ECSP961938A - NEW INTERMEDIATES AND THEIR USE TO PREPARE BISINDOLYL MALEIMIDES WITH A BRIDGE N, N-CASE X - 10386 - Google Patents

NEW INTERMEDIATES AND THEIR USE TO PREPARE BISINDOLYL MALEIMIDES WITH A BRIDGE N, N-CASE X - 10386

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Publication number
ECSP961938A
ECSP961938A ECSP961938A ECSP961938A EC SP961938 A ECSP961938 A EC SP961938A EC SP961938 A ECSP961938 A EC SP961938A EC SP961938 A ECSP961938 A EC SP961938A
Authority
EC
Ecuador
Prior art keywords
bridge
prepare
case
new intermediates
bisindolyl maleimides
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Leonard Larry Winneroski
Margaret Mary Faul
Christine Ann Krumrich
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP961938 priority Critical patent/ECSP961938A/en
Publication of ECSP961938A publication Critical patent/ECSP961938A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)

Abstract

El invento se refiere a compuestos de fórmula: (gráfico), la invención proporciona además el uso de estos compuestos para preparar bisindolilmaleimidas con un puente N, N¿. Además, la invención proporciona formulaciones farmacéuticas y los procedimientos de uso para inhibir la proteína quinasa C en mamíferos.The invention relates to compounds of formula: (graph), the invention further provides the use of these compounds to prepare bisindolylmaleimides with an N, N¿ bridge. Furthermore, the invention provides pharmaceutical formulations and methods of use for inhibiting protein kinase C in mammals.

ECSP961938 1996-11-18 1996-11-18 NEW INTERMEDIATES AND THEIR USE TO PREPARE BISINDOLYL MALEIMIDES WITH A BRIDGE N, N-CASE X - 10386 ECSP961938A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP961938 ECSP961938A (en) 1996-11-18 1996-11-18 NEW INTERMEDIATES AND THEIR USE TO PREPARE BISINDOLYL MALEIMIDES WITH A BRIDGE N, N-CASE X - 10386

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP961938 ECSP961938A (en) 1996-11-18 1996-11-18 NEW INTERMEDIATES AND THEIR USE TO PREPARE BISINDOLYL MALEIMIDES WITH A BRIDGE N, N-CASE X - 10386

Publications (1)

Publication Number Publication Date
ECSP961938A true ECSP961938A (en) 1998-04-17

Family

ID=42042664

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP961938 ECSP961938A (en) 1996-11-18 1996-11-18 NEW INTERMEDIATES AND THEIR USE TO PREPARE BISINDOLYL MALEIMIDES WITH A BRIDGE N, N-CASE X - 10386

Country Status (1)

Country Link
EC (1) ECSP961938A (en)

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