ECSP982743A - PIRROL AMIDES SYNTHESIS PROCEDURES - Google Patents
PIRROL AMIDES SYNTHESIS PROCEDURESInfo
- Publication number
- ECSP982743A ECSP982743A ECSP982743A ECSP982743A EC SP982743 A ECSP982743 A EC SP982743A EC SP982743 A ECSP982743 A EC SP982743A EC SP982743 A ECSP982743 A EC SP982743A
- Authority
- EC
- Ecuador
- Prior art keywords
- pirrol
- synthesis procedures
- amides synthesis
- followed
- reaction
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- -1 PIRROL AMIDES Chemical class 0.000 title 1
- 230000015572 biosynthetic process Effects 0.000 title 1
- 238000003786 synthesis reaction Methods 0.000 title 1
- RLOQBKJCOAXOLR-UHFFFAOYSA-N 1h-pyrrole-2-carboxamide Chemical class NC(=O)C1=CC=CN1 RLOQBKJCOAXOLR-UHFFFAOYSA-N 0.000 abstract 1
- RGHQKFQZGLKBCF-UHFFFAOYSA-N 2-bromoethyl acetate Chemical compound CC(=O)OCCBr RGHQKFQZGLKBCF-UHFFFAOYSA-N 0.000 abstract 1
- QGZKDVFQNNGYKY-UHFFFAOYSA-O Ammonium Chemical compound [NH4+] QGZKDVFQNNGYKY-UHFFFAOYSA-O 0.000 abstract 1
- 102000004300 GABA-A Receptors Human genes 0.000 abstract 1
- 108090000839 GABA-A Receptors Proteins 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 150000004982 aromatic amines Chemical class 0.000 abstract 1
- 150000004820 halides Chemical class 0.000 abstract 1
Landscapes
- Pyrrole Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Un procedimiento para preparar pirrol-carboxamidas que se unen selectivamente a receptores GABA a ; que comprende hacer reaccionar 1,3 -cicloalcanodionas con bromoetilacetato, seguido por la reacción del producto resultante con un haluro de ácido, seguido por la reacción con una amina aromática y, finalmente, con una fuente de amonio a una temperatura elevada.A procedure for preparing pyrrole-carboxamides that selectively bind to GABA a receptors; which comprises reacting 1,3-cycloalkanediones with bromoethylacetate, followed by reaction of the resulting product with an acid halide, followed by reaction with an aromatic amine and, finally, with an ammonium source at an elevated temperature.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP982743 ECSP982743A (en) | 1998-11-13 | 1998-11-13 | PIRROL AMIDES SYNTHESIS PROCEDURES |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP982743 ECSP982743A (en) | 1998-11-13 | 1998-11-13 | PIRROL AMIDES SYNTHESIS PROCEDURES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP982743A true ECSP982743A (en) | 1999-04-16 |
Family
ID=42043662
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP982743 ECSP982743A (en) | 1998-11-13 | 1998-11-13 | PIRROL AMIDES SYNTHESIS PROCEDURES |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP982743A (en) |
-
1998
- 1998-11-13 EC ECSP982743 patent/ECSP982743A/en unknown
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