A (es)
PE (2) PE20130574A1 (es)
PH (1) PH12012502485A1 (es)
RU (1) RU2602188C2 (es)
SG (1) SG186301A1 (es)
TW (1) TW201202249A (es)
UA (1) UA112632C2 (es)
WO (1) WO2011159745A1 (es)
ZA (1) ZA201209386B (es)

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US8968779B2 (en) * 2010-06-16 2015-03-03 Teijin Pharma Limited Controlled release coat-core tablet
PH12012502487A1 (en) * 2010-06-25 2017-08-09 Teijin Pharma Ltd Sustained-release therapeutic agent for hypertension and renal dysfunction
NZ605562A (en) * 2010-07-09 2013-11-29 Teijin Pharma Ltd Deuterated benzylbenzene derivatives and methods of use
WO2012153313A1 (en) * 2011-05-11 2012-11-15 Ranbaxy Laboratories Limited Pharmaceutical composition of febuxostat
WO2012172461A1 (en) * 2011-06-13 2012-12-20 Ranbaxy Laboratories Limited Pharmaceutical compositions of febuxostat
CA2862602A1 (en) * 2012-01-27 2013-08-01 Teijin Pharma Limited Therapeutic agent for diabetes
WO2014009817A1 (en) * 2012-07-12 2014-01-16 Alembic Pharmaceuticals Limited Pharmaceutical composition of febuxostat
CN102973530B (zh) * 2012-12-14 2016-08-03 贵州信邦制药股份有限公司 一种非布索坦双层肠溶片剂及其制备方法
WO2014125504A2 (en) * 2013-02-18 2014-08-21 Hetero Research Foundation Pharmaceutical compositions of febuxostat
US20140357683A1 (en) * 2013-05-31 2014-12-04 Takeda Pharmaceuticals U.S.A., Inc. Methods of treatment and compositions with xanthine oxidase inhibitors
EP2881116A1 (en) * 2013-12-05 2015-06-10 Ranbaxy Laboratories Limited Febuxostat composition
JP2018513203A (ja) * 2015-04-20 2018-05-24 ティダブリューアイ・バイオテクノロジー・インコーポレイテッドＴＷＩ Ｂｉｏｔｅｃｈｎｏｌｏｇｙ， Ｉｎｃ． ジアセレインを含有する製剤及びそれを用いて尿酸の血中濃度を低下させる方法
TWI684465B (zh) * 2015-04-22 2020-02-11 安成生物科技股份有限公司 含雙醋瑞因之製劑及使用其於降低尿酸血中濃度的方法
US20180344749A1 (en) * 2015-12-10 2018-12-06 Cogwellin, LLC Controlled release formulations of saliclate-releasing actives
CN106279024B (zh) * 2016-07-19 2018-09-14 华南理工大学 一种黄嘌呤氧化还原酶抑制剂及其制备方法与应用
CN106146419A (zh) * 2016-08-01 2016-11-23 沈阳药科大学 黄嘌呤氧化酶抑制剂
AU2017364804A1 (en) * 2016-11-28 2019-05-02 Teijin Pharma Limited Therapeutic drug or prophylactic drug for diabetic nephropathy
WO2018228440A1 (zh) * 2017-06-14 2018-12-20 江苏恒瑞医药股份有限公司 一种非布司他控释组合物及其制备方法
CN109721586B (zh) * 2017-10-27 2021-03-02 中国医科大学 一种5-苄基-3-吡啶基-1h-1,2,4-三唑类化合物及其制备方法和用途
CN108484494B (zh) * 2018-06-15 2021-07-30 沈阳药科大学 2-氧代-1,2-二氢吡啶-4-甲酸类化合物
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