ECSP961937A - PROTEIN KINASE INHIBITOR "C" - Google Patents

PROTEIN KINASE INHIBITOR "C"

Info

Publication number
ECSP961937A
ECSP961937A ECSP961937A ECSP961937A EC SP961937 A ECSP961937 A EC SP961937A EC SP961937 A ECSP961937 A EC SP961937A EC SP961937 A ECSP961937 A EC SP961937A
Authority
EC
Ecuador
Prior art keywords
protein kinase
kinase inhibitor
bisindolylmaleimide
solvates
mammals
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Leonard Larry Winneroski
Margaret Mary Faul
Nagy Alphonse Farid
Gary Lowell Engel
Michael Robert Jirousek
Lori Ann Richardson
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP961937 priority Critical patent/ECSP961937A/en
Publication of ECSP961937A publication Critical patent/ECSP961937A/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

El invento se refiere a nuevos derivados macrocíclicos bisindolilmaleimida de fórmula: (gráfico) y sus solvatos. La invención proporciona además la preparación, formulaciones farmacéuticas y procedimientos de uso para inhibir la proteína quinasa C en mamíferos.The invention relates to novel macrocyclic bisindolylmaleimide derivatives of the formula: (graph) and their solvates. The invention further provides the preparation, pharmaceutical formulations and methods of use for inhibiting protein kinase C in mammals.

ECSP961937 1996-11-18 1996-11-18 PROTEIN KINASE INHIBITOR "C" ECSP961937A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP961937 ECSP961937A (en) 1996-11-18 1996-11-18 PROTEIN KINASE INHIBITOR "C"

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP961937 ECSP961937A (en) 1996-11-18 1996-11-18 PROTEIN KINASE INHIBITOR "C"

Publications (1)

Publication Number Publication Date
ECSP961937A true ECSP961937A (en) 1998-04-17

Family

ID=42042663

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP961937 ECSP961937A (en) 1996-11-18 1996-11-18 PROTEIN KINASE INHIBITOR "C"

Country Status (1)

Country Link
EC (1) ECSP961937A (en)

Similar Documents

Publication Publication Date Title
ES2122764T3 (en) PROTEIN QUINASE C. INHIBITOR
MX9707431A (en) Protein kinase c inhibitors.
NO944643L (en) Protein kinase C inhibitors
MX9100628A (en) PEPTIDOMIMETIC COMPOUNDS OF BOROLISINA AND PROCEDURE FOR ITS PREPARATION.
ES2138691T3 (en) PROCEDURE FOR THE OBTAINING OF DERIVATIVES OF N-ACIL-5-FLUOROCITIDINA.
BG107171A (en) PURIN DERIVATIVES
DK0971717T3 (en) Cytotoxic amino sugar and related sugar derivatives of indolopyrrolocarbazoles
DE69917663D1 (en) 2-Methyl-THIENO BENZODIAZEPINE FORMULATION
ECSP961937A (en) PROTEIN KINASE INHIBITOR "C"
YU61096A (en) Novel intermediates, their use in the synthesis of n,n'-bridged bisindolylmaleimides and pharmaceutical formulations
ES2175661T3 (en) DERIVATIVES OF ISOFLAVONA, PROCEDURES FOR THE PREPARATION OF THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
AR008474A1 (en) DERIVATIVE OF 9-DIHYDROERYTHROMYCIN A 6.9; 11,12-DICICLOCARBONATO, PHARMACEUTICAL COMPOSITION AND BACTERICIDE PREPARATION THAT CONTAIN IT AND ITS USE
TR199701011A2 (en) 1-carb-(detia)-cephalosporin t�revleri.
ECSP961938A (en) NEW INTERMEDIATES AND THEIR USE TO PREPARE BISINDOLYL MALEIMIDES WITH A BRIDGE N, N-CASE X - 10386
ECSP972242A (en) PHARMACEUTICAL PRODUCT CRYSTALLINE