ECSP15031293A - THERAPEUTICALLY ACTIVE PYRAZOLO-PYRIMIDINE DERIVATIVES - Google Patents

THERAPEUTICALLY ACTIVE PYRAZOLO-PYRIMIDINE DERIVATIVES

Info

Publication number
ECSP15031293A
ECSP15031293A ECIEPI201531293A ECPI201531293A ECSP15031293A EC SP15031293 A ECSP15031293 A EC SP15031293A EC IEPI201531293 A ECIEPI201531293 A EC IEPI201531293A EC PI201531293 A ECPI201531293 A EC PI201531293A EC SP15031293 A ECSP15031293 A EC SP15031293A
Authority
EC
Ecuador
Prior art keywords
pyrimidine derivatives
therapeutically active
pyrazolo
active pyrazolo
oncological
Prior art date
Application number
ECIEPI201531293A
Other languages
Spanish (es)
Inventor
Qiuya Huang
Richard Jeremy Franklin
Bart Vanderhoydonck
Daniel James Ford
James Thomas Reuberson
Helen Tracey Horsley
Anant Ramrao Ghawalkar
Original Assignee
Katholieke Univ Leuven K U Leuven R D
Ucb Biopharma Sprl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Katholieke Univ Leuven K U Leuven R D, Ucb Biopharma Sprl filed Critical Katholieke Univ Leuven K U Leuven R D
Publication of ECSP15031293A publication Critical patent/ECSP15031293A/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Una serie de derivados de pirazolo[3,4-d]pirimidina que se sustituyen en la posición 4 mediante un resto monocíclico diaza, bicíclico con puente o espirocíclico, son beneficiosos en el tratamiento y/o prevención de varias dolencias humanas, incluidos trastornos inflamatorios, autoinmunes y oncológicos; enfermedades virales y malaria; y rechazo de trasplante de órganos y células.A series of pyrazolo [3,4-d] pyrimidine derivatives that are substituted at the 4-position by a diaza monocyclic, bridged bicyclic, or spirocyclic moiety, are beneficial in the treatment and / or prevention of various human ailments, including inflammatory disorders. , autoimmune and oncological; viral diseases and malaria; and organ and cell transplant rejection.

ECIEPI201531293A 2012-12-20 2015-07-20 THERAPEUTICALLY ACTIVE PYRAZOLO-PYRIMIDINE DERIVATIVES ECSP15031293A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB1223021.5A GB201223021D0 (en) 2012-12-20 2012-12-20 Therapeutic agents

Publications (1)

Publication Number Publication Date
ECSP15031293A true ECSP15031293A (en) 2018-07-31

Family

ID=47682284

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201531293A ECSP15031293A (en) 2012-12-20 2015-07-20 THERAPEUTICALLY ACTIVE PYRAZOLO-PYRIMIDINE DERIVATIVES

Country Status (4)

Country Link
EC (1) ECSP15031293A (en)
GB (1) GB201223021D0 (en)
GT (1) GT201500169A (en)
MA (1) MA38279B1 (en)

Also Published As

Publication number Publication date
GB201223021D0 (en) 2013-02-06
GT201500169A (en) 2019-08-30
MA38279A1 (en) 2018-02-28
MA38279B1 (en) 2018-10-31

Similar Documents

Publication Publication Date Title
MX376436B (en) THERAPEUTICLY ACTIVE PYRAZOLO-PYRIMIDINE DERIVATIVES.
WO2013024291A3 (en) Therapeutically active fused pyrimidine derivatives
UY36171A (en) BICYCLIC HETEROAROMATIC DERIVATIVES FUSED AS QUINASE INHIBITORS
AR093490A1 (en) DOSAGE FORMS OF SUSTAINED LIBERATION RUXOLITINIB
BR112016011484A2 (en) IMIDAZOPYRIMIDINE DERIVATIVES AS MODULATORS OF TNF ACTIVITY
CY1119840T1 (en) CYCLICALLY SUBSTITUTED SOURCES AND USE OF THESE
MX2019003649A (en) NOVELTY JAK1 SELECTIVE INHIBITORS AND USES OF THEM.
BR112018006135A2 (en) fused pyrazole derivatives as kinase inhibitors
CL2014001752A1 (en) Substituted bicyclic compounds; pharmaceutical composition that includes them; and use in the treatment of diseases such as cancer, Alzheimer's, AIDS, among others.
MX386924B (en) PYRROLO[3,2-D]PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS AND OTHER DISEASES.
BR112015007503A2 (en) therapeutically active oxazoline derivatives
CR20140200A (en) SOLID FORMS OF 3- (5-AMINO-2-METHYL-4-OXO-AH-QUINAZOLIN-3-IL) -PIPERIDIN-2,6-DIONA, AND ITS PHARMACEUTICAL COMPOSITIONS AND THEIR USES
BR112016011483A2 (en) IMIDAZOTRIAZINE DERIVATIVES AS MODULATORS OF TNF ACTIVITY
BR112016029632A2 (en) fused bicyclic heteroaromatic derivatives as kinase inhibitors
CL2015002030A1 (en) Substituted bicyclic dihydropyrimidinomas and their use as inhibitors of neutrophilic elastase activity
BR112016029635A2 (en) pyrazolo pyridine derivatives as kinase inhibitors
MX2015014677A (en) PHARMACEUTICAL FORMULATIONS, PROCESS, SOLID FORMS AND METHODS OF USE RELATED TO 1-ETIL-7- (2-METHYL-6- (1H-1,2,4-TRIAZOL-3-II) PI RIDIN-3-II) -3 , 4-HYDROPIRAZINE [2,3-B] PIRAZIN-2 (1H) -ONA.
CR20160155A (en) TIENOURACILCARBOXAMIDAS AND USES OF THE SAME
DK3596080T3 (en) PHARMACOLOGICAL ACTIVE ALICYCLIC-SUBSTITUTED PYRAZOLO [1,5-A] PYRIMIDINE DERIVATIVES
ECSP15031293A (en) THERAPEUTICALLY ACTIVE PYRAZOLO-PYRIMIDINE DERIVATIVES
UA114825C2 (en) Therapeutically active derivatives of pyrazolopyrimidine
EA201891349A1 (en) HEXAGIDROPYRAZINOTRIASINON DERIVATIVES AS KINASE INHIBITORS
EA201890826A1 (en) CONDENSED PYRIDINE DERIVATIVES AS KINASE INHIBITORS
AR125919A2 (en) SUSTAINED-RELEASE RUXOLITINIB DOSAGE FORMS
ECSP15025357A (en) SUSTAINED RELEASE RUXOLITINIB DOSAGE FORMS