ECSP961876A - PHARMACEUTICAL FORMULATIONS - Google Patents

PHARMACEUTICAL FORMULATIONS

Info

Publication number
ECSP961876A
ECSP961876A ECSP961876A ECSP961876A EC SP961876 A ECSP961876 A EC SP961876A EC SP961876 A ECSP961876 A EC SP961876A EC SP961876 A ECSP961876 A EC SP961876A
Authority
EC
Ecuador
Prior art keywords
darifenacin
pharmaceutically acceptable
patient
dosage form
pharmaceutical formulations
Prior art date
Application number
Other languages
Spanish (es)
Inventor
John Michael Humphrey
Thomas Francis Dolan
Donald John Nichols
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP961876 priority Critical patent/ECSP961876A/en
Publication of ECSP961876A publication Critical patent/ECSP961876A/en

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  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

El invento proporciona una forma de dosificación farmacéutica adaptada para la administración en el tracto gastrointestinal de un paciente que comprende darifenacina, o una de sus sales farmacéuticamente aceptable y un adyuvante diluyente o vehículo farmacéuticamente aceptable caracterizada porque la forma de dosificación está adaptada para liberar al menos el 10% en peso de la darifenacina o de su sal farmacéuticamente aceptable, en el tracto gastrointestinal inferior del paciente. La formulación minimiza los efectos secundarios indeseados y aumenta la biodisponibilidad de la darifenacina.The invention provides a pharmaceutical dosage form adapted for administration to the gastrointestinal tract of a patient comprising darifenacin, or a pharmaceutically acceptable salt thereof and a diluting adjuvant or pharmaceutically acceptable carrier characterized in that the dosage form is adapted to release at least 10% by weight of darifenacin or its pharmaceutically acceptable salt, in the patient's lower gastrointestinal tract. The formulation minimizes unwanted side effects and increases the bioavailability of darifenacin.

ECSP961876 1996-09-13 1996-09-13 PHARMACEUTICAL FORMULATIONS ECSP961876A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP961876 ECSP961876A (en) 1996-09-13 1996-09-13 PHARMACEUTICAL FORMULATIONS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP961876 ECSP961876A (en) 1996-09-13 1996-09-13 PHARMACEUTICAL FORMULATIONS

Publications (1)

Publication Number Publication Date
ECSP961876A true ECSP961876A (en) 1997-11-28

Family

ID=42042602

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP961876 ECSP961876A (en) 1996-09-13 1996-09-13 PHARMACEUTICAL FORMULATIONS

Country Status (1)

Country Link
EC (1) ECSP961876A (en)

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