ECSP992897A - INTEGRIN RECEPTOR ANTAGONISTS - Google Patents
INTEGRIN RECEPTOR ANTAGONISTSInfo
- Publication number
- ECSP992897A ECSP992897A ECSP992897A ECSP992897A EC SP992897 A ECSP992897 A EC SP992897A EC SP992897 A ECSP992897 A EC SP992897A EC SP992897 A ECSP992897 A EC SP992897A
- Authority
- EC
- Ecuador
- Prior art keywords
- receptor antagonists
- integrin receptor
- alpha
- compounds
- present
- Prior art date
Links
- 229940127449 Integrin Receptor Antagonists Drugs 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000002401 inhibitory effect Effects 0.000 abstract 2
- 201000001320 Atherosclerosis Diseases 0.000 abstract 1
- 208000006386 Bone Resorption Diseases 0.000 abstract 1
- 206010012689 Diabetic retinopathy Diseases 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 206010027476 Metastases Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 230000033115 angiogenesis Effects 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 230000024279 bone resorption Effects 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 208000002780 macular degeneration Diseases 0.000 abstract 1
- 230000009401 metastasis Effects 0.000 abstract 1
- 239000002464 receptor antagonist Substances 0.000 abstract 1
- 229940044551 receptor antagonist Drugs 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
- 230000004614 tumor growth Effects 0.000 abstract 1
- 230000002792 vascular Effects 0.000 abstract 1
- 230000003612 virological effect Effects 0.000 abstract 1
- 230000029663 wound healing Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere a compuestos y derivados de los mismos, su sintesis, y su uso como antagonistas del receptor integrina. Más particularmente los compuestos de la presente invención son antagonistas de los receptores integrina alfa vB3, alfa v b5, y/o, av b6 y son útiles para inhibir la resorción ósea, tratar y prevenir osteoporosis, e inhibir la resyenosis vascular, retinopatia diabética, degeneración macular, angiogenésis, ateroesclerosis, inflamación, cicatrización de heridas, enfermedad viral y crecimiento de tumos y metástasis.The present invention relates to compounds and derivatives thereof, their synthesis, and their use as integrin receptor antagonists. More particularly the compounds of the present invention are alpha vB3, alpha v b5, and / or av b6 receptor antagonists and are useful for inhibiting bone resorption, treating and preventing osteoporosis, and inhibiting vascular resyenosis, diabetic retinopathy, macular degeneration, angiogenesis, atherosclerosis, inflammation, wound healing, viral disease, and tumor growth and metastasis.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992897 ECSP992897A (en) | 1999-03-24 | 1999-03-24 | INTEGRIN RECEPTOR ANTAGONISTS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992897 ECSP992897A (en) | 1999-03-24 | 1999-03-24 | INTEGRIN RECEPTOR ANTAGONISTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP992897A true ECSP992897A (en) | 1999-06-01 |
Family
ID=42043885
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP992897 ECSP992897A (en) | 1999-03-24 | 1999-03-24 | INTEGRIN RECEPTOR ANTAGONISTS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP992897A (en) |
-
1999
- 1999-03-24 EC ECSP992897 patent/ECSP992897A/en unknown
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