ECSP982708A - CYCLIC AMINO ACIDS AND THEIR DERIVATIVES USEFUL AS PHARMACEUTICAL AGENTS - Google Patents
CYCLIC AMINO ACIDS AND THEIR DERIVATIVES USEFUL AS PHARMACEUTICAL AGENTSInfo
- Publication number
- ECSP982708A ECSP982708A ECSP982708A ECSP982708A EC SP982708 A ECSP982708 A EC SP982708A EC SP982708 A ECSP982708 A EC SP982708A EC SP982708 A ECSP982708 A EC SP982708A
- Authority
- EC
- Ecuador
- Prior art keywords
- amino acids
- cyclic amino
- pharmaceutical agents
- derivatives useful
- disorders
- Prior art date
Links
- 150000001413 amino acids Chemical class 0.000 title 1
- 239000008177 pharmaceutical agent Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 208000035475 disorder Diseases 0.000 abstract 2
- 208000002551 irritable bowel syndrome Diseases 0.000 abstract 2
- 208000019901 Anxiety disease Diseases 0.000 abstract 1
- 208000018522 Gastrointestinal disease Diseases 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 230000036506 anxiety Effects 0.000 abstract 1
- 206010003246 arthritis Diseases 0.000 abstract 1
- -1 cyclic amino acids Chemical class 0.000 abstract 1
- 206010015037 epilepsy Diseases 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 230000000626 neurodegenerative effect Effects 0.000 abstract 1
- 230000002981 neuropathic effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 206010042772 syncope Diseases 0.000 abstract 1
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
La invención constituye una serie novedosa de aminoácidos cíclicos útiles para el tratamiento de: epilepsia, desmayos, trastornos, neurodegenerativos, depresión, ansiedad, pánico, dolor, trastornos neuropatológicos, trastornos gastrointestinales tales como el sindrome de intestino irritable (IBS) e inflamación, en especial artritis. Se incluye una composición farmacéutica que contiene un compuesto de la invención, asi como los métodos para preparar los compuestos y los intermedios útiles en la preparación de los compuestos finales.The invention constitutes a novel series of cyclic amino acids useful for the treatment of: epilepsy, fainting, disorders, neurodegenerative, depression, anxiety, panic, pain, neuropathological disorders, gastrointestinal disorders such as irritable bowel syndrome (IBS) and inflammation, in special arthritis. A pharmaceutical composition containing a compound of the invention is included, as well as methods for preparing the compounds and intermediates useful in preparing the final compounds.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP982708 ECSP982708A (en) | 1998-10-26 | 1998-10-26 | CYCLIC AMINO ACIDS AND THEIR DERIVATIVES USEFUL AS PHARMACEUTICAL AGENTS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP982708 ECSP982708A (en) | 1998-10-26 | 1998-10-26 | CYCLIC AMINO ACIDS AND THEIR DERIVATIVES USEFUL AS PHARMACEUTICAL AGENTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP982708A true ECSP982708A (en) | 1999-04-21 |
Family
ID=42043626
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP982708 ECSP982708A (en) | 1998-10-26 | 1998-10-26 | CYCLIC AMINO ACIDS AND THEIR DERIVATIVES USEFUL AS PHARMACEUTICAL AGENTS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP982708A (en) |
-
1998
- 1998-10-26 EC ECSP982708 patent/ECSP982708A/en unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CY1105062T1 (en) | CYCLIC AMINO ACIDS AND THEIR DERIVATIVES USEFUL AS THERAPEUTIC AGENTS | |
| CU23393A3 (en) | INHIBITING COMPOUNDS OF RAF KINASA AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| HN1998000157A (en) | PROSTAGLANDIN AGONISTS | |
| GT200500007A (en) | [1,8] NAFTIRIDIN-2-WAVES AND RELATED COMPOUNDS FOR THE TREATMENT OF CHICHOPHRENIA. | |
| CU23112A3 (en) | BICYCLE AMINO ACIDS AS PHARMACEUTICAL AGENTS | |
| AR002705A1 (en) | A NEW INDOLINA COMPOUND, A PROCESS FOR ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN IT. | |
| CO4810373A1 (en) | ARYL-CONDENSED AZAPOLYCLIC COMPOUNDS | |
| UY28482A1 (en) | NEW COMPOUNDS | |
| AR035861A1 (en) | CONDENSED BICYCLE OR TRICYCLIC AMINO ACIDS COMPOUNDS, PREPARATION PROCEDURE, PHARMACEUTICAL COMPOSITIONS AND THEIR USE IN THE PREPARATION OF MEDICINES | |
| UY27740A1 (en) | NEW COMPOUNDS | |
| CL2008000762A1 (en) | COMPOUNDS DERIVED FROM PYRIMIDINS; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE FOR THE TREATMENT OF PSORIASIS, DIABETES, REUMATOID ARTHRITIS, AMONG OTHER DISEASES (DIVISIONAL APPLICATION 1147-02). | |
| PE20050355A1 (en) | COMPOSITIONS REFERRED TO INHIBITORS OF VOLTAGE REGULATED ION CHANNELS | |
| SV2002000696A (en) | IMIDAZOL COMPOUNDS CONDENSED WITH ARILO OR HETEROARILO AS ANTI-INFLAMMATORY AND ANALGESIC AGENTS PC9985AHXK / BB | |
| GT199800046A (en) | PIRAZINE COMPOUNDS. | |
| AR019365A1 (en) | COMPOSITE OF 1-PIPERIDIN-3-PHENYL-BUTIL-NAFTAMIDE, PROCESS TO PREPARE IT, PHARMACEUTICAL COMPOSITION AND USE TO MANUFACTURE A USEFUL MEDICINAL PRODUCT FOR THE PROCESSING OF A DISEASE BY ENDOGENIC NEUROPEPTIDIC TACHYCINES | |
| ECSP045498A (en) | "DIFENILAZETIDINONAS REPLACED IN RING, METHOD FOR ITS PRODUCTION, MEDICATIONS THAT UNDERSTAND THESE COMPOUNDS AND THEIR USE" | |
| UY28144A1 (en) | THERAPEUTIC AGENTS | |
| ECSP055599A (en) | 5HT2a RECEPTOR AGONISM FOR THE TREATMENT OF THERMOREGULATORY DYSFUNCTION | |
| PA8542601A1 (en) | LIPID REDUCING BIFENYL CARBOXAMIDS | |
| MX9303670A (en) | DERIVATIVES OF BICYCLOOCTANE AND BICYCLOHEPTANE, METO DO FOR ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM. | |
| AR007240A1 (en) | ANALOGS OF VITAMIN D3 FLUORATED, MIXTURES AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND THEIR USE TO DEVELOP A PHARMACEUTICAL COMPOSITION | |
| DOP2002000372A (en) | CONDENSED BICYCLE OR TRICYCLE AMINO ACIDS | |
| AR041865A1 (en) | THERAPEUTIC DERIVATIVES OF PROLINA AND ITS USE IN THE TREATMENT OF EPILEPSY AND PAIN | |
| BRPI0411800A (en) | drug candidates and methods for their preparation | |
| BR0011039A (en) | Gaba analogs replaced with 3-heteroarylalkyl |