ECSP21019076A - Método de producción de derivados de 4-metoxipirrol - Google Patents

Método de producción de derivados de 4-metoxipirrol

Info

Publication number
ECSP21019076A
ECSP21019076A ECSENADI202119076A ECDI202119076A ECSP21019076A EC SP21019076 A ECSP21019076 A EC SP21019076A EC SENADI202119076 A ECSENADI202119076 A EC SENADI202119076A EC DI202119076 A ECDI202119076 A EC DI202119076A EC SP21019076 A ECSP21019076 A EC SP21019076A
Authority
EC
Ecuador
Prior art keywords
methoxypirrol
production method
derivatives production
derivatives
present disclosure
Prior art date
Application number
ECSENADI202119076A
Other languages
English (en)
Inventor
Jeong Hyun Son
Deok Ki Eom
Jeong Taek Shin
Original Assignee
Dae Woong Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dae Woong Pharma filed Critical Dae Woong Pharma
Publication of ECSP21019076A publication Critical patent/ECSP21019076A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • C07D207/48—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Compositions Of Macromolecular Compounds (AREA)

Abstract

La presente divulgación se refiere a un método de fabricación de derivados de 4-metoxipirrol. La realización de la presente divulgación es útil para la producción industrial en masa de derivados de 4-metoxipirrol, ya que se mejoran el rendimiento y la eficiencia del procedimiento y se evita el uso de reactivos peligrosos y reactivos contaminantes para el medioambiente.
ECSENADI202119076A 2018-09-19 2021-03-18 Método de producción de derivados de 4-metoxipirrol ECSP21019076A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR20180112196 2018-09-19
KR1020190110997A KR102126576B1 (ko) 2018-09-19 2019-09-06 4-메톡시 피롤 유도체의 제조 방법

Publications (1)

Publication Number Publication Date
ECSP21019076A true ECSP21019076A (es) 2021-05-31

Family

ID=69959291

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSENADI202119076A ECSP21019076A (es) 2018-09-19 2021-03-18 Método de producción de derivados de 4-metoxipirrol

Country Status (21)

Country Link
US (1) US12110271B2 (es)
EP (1) EP3854784B1 (es)
JP (1) JP7253624B2 (es)
KR (1) KR102126576B1 (es)
CN (1) CN112739684B (es)
AU (1) AU2019343857B2 (es)
BR (1) BR112021005156A2 (es)
CL (1) CL2021000639A1 (es)
CO (1) CO2021003195A2 (es)
DO (1) DOP2021000042A (es)
EC (1) ECSP21019076A (es)
JO (1) JOP20210040A1 (es)
MA (1) MA53673A (es)
MX (1) MX2021003137A (es)
MY (1) MY205351A (es)
PE (1) PE20211736A1 (es)
PH (1) PH12021550523A1 (es)
RU (1) RU2763287C1 (es)
SA (1) SA521421372B1 (es)
SG (1) SG11202101919VA (es)
TN (1) TN2021000035A1 (es)

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KR102126576B1 (ko) 2018-09-19 2020-06-24 주식회사 대웅제약 4-메톡시 피롤 유도체의 제조 방법
DK4245298T3 (en) 2020-12-18 2026-03-30 Daewoong Pharmaceutical Co Ltd Hidtil ukendt formulering til oral administration, som omfatter 1-(5-(2,4-difluorphenyl)-1-((3-fluorphenyl)sulfonyl)-4-methoxy-1h-pyrrol-3-yl)-n-methylmethanamin
KR102556500B1 (ko) * 2021-11-19 2023-07-19 하나제약 주식회사 피롤 유도체 또는 이의 약학적 또는 식품학적으로 허용 가능한 염, 및 이를 유효성분으로 포함하는 위장 질환의 예방, 개선 또는 치료용 조성물
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CN119365448A (zh) * 2022-05-23 2025-01-24 日东制药株式会社 一种6-甲氧基吡啶-3-基衍生物的制备方法
CN117820193A (zh) * 2022-09-29 2024-04-05 安徽皓元药业有限公司 一种非苏拉赞盐酸盐晶型a及其制备方法
KR102938657B1 (ko) 2023-02-15 2026-03-12 주식회사 대웅제약 4-메톡시 피롤 유도체의 제조 방법
WO2025023734A1 (en) * 2023-07-26 2025-01-30 Yunovia Co., Ltd. Method for preparing intermediates of 6-methoxypyridine-3-yl derivatives

