ECSP15021681A - FUSED TRICYCLIC DERIVATIVES OF THIOPHENE AS JAK INHIBITORS - Google Patents

FUSED TRICYCLIC DERIVATIVES OF THIOPHENE AS JAK INHIBITORS

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Publication number
ECSP15021681A
ECSP15021681A ECIEPI201521681A ECPI201521681A ECSP15021681A EC SP15021681 A ECSP15021681 A EC SP15021681A EC IEPI201521681 A ECIEPI201521681 A EC IEPI201521681A EC PI201521681 A ECPI201521681 A EC PI201521681A EC SP15021681 A ECSP15021681 A EC SP15021681A
Authority
EC
Ecuador
Prior art keywords
thiophene
fused tricyclic
tricyclic derivatives
jak inhibitors
jak
Prior art date
Application number
ECIEPI201521681A
Other languages
Spanish (es)
Inventor
Wenyu Zhu
Joseph Glenn
Yun-Long Li
Song Mei
Original Assignee
Howe Arlene R
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Howe Arlene R filed Critical Howe Arlene R
Publication of ECSP15021681A publication Critical patent/ECSP15021681A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención proporciona derivados tricíclicos fusionados de tiofeno, así como sus composiciones y métodos para su utilización, que modulan la actividad de la cinasa Janus (JAK) y que son útiles para el tratamiento de enfermedades relacionadas con la actividad de JAK incluyendo, por ejemplo, trastornos inflamatorios, trastornos autoinmunitarios, cáncer y otras enfermedades.The present invention provides fused tricyclic derivatives of thiophene, as well as their compositions and methods for their use, which modulate Janus kinase (JAK) activity and which are useful for the treatment of diseases related to JAK activity including, for example , inflammatory disorders, autoimmune disorders, cancer and other diseases.

ECIEPI201521681A 2012-11-01 2015-06-01 FUSED TRICYCLIC DERIVATIVES OF THIOPHENE AS JAK INHIBITORS ECSP15021681A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261721308P 2012-11-01 2012-11-01

Publications (1)

Publication Number Publication Date
ECSP15021681A true ECSP15021681A (en) 2017-05-31

Family

ID=73015675

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201521681A ECSP15021681A (en) 2012-11-01 2015-06-01 FUSED TRICYCLIC DERIVATIVES OF THIOPHENE AS JAK INHIBITORS

Country Status (1)

Country Link
EC (1) ECSP15021681A (en)

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