ECSP14013328A - Preparacion de liberacion sostenida - Google Patents

Preparacion de liberacion sostenida

Info

Publication number
ECSP14013328A
ECSP14013328A ECSP14013328A ECSP14013328A EC SP14013328 A ECSP14013328 A EC SP14013328A EC SP14013328 A ECSP14013328 A EC SP14013328A EC SP14013328 A ECSP14013328 A EC SP14013328A
Authority
EC
Ecuador
Prior art keywords
sustained release
release preparation
pioglitazone
salt
hours
Prior art date
Application number
Other languages
English (en)
Inventor
Yutaka Tanoue
Yusuke Murakawa
Yumiki Ishii
Kaoru Takenaka
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47178262&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP14013328(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of ECSP14013328A publication Critical patent/ECSP14013328A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se proporciona una preparación de liberación sostenida que contiene pioglitazona o una sal de esta como un ingrediente activo y que muestra superior sostenibilidad. Una preparación de liberación sostenida que contiene pioglitazona o una sal de esta, que muestra una relación de disolución de pioglitazona de 25-58% promedio en el punto de tiempo de 2 horas, y 60-100% de promedio en el punto de tiempo de 4 horas, en una prueba de disolución de acuerdo con el método de paletas USP de 50 rpm y usando buffer de KCl/HCl pH 2,0 a 37 C como una solución de ensayo.
ECSP14013328 2011-10-21 2014-04-29 Preparacion de liberacion sostenida ECSP14013328A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2011232302 2011-10-21

Publications (1)

Publication Number Publication Date
ECSP14013328A true ECSP14013328A (es) 2014-05-31

Family

ID=47178262

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP14013328 ECSP14013328A (es) 2011-10-21 2014-04-29 Preparacion de liberacion sostenida

Country Status (30)

Country Link
US (1) US9907789B2 (es)
EP (1) EP2768487B1 (es)
JP (1) JP6093762B2 (es)
KR (1) KR20140081826A (es)
CN (1) CN104039313A (es)
AP (1) AP2014007645A0 (es)
AR (1) AR088398A1 (es)
AU (1) AU2012326976B2 (es)
BR (1) BR112014008744A2 (es)
CA (1) CA2852417A1 (es)
CL (1) CL2014000992A1 (es)
CO (1) CO6960544A2 (es)
CR (1) CR20140213A (es)
DO (1) DOP2014000077A (es)
EA (1) EA201490840A1 (es)
EC (1) ECSP14013328A (es)
IL (1) IL232114A0 (es)
IN (1) IN2014DN03169A (es)
MA (1) MA35717B1 (es)
MX (1) MX2014004679A (es)
NZ (1) NZ624275A (es)
PE (1) PE20141189A1 (es)
PH (1) PH12014500856A1 (es)
SG (2) SG2014012025A (es)
TN (1) TN2014000152A1 (es)
TW (1) TW201323018A (es)
UA (1) UA113858C2 (es)
UY (1) UY34403A (es)
WO (1) WO2013058409A1 (es)
ZA (1) ZA201403103B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20141189A1 (es) 2011-10-21 2014-09-24 Takeda Pharmaceutical Preparacion de liberacion sostenida
CN105121418A (zh) 2012-04-20 2015-12-02 吉利德科学公司 苯并噻唑-6-基乙酸衍生物及其治疗hiv感染的用途
US20150141517A1 (en) 2013-11-15 2015-05-21 Shin-Etsu Chemical Co., Ltd. Granulated composite, rapid release tablet and method for producing same
KR102485766B1 (ko) 2019-12-11 2023-01-09 한국유나이티드제약 주식회사 생체이용률이 향상된 피오글리타존 함유 약학조성물
UY39094A (es) * 2020-02-27 2021-07-30 Hk Inno N Corp Composición farmacéutica que comprende compuesto derivado de bencimidazol
JP2023066053A (ja) * 2021-10-28 2023-05-15 東和薬品株式会社 放出制御医薬組成物
WO2025064867A1 (en) * 2023-09-21 2025-03-27 Yuva Biosciences, Inc. Delivery system for mitochondrial health enhancers

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JPH0624991A (ja) 1991-06-20 1994-02-01 Tokyo Tanabe Co Ltd ウルソデスオキシコール酸持続性製剤
JPH0624959A (ja) 1991-10-04 1994-02-01 Bayer Yakuhin Kk 胃内浮遊型薬物徐放性固形製剤
JP3140465B2 (ja) 1992-09-18 2001-03-05 山之内製薬株式会社 ハイドロゲル徐放性製剤
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Also Published As

Publication number Publication date
ZA201403103B (en) 2015-08-26
US20140248362A1 (en) 2014-09-04
IN2014DN03169A (es) 2015-05-22
JP6093762B2 (ja) 2017-03-08
IL232114A0 (en) 2014-06-30
EP2768487B1 (en) 2020-06-03
AU2012326976A2 (en) 2014-06-12
AP2014007645A0 (en) 2014-05-31
MX2014004679A (es) 2014-08-01
SG10201700121YA (en) 2017-03-30
WO2013058409A1 (en) 2013-04-25
CA2852417A1 (en) 2013-04-25
CO6960544A2 (es) 2014-05-30
US9907789B2 (en) 2018-03-06
PE20141189A1 (es) 2014-09-24
AU2012326976A1 (en) 2014-05-29
UY34403A (es) 2013-05-31
DOP2014000077A (es) 2014-07-15
EA201490840A1 (ru) 2014-08-29
TN2014000152A1 (en) 2015-09-30
CR20140213A (es) 2014-06-18
AR088398A1 (es) 2014-05-28
CL2014000992A1 (es) 2014-09-05
NZ624275A (en) 2016-09-30
MA35717B1 (fr) 2014-12-01
JP2014530802A (ja) 2014-11-20
TW201323018A (zh) 2013-06-16
KR20140081826A (ko) 2014-07-01
BR112014008744A2 (pt) 2017-04-18
UA113858C2 (uk) 2017-03-27
AU2012326976B2 (en) 2017-08-17
CN104039313A (zh) 2014-09-10
EP2768487A1 (en) 2014-08-27
PH12014500856A1 (en) 2014-05-19
SG2014012025A (en) 2014-06-27

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