ECSP19014247A - Formas de dosificación para tratar y prevenir trastornos del sueño - Google Patents

Formas de dosificación para tratar y prevenir trastornos del sueño

Info

Publication number
ECSP19014247A
ECSP19014247A ECSENADI201914247A ECDI201914247A ECSP19014247A EC SP19014247 A ECSP19014247 A EC SP19014247A EC SENADI201914247 A ECSENADI201914247 A EC SENADI201914247A EC DI201914247 A ECDI201914247 A EC DI201914247A EC SP19014247 A ECSP19014247 A EC SP19014247A
Authority
EC
Ecuador
Prior art keywords
dosage forms
treat
sleep disorders
prevent sleep
animal
Prior art date
Application number
ECSENADI201914247A
Other languages
English (en)
Inventor
Garth Whiteside
Donald J Kyle
Stephen C Harris
Ram P Kapil
Original Assignee
Purdue Pharma Lp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Purdue Pharma Lp filed Critical Purdue Pharma Lp
Publication of ECSP19014247A publication Critical patent/ECSP19014247A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M21/00Other devices or methods to cause a change in the state of consciousness; Devices for producing or ending sleep by mechanical, optical, or acoustical means, e.g. for hypnosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Anesthesiology (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Physics & Mathematics (AREA)
  • Acoustics & Sound (AREA)
  • Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

La descripción se refiere a formas de dosificación para tratar o prevenir un trastorno del sueño por administración de un compuesto de la fórmula (1) (ver figura), o un compuesto de la fórmula (1A), (1B), (1C), (1D), (1E), o (1F) a un animal que necesita de tal tratamiento. En determinadas modalidades, tales compuestos tratan o previenen de modo eficaz un trastorno del sueño en el animal, mientras se producen menos cantidad de efectos colaterales en comparación con compuestos previamente disponibles.
ECSENADI201914247A 2016-07-26 2019-02-26 Formas de dosificación para tratar y prevenir trastornos del sueño ECSP19014247A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662366960P 2016-07-26 2016-07-26
US201762536097P 2017-07-24 2017-07-24
PCT/IB2017/054506 WO2018020418A1 (en) 2016-07-26 2017-07-25 Treatment and prevention of sleep disorders

Publications (1)

Publication Number Publication Date
ECSP19014247A true ECSP19014247A (es) 2019-05-31

Family

ID=59714072

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSENADI201914247A ECSP19014247A (es) 2016-07-26 2019-02-26 Formas de dosificación para tratar y prevenir trastornos del sueño

Country Status (20)

Country Link
US (4) US10974081B2 (es)
EP (1) EP3490563A1 (es)
JP (2) JP7198197B2 (es)
KR (2) KR102531366B1 (es)
CN (1) CN109689058B (es)
AU (2) AU2017304898B2 (es)
BR (1) BR112019001457A2 (es)
CA (1) CA3031388C (es)
CL (1) CL2019000190A1 (es)
EC (1) ECSP19014247A (es)
IL (1) IL264294B (es)
JO (1) JOP20190008A1 (es)
MX (1) MX388469B (es)
NZ (1) NZ750817A (es)
PH (1) PH12019500177A1 (es)
SG (1) SG11201900486WA (es)
TN (1) TN2019000019A1 (es)
TW (1) TWI661827B (es)
WO (1) WO2018020418A1 (es)
ZA (1) ZA201901055B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JOP20190008A1 (ar) 2016-07-26 2019-01-24 Purdue Pharma Lp علاج ومنع اضطرابات النوم
CN111601591A (zh) * 2018-01-24 2020-08-28 普渡制药公司 睡眠障碍的治疗和预防
CA3097445A1 (en) * 2018-04-16 2019-10-24 Technologies Hop-Child, Inc. Systems and methods for the determination of arousal states, calibrated communication signals and monitoring arousal states
KR102198846B1 (ko) * 2018-06-29 2021-01-05 다인기술 주식회사 배뇨에 관한 설문을 수행하는 방법, 시스템 및 비일시성의 컴퓨터 판독 가능 기록 매체
CN111359074B (zh) * 2018-12-26 2022-08-02 财团法人工业技术研究院 个人化参数学习方法、睡眠辅助装置及存储介质
US11547350B2 (en) 2018-12-26 2023-01-10 Industrial Technology Research Institute Personalized parameter learning method, sleep-aid device and non-transitory computer readable medium
US12371427B2 (en) * 2019-01-31 2025-07-29 Purdue Pharma L.P. Polymorphic forms of a substituted-quinoxaline-type bridged-piperidine compound
KR20220062361A (ko) * 2019-09-13 2022-05-16 다케다 야쿠힌 고교 가부시키가이샤 과도한 졸림의 치료를 위한 오렉신 2 수용체 효능제의 용도
CN114159568B (zh) * 2020-09-11 2025-08-01 北京原基华毅生物科技有限公司 Sik抑制剂在制备用于预防和/或治疗睡眠障碍的药物中的应用
BR112023023702A2 (pt) 2021-05-21 2024-01-30 Purdue Pharma Lp Métodos de tratamento da cistite intersticial/síndrome da dor na bexiga
TWI804037B (zh) * 2021-11-02 2023-06-01 長庚醫療財團法人高雄長庚紀念醫院 生酮飲食之評估系統及其運作方法
CN119421705A (zh) * 2022-06-24 2025-02-11 普渡制药公司 治疗或预防膀胱过度活动综合征的方法
AU2024364388A1 (en) 2023-10-19 2026-03-19 Purdue Pharma L.P. Sunobinop for use in method of treating alcohol use disorder

