ECSP961694A - PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M) - Google Patents
PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M)Info
- Publication number
- ECSP961694A ECSP961694A ECSP961694A ECSP961694A EC SP961694 A ECSP961694 A EC SP961694A EC SP961694 A ECSP961694 A EC SP961694A EC SP961694 A ECSP961694 A EC SP961694A
- Authority
- EC
- Ecuador
- Prior art keywords
- procedure
- case
- olanzapine
- preparing
- methyl
- Prior art date
Links
- KVWDHTXUZHCGIO-UHFFFAOYSA-N olanzapine Chemical compound C1CN(C)CCN1C1=NC2=CC=CC=C2NC2=C1C=C(C)S2 KVWDHTXUZHCGIO-UHFFFAOYSA-N 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 229960005017 olanzapine Drugs 0.000 title abstract 2
- 239000012453 solvate Substances 0.000 abstract 2
- 230000001476 alcoholic effect Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Landscapes
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
El invento se refiere a un nuevo procedimiento para preparar 2-metil-4-(4-metil-1-piperacinil)-10H-tieno[2,3-b][1,5] benzodiacepina (denominada en lo sucesivo con su nombre genérico "olanzapina") y a nuevos solvatos alcohólicos valiosos en este procedimiento, especilamente una forma de solvato monometanólico cristalino de un compuesto de la siguiente fórmula: (gráfico).The invention relates to a new process for preparing 2-methyl-4- (4-methyl-1-piperazinyl) -10H-thieno [2,3-b] [1,5] benzodiazepine (hereinafter named Generic "Olanzapine") and to new valuable alcoholic solvates in this process, specifically a form of crystalline monomethanolic solvate of a compound of the following formula: (graph).
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP961694 ECSP961694A (en) | 1996-03-21 | 1996-03-21 | PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M) |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP961694 ECSP961694A (en) | 1996-03-21 | 1996-03-21 | PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M) |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP961694A true ECSP961694A (en) | 1997-11-04 |
Family
ID=42042426
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP961694 ECSP961694A (en) | 1996-03-21 | 1996-03-21 | PROCEDURE FOR PREPARING OLANZAPINE (CASE X - 9992M) |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP961694A (en) |
-
1996
- 1996-03-21 EC ECSP961694 patent/ECSP961694A/en unknown
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