ECSP17050310A - Ciclopropabenzofuranil-piridopirazindionas novedosas - Google Patents

Ciclopropabenzofuranil-piridopirazindionas novedosas

Info

Publication number
ECSP17050310A
ECSP17050310A ECIEPI201750310A ECPI201750310A ECSP17050310A EC SP17050310 A ECSP17050310 A EC SP17050310A EC IEPI201750310 A ECIEPI201750310 A EC IEPI201750310A EC PI201750310 A ECPI201750310 A EC PI201750310A EC SP17050310 A ECSP17050310 A EC SP17050310A
Authority
EC
Ecuador
Prior art keywords
pyridopyrazindionas
novedosas
ciclopropabenzofuranil
please see
attached document
Prior art date
Application number
ECIEPI201750310A
Other languages
English (en)
Inventor
Martin Youngjin Pettersson
Patrick Robert Verhoest
Gregory Wayne Kauffman
Ende Christopher William Am
Antonia Friederike Stepan
Douglas Scott Johnson
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of ECSP17050310A publication Critical patent/ECSP17050310A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

FAVOR VER DOCUMENTO ADJUNTO
ECIEPI201750310A 2015-02-03 2017-08-03 Ciclopropabenzofuranil-piridopirazindionas novedosas ECSP17050310A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562111222P 2015-02-03 2015-02-03

Publications (1)

Publication Number Publication Date
ECSP17050310A true ECSP17050310A (es) 2017-11-30

Family

ID=55299692

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201750310A ECSP17050310A (es) 2015-02-03 2017-08-03 Ciclopropabenzofuranil-piridopirazindionas novedosas

Country Status (22)

Country Link
US (2) US20160222007A1 (es)
EP (1) EP3253755B1 (es)
JP (1) JP6628805B2 (es)
KR (1) KR102000382B1 (es)
CN (1) CN107406445B (es)
AR (1) AR103582A1 (es)
AU (1) AU2016214102B2 (es)
BR (1) BR112017015693A2 (es)
CA (1) CA2919338A1 (es)
DK (1) DK3253755T3 (es)
EA (1) EA033423B1 (es)
EC (1) ECSP17050310A (es)
ES (1) ES2818806T3 (es)
IL (1) IL253635A0 (es)
MX (1) MX368391B (es)
PE (1) PE20171318A1 (es)
PH (1) PH12017501369A1 (es)
SG (1) SG11201705780PA (es)
TN (1) TN2017000342A1 (es)
TW (1) TWI616445B (es)
UY (1) UY36546A (es)
WO (1) WO2016125048A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20210393621A1 (en) 2018-10-26 2021-12-23 The Research Foundation For The State University Of New York Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia
KR102271305B1 (ko) 2020-05-21 2021-06-30 주식회사 아리바이오 치매 예방 및 치료용 조성물
CN111978324A (zh) * 2020-08-28 2020-11-24 开封康诺药业有限公司 一种多索茶碱的晶型及其制备方法
KR102272907B1 (ko) 2020-11-05 2021-07-05 주식회사 아리바이오 치매 예방 및 치료용 조성물
KR102272910B1 (ko) 2021-01-28 2021-07-06 주식회사 아리바이오 당뇨병을 동반한 치매 예방 및 치료용 조성물
KR102311224B1 (ko) * 2021-04-23 2021-10-13 주식회사 아리바이오 Pde5 억제제와 글루코코르티코이드 수용체 길항제 병용투여를 통한 치매 예방 및 치료용 조성물

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