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3536809A (en) 1969-02-17 1970-10-27 Alza Corp Medication method
US3598123A (en) 1969-04-01 1971-08-10 Alza Corp Bandage for administering drugs
US3845770A (en) 1972-06-05 1974-11-05 Alza Corp Osmatic dispensing device for releasing beneficial agent
US3916899A (en) 1973-04-25 1975-11-04 Alza Corp Osmotic dispensing device with maximum and minimum sizes for the passageway
US4008719A (en) 1976-02-02 1977-02-22 Alza Corporation Osmotic system having laminar arrangement for programming delivery of active agent
IE58110B1 (en) 1984-10-30 1993-07-14 Elan Corp Plc Controlled release powder and process for its preparation
US5073543A (en) 1988-07-21 1991-12-17 G. D. Searle & Co. Controlled release formulations of trophic factors in ganglioside-lipsome vehicle
IT1229203B (it) 1989-03-22 1991-07-25 Bioresearch Spa Impiego di acido 5 metiltetraidrofolico, di acido 5 formiltetraidrofolico e dei loro sali farmaceuticamente accettabili per la preparazione di composizioni farmaceutiche in forma a rilascio controllato attive nella terapia dei disturbi mentali organici e composizioni farmaceutiche relative.
US5120548A (en) 1989-11-07 1992-06-09 Merck & Co., Inc. Swelling modulated polymeric drug delivery device
US5733566A (en) 1990-05-15 1998-03-31 Alkermes Controlled Therapeutics Inc. Ii Controlled release of antiparasitic agents in animals
US5698155A (en) 1991-05-31 1997-12-16 Gs Technologies, Inc. Method for the manufacture of pharmaceutical cellulose capsules
US5580578A (en) 1992-01-27 1996-12-03 Euro-Celtique, S.A. Controlled release formulations coated with aqueous dispersions of acrylic polymers
US5591767A (en) 1993-01-25 1997-01-07 Pharmetrix Corporation Liquid reservoir transdermal patch for the administration of ketorolac
IT1270594B (it) 1994-07-07 1997-05-07 Recordati Chem Pharm Composizione farmaceutica a rilascio controllato di moguisteina in sospensione liquida
ATE301457T1 (de) 1995-06-12 2005-08-15 Searle & Co Mittel, enthaltend einen cyclooxygenase-2 inhibitor und einen 5-lipoxygenase inhibitor
US6572891B1 (en) 1999-10-23 2003-06-03 Alkaloid Ad Sublingual oral dosage form
DK1491212T3 (da) 2002-03-29 2012-10-29 Mitsubishi Tanabe Pharma Corp Middel til behandling af søvnforstyrrelser
AU2004238321B2 (en) 2003-05-07 2009-08-27 Samyang Biopharmaceuticals Corporation Highly plastic granules for making fast melting tablets
US8067603B2 (en) 2003-09-25 2011-11-29 Solvay Pharmaceuticals B.V. Benzimidazolone and quinazolinone derivatives as agonists on human ORL1 receptors
US7355045B2 (en) 2004-01-05 2008-04-08 Applera Corporation Isotopically enriched N-substituted piperazine acetic acids and methods for the preparation thereof
WO2006025267A1 (ja) 2004-08-31 2006-03-09 Mitsubishi Pharma Corporation Per2タンパク質レベルの低下を作用機序とする睡眠障害治療薬
PL2063861T3 (pl) 2006-09-15 2015-07-31 Echo Pharmaceuticals Bv Jednostka dawkowania do podawania podjęzykowego, podpoliczkowego lub doustnego nierozpuszczalnych w wodzie substancji aktywnych farmaceutycznie
JP5554709B2 (ja) * 2007-08-31 2014-07-23 パーデュー、ファーマ、リミテッド、パートナーシップ 置換キノキサリンタイプピペリジン化合物とその使用
MY173730A (en) 2008-03-11 2020-02-18 Takeda Pharmaceuticals Co Orally-disintegrating solid preparation
ES2393849T7 (es) * 2008-07-21 2015-01-28 Purdue Pharma Lp Compuestos de piperidina puenteada, de tipo quinoxalina sustituida, y usos de los mismos
US9290488B2 (en) 2011-12-01 2016-03-22 Purdue Pharma L.P. Azetidine-substituted quinoxalines as opioid receptor like-1 modulators
US10118927B2 (en) * 2012-12-27 2018-11-06 Purdue Pharma L.P. Substituted piperidin-4-amino-type compounds and uses thereof
WO2014102592A2 (en) * 2012-12-27 2014-07-03 Purdue Pharma L.P. Oxime/substituted quinoxaline-type piperidine compounds and uses thereof
JOP20190008A1 (ar) 2016-07-26 2019-01-24 Purdue Pharma Lp علاج ومنع اضطرابات النوم

