ECSP961953A - PREPARATIONS CONTAINING CYCLOSPORIN - Google Patents
PREPARATIONS CONTAINING CYCLOSPORINInfo
- Publication number
- ECSP961953A ECSP961953A ECSP961953A ECSP961953A EC SP961953 A ECSP961953 A EC SP961953A EC SP961953 A ECSP961953 A EC SP961953A EC SP961953 A ECSP961953 A EC SP961953A
- Authority
- EC
- Ecuador
- Prior art keywords
- preparations containing
- containing cyclosporin
- cyclosporine
- solvents
- fatty acid
- Prior art date
Links
- PMATZTZNYRCHOR-CGLBZJNRSA-N Cyclosporin A Chemical compound CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O PMATZTZNYRCHOR-CGLBZJNRSA-N 0.000 title abstract 3
- 238000002360 preparation method Methods 0.000 title abstract 3
- 108010036949 Cyclosporine Proteins 0.000 title abstract 2
- 229960001265 ciclosporin Drugs 0.000 title abstract 2
- 229930182912 cyclosporin Natural products 0.000 title abstract 2
- 229930105110 Cyclosporin A Natural products 0.000 title 1
- 229940079593 drug Drugs 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 2
- 239000002904 solvent Substances 0.000 abstract 2
- 239000002202 Polyethylene glycol Substances 0.000 abstract 1
- 235000014113 dietary fatty acids Nutrition 0.000 abstract 1
- 229930195729 fatty acid Natural products 0.000 abstract 1
- 239000000194 fatty acid Substances 0.000 abstract 1
- -1 hydroxy fatty acid esters Chemical class 0.000 abstract 1
- 230000003589 nefrotoxic effect Effects 0.000 abstract 1
- 229920001223 polyethylene glycol Polymers 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Landscapes
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La invención se refiere a la preparación y al uso de preparados de medicamentos que contienen ciclosporina (s), que contiene una alta proporción de una combinación especial de agentes solubilizantes, como por ejemplos determinados ésteres de ácidos grasos hidroxi saturados con polietilenglicol y uno o más solventes o substancias portadoras. Los medicamentos preparados de acuerdo con la invención se caracterizan por una biodisponibilidad superior y al mismo tiempo menores efectos nefrotóxicos.The invention relates to the preparation and use of cyclosporine (s) containing drug preparations, which contain a high proportion of a special combination of solubilizing agents, such as for example certain hydroxy fatty acid esters saturated with polyethylene glycol and one or more solvents or carrier substances. Medicines prepared according to the invention are characterized by superior bioavailability and at the same time less nephrotoxic effects.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP961953 ECSP961953A (en) | 1996-11-28 | 1996-11-28 | PREPARATIONS CONTAINING CYCLOSPORIN |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP961953 ECSP961953A (en) | 1996-11-28 | 1996-11-28 | PREPARATIONS CONTAINING CYCLOSPORIN |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP961953A true ECSP961953A (en) | 1998-01-22 |
Family
ID=42042679
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP961953 ECSP961953A (en) | 1996-11-28 | 1996-11-28 | PREPARATIONS CONTAINING CYCLOSPORIN |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP961953A (en) |
-
1996
- 1996-11-28 EC ECSP961953 patent/ECSP961953A/en unknown
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