ECSP961814A - NEW AZEPANOS AND HOMOLOGES OF ITS RING (CASE RAN 4070/103) - Google Patents

NEW AZEPANOS AND HOMOLOGES OF ITS RING (CASE RAN 4070/103)

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Publication number
ECSP961814A
ECSP961814A ECSP961814A ECSP961814A EC SP961814 A ECSP961814 A EC SP961814A EC SP961814 A ECSP961814 A EC SP961814A EC SP961814 A ECSP961814 A EC SP961814A
Authority
EC
Ecuador
Prior art keywords
azepanos
homologes
ring
new
phenyl
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Pierre Barbier
Josef Stadlwieser
Sven Taylor
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP961814 priority Critical patent/ECSP961814A/en
Publication of ECSP961814A publication Critical patent/ECSP961814A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

El invento se refiere a: Compuestos de fórmula general (gráfico), en donde R1 es fenilo o alfa o beta-naftilo, los cuales pueden estar sustituidos con hidroxilo, alquilo inferior, alcoxilo inferior, alcoxi carbonilo inferior, fenoxilo, aciloxilo, hidroxifenoxi-sulfonilo, halógeno, nitro amino, acilamino o N -alquil acilamino inferior; R2 es fenilo o fenilo sustituido con hidroxilo o aciloxilo; Y es un enlace carbono carbono o es vinileno; y n es 1,2, ó 3 y las sales de adición ácida farmacéuticamente aceptables de los mismos.The invention relates to: Compounds of general formula (graph), wherein R1 is phenyl or alpha or beta-naphthyl, which may be substituted with hydroxyl, lower alkyl, lower alkoxy, lower alkoxycarbonyl, phenoxy, acyloxy, hydroxyphenoxy- sulfonyl, halogen, nitro amino, acylamino or N-lower alkyl acylamino; R2 is phenyl or phenyl substituted by hydroxyl or acyloxy; Y is a carbon-carbon bond or is vinylene; and n is 1,2, or 3 and the pharmaceutically acceptable acid addition salts thereof.

ECSP961814 1996-07-05 1996-07-05 NEW AZEPANOS AND HOMOLOGES OF ITS RING (CASE RAN 4070/103) ECSP961814A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP961814 ECSP961814A (en) 1996-07-05 1996-07-05 NEW AZEPANOS AND HOMOLOGES OF ITS RING (CASE RAN 4070/103)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP961814 ECSP961814A (en) 1996-07-05 1996-07-05 NEW AZEPANOS AND HOMOLOGES OF ITS RING (CASE RAN 4070/103)

Publications (1)

Publication Number Publication Date
ECSP961814A true ECSP961814A (en) 1997-12-09

Family

ID=42042544

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP961814 ECSP961814A (en) 1996-07-05 1996-07-05 NEW AZEPANOS AND HOMOLOGES OF ITS RING (CASE RAN 4070/103)

Country Status (1)

Country Link
EC (1) ECSP961814A (en)

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