ECSP992825A - PIPERACINE DERIVATIVES AS NEUROKININ ANTAGONISTS - Google Patents

PIPERACINE DERIVATIVES AS NEUROKININ ANTAGONISTS

Info

Publication number
ECSP992825A
ECSP992825A ECSP992825A ECSP992825A EC SP992825 A ECSP992825 A EC SP992825A EC SP992825 A ECSP992825 A EC SP992825A EC SP992825 A ECSP992825 A EC SP992825A
Authority
EC
Ecuador
Prior art keywords
piperacine
derivatives
neurokinin antagonists
neurokinin
antagonists
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Neng Yang Shih
David Blythin
Ho-Jane Shue
Xiao Chen
Kevin D Mccormick
John J Piwinski
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP992825 priority Critical patent/ECSP992825A/en
Publication of ECSP992825A publication Critical patent/ECSP992825A/en

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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención se refiere a antagonista de neuroquinina de la fórmula (gráfico), donde Z, Rc, y m, u, Ar2, n X, Rc¿, I y Ar2, son según se describe en la presente invención. Estos compuestos son útiles en el tratamiento de enfermedades tales como asma, ansiedad, depresión, émesis y nocicepción.The invention relates to a neuroquinine antagonist of the formula (graph), where Z, Rc, and m, u, Ar2, n X, Rc¿, I and Ar2, are as described in the present invention. These compounds are useful in the treatment of diseases such as asthma, anxiety, depression, emesis, and nociception.

ECSP992825 1999-01-11 1999-01-11 PIPERACINE DERIVATIVES AS NEUROKININ ANTAGONISTS ECSP992825A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP992825 ECSP992825A (en) 1999-01-11 1999-01-11 PIPERACINE DERIVATIVES AS NEUROKININ ANTAGONISTS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP992825 ECSP992825A (en) 1999-01-11 1999-01-11 PIPERACINE DERIVATIVES AS NEUROKININ ANTAGONISTS

Publications (1)

Publication Number Publication Date
ECSP992825A true ECSP992825A (en) 1999-05-17

Family

ID=42043818

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP992825 ECSP992825A (en) 1999-01-11 1999-01-11 PIPERACINE DERIVATIVES AS NEUROKININ ANTAGONISTS

Country Status (1)

Country Link
EC (1) ECSP992825A (en)

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