Also Published As

Publication number Publication date
US11738023B2 (en) 2023-08-29
BR112019001457A2 (pt) 2019-05-07
WO2018020418A1 (en) 2018-02-01
AU2017304898A1 (en) 2019-03-07
JP2021120379A (ja) 2021-08-19
AU2017304898B2 (en) 2020-08-20
TWI661827B (zh) 2019-06-11
TW201817423A (zh) 2018-05-16
TN2019000019A1 (en) 2020-07-15
AU2020273332A1 (en) 2020-12-17
MX2019001036A (es) 2019-06-10
CN109689058B (zh) 2022-03-22
CN109689058A (zh) 2019-04-26
CA3031388C (en) 2023-02-14
CA3031388A1 (en) 2018-02-01
CL2019000190A1 (es) 2019-06-07
AU2020273332B2 (en) 2022-11-24
EP3490563A1 (en) 2019-06-05
KR102531366B1 (ko) 2023-05-12
KR102210209B1 (ko) 2021-02-01
ZA201901055B (en) 2019-12-18
KR20210013319A (ko) 2021-02-03
MX388469B (es) 2025-03-20
US12370191B2 (en) 2025-07-29
IL264294A (en) 2019-02-28
JP2019523269A (ja) 2019-08-22
JP7291172B2 (ja) 2023-06-14
JOP20190008A1 (ar) 2019-01-24
IL264294B (en) 2022-06-01
PH12019500177A1 (en) 2019-10-14
NZ750817A (en) 2020-07-31
SG11201900486WA (en) 2019-02-27
JP7198197B2 (ja) 2022-12-28
US10974081B2 (en) 2021-04-13
US20260007660A1 (en) 2026-01-08
KR20190029682A (ko) 2019-03-20
US20240058333A1 (en) 2024-02-22
US20190282836A1 (en) 2019-09-19
US20210330994A1 (en) 2021-10-28

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