ECSP982729A - LEAGUES OF THE RECEPTOR H3 OF THE TYPE FENIL- ALQUIL- IMIDAZOLES - Google Patents
LEAGUES OF THE RECEPTOR H3 OF THE TYPE FENIL- ALQUIL- IMIDAZOLESInfo
- Publication number
- ECSP982729A ECSP982729A ECSP982729A ECSP982729A EC SP982729 A ECSP982729 A EC SP982729A EC SP982729 A ECSP982729 A EC SP982729A EC SP982729 A ECSP982729 A EC SP982729A
- Authority
- EC
- Ecuador
- Prior art keywords
- formula
- imidazoles
- diseases
- salt
- compound
- Prior art date
Links
- 150000003839 salts Chemical class 0.000 abstract 3
- 208000026935 allergic disease Diseases 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 210000001035 gastrointestinal tract Anatomy 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 239000012453 solvate Substances 0.000 abstract 2
- 208000024827 Alzheimer disease Diseases 0.000 abstract 1
- 208000024172 Cardiovascular disease Diseases 0.000 abstract 1
- 208000010412 Glaucoma Diseases 0.000 abstract 1
- 229940124056 Histamine H1 receptor antagonist Drugs 0.000 abstract 1
- 206010020751 Hypersensitivity Diseases 0.000 abstract 1
- 208000001953 Hypotension Diseases 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 208000019695 Migraine disease Diseases 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 230000007815 allergy Effects 0.000 abstract 1
- 210000003169 central nervous system Anatomy 0.000 abstract 1
- 239000000938 histamine H1 antagonist Substances 0.000 abstract 1
- 230000036543 hypotension Effects 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- 208000019116 sleep disease Diseases 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Se describen fenil-alquil-imidazoles nuevos de la fórmula (gráfico), o sus sales o solvatos farmacéuticamente aceptables, donde A y R son como definimos en la especificación además se describen los métodos para tratar la alergia, inflamación, enfermedades cardiovasculares, hipotensión, glaucoma, trastornos del sueño, enfermedades del tracto gastrointestinal, estados de hiper e hipo-movilidad del tracto gastrointestinal, enfermedades del sistema nervioso central, enfermedad de Alzheimer, esquizofreni, obesidad y migrañas, que comprenden administar una cantidad efectiva de un compuesto de la fórmula I (o su sal o sovato) a un paciente que necesita este tratamiento. Además se describen los métodos para el tratamiento de las respuestas alérgicas de las vias areas superiores que comprenden administrar un compuesto, su sal o solvato de la fórmula I en combinación o mezcla con un antagonista del receptor H1 de histamina.Novel phenyl-alkyl-imidazoles of the formula (graph), or their pharmaceutically acceptable salts or solvates are described, where A and R are as defined in the specification, and methods for treating allergy, inflammation, cardiovascular disease, hypotension, are described. glaucoma, sleep disorders, diseases of the gastrointestinal tract, hyper and hypo-mobility states of the gastrointestinal tract, diseases of the central nervous system, Alzheimer's disease, schizophreni, obesity and migraines, which comprise administering an effective amount of a compound of the formula I (or your salt or sovate) to a patient who needs this treatment. In addition, methods for the treatment of allergic responses of the upper airways are described, which comprise administering a compound, its salt or solvate of formula I in combination or mixture with a histamine H1 receptor antagonist.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP982729 ECSP982729A (en) | 1998-11-05 | 1998-11-05 | LEAGUES OF THE RECEPTOR H3 OF THE TYPE FENIL- ALQUIL- IMIDAZOLES |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP982729 ECSP982729A (en) | 1998-11-05 | 1998-11-05 | LEAGUES OF THE RECEPTOR H3 OF THE TYPE FENIL- ALQUIL- IMIDAZOLES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP982729A true ECSP982729A (en) | 1999-05-06 |
Family
ID=42043647
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP982729 ECSP982729A (en) | 1998-11-05 | 1998-11-05 | LEAGUES OF THE RECEPTOR H3 OF THE TYPE FENIL- ALQUIL- IMIDAZOLES |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP982729A (en) |
-
1998
- 1998-11-05 EC ECSP982729 patent/ECSP982729A/en unknown
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