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WO2007114338A1 (ja) * 2006-03-31 2007-10-11 Takeda Pharmaceutical Company Limited 酸分泌抑制薬
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KR102081920B1 (ko) 2016-03-25 2020-02-26 주식회사 대웅제약 1-(5-(2,4-다이플루오로페닐)-1-((3-플루오로페닐)술포닐)-4-메톡시-1h-피롤-3-일)-n-메틸메탄아민 염의 신규한 결정형
KR20170113040A (ko) 2016-03-25 2017-10-12 주식회사 대웅제약 1-(5-(2,4-다이플루오로페닐)-1-((3-플루오로페닐)술포닐)-4-메톡시-1h-피롤-3-일)-n-메틸메탄아민의 신규한 산부가염
CN107879964B (zh) * 2016-09-29 2023-02-10 江苏柯菲平医药股份有限公司 1-(5-(2-氟苯基)-1-(3-(3-甲氧丙氧基)苯磺酰氯)-1h-吡咯-3-基)-n-甲基胺的制备方法
KR102233456B1 (ko) 2017-05-31 2021-03-29 주식회사 대웅제약 4-메톡시피롤 유도체의 중간체 제조 방법
KR102233455B1 (ko) 2017-06-21 2021-03-29 주식회사 대웅제약 4-메톡시피롤 유도체의 중간체 제조 방법
CN108503621B (zh) * 2017-12-25 2021-09-14 上海中拓医药科技有限公司 一种富马酸沃诺拉赞的制备方法
KR102126576B1 (ko) 2018-09-19 2020-06-24 주식회사 대웅제약 4-메톡시 피롤 유도체의 제조 방법
WO2020060213A1 (ko) 2018-09-19 2020-03-26 주식회사 대웅제약 4-메톡시 피롤 유도체의 제조 방법
TN2023000270A1 (en) 2021-05-26 2025-07-02 Daewoong Pharmaceutical Co Ltd Medicine container containing liquid pharmaceutical composition of 1-(5-(2,4-difluorophenyl)-1-((3-fluorophenyl)sulfonyl)-4-methoxy-1h-pyrrol-3-yl)-n-methylmethanamine

Also Published As

Publication number Publication date
KR20200033178A (ko) 2020-03-27
AU2019343857A1 (en) 2021-04-15
KR102126576B1 (ko) 2020-06-24
US12110271B2 (en) 2024-10-08
US20210221770A1 (en) 2021-07-22
CN112739684A (zh) 2021-04-30
TN2021000035A1 (en) 2022-10-03
CO2021003195A2 (es) 2021-04-08
JOP20210040A1 (ar) 2021-03-07
CA3110830A1 (en) 2020-03-26
MX2021003137A (es) 2021-05-14
BR112021005156A2 (pt) 2021-06-15
PE20211736A1 (es) 2021-09-06
AU2019343857B2 (en) 2021-12-02
PH12021550523A1 (en) 2022-02-21
NZ773997A (en) 2024-03-22
EP3854784A4 (en) 2022-03-30
EP3854784B1 (en) 2026-04-15
CN112739684B (zh) 2024-06-04
SG11202101919VA (en) 2021-04-29
RU2763287C1 (ru) 2021-12-28
JP7253624B2 (ja) 2023-04-06
JP2021535934A (ja) 2021-12-23
MY205351A (en) 2024-10-17
EP3854784A1 (en) 2021-07-28
MA53673A (fr) 2022-03-30
SA521421372B1 (ar) 2024-01-25
DOP2021000042A (es) 2021-05-31
CL2021000639A1 (es) 2021-08-06

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