ECSP992901A - 2- METHYL-THYENE BENZODIAZEPINE FORMULATION - Google Patents
2- METHYL-THYENE BENZODIAZEPINE FORMULATIONInfo
- Publication number
- ECSP992901A ECSP992901A ECSP992901A ECSP992901A EC SP992901 A ECSP992901 A EC SP992901A EC SP992901 A ECSP992901 A EC SP992901A EC SP992901 A ECSP992901 A EC SP992901A
- Authority
- EC
- Ecuador
- Prior art keywords
- thyene
- methyl
- formulation
- olanzapine
- benzodiazepine formulation
- Prior art date
Links
- 238000009472 formulation Methods 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title abstract 2
- SVUOLADPCWQTTE-UHFFFAOYSA-N 1h-1,2-benzodiazepine Chemical compound N1N=CC=CC2=CC=CC=C12 SVUOLADPCWQTTE-UHFFFAOYSA-N 0.000 title 1
- 229940049706 benzodiazepine Drugs 0.000 title 1
- HVYWMOMLDIMFJA-DPAQBDIFSA-N cholesterol Chemical compound C1C=C2C[C@@H](O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H]([C@H](C)CCCC(C)C)[C@@]1(C)CC2 HVYWMOMLDIMFJA-DPAQBDIFSA-N 0.000 abstract 2
- 229960005017 olanzapine Drugs 0.000 abstract 2
- KVWDHTXUZHCGIO-UHFFFAOYSA-N olanzapine Chemical compound C1CN(C)CCN1C1=NC2=CC=CC=C2NC2=C1C=C(C)S2 KVWDHTXUZHCGIO-UHFFFAOYSA-N 0.000 abstract 2
- 239000012453 solvate Substances 0.000 abstract 2
- IUDQMMSLVSVGDZ-UHFFFAOYSA-N chembl1201741 Chemical compound C1CN(C)CCN1C1=NC2=CC=CC=C2NC2=C1C=C(C)S2.C1=CC=C2C(CC=3C4=CC=CC=C4C=C(C=3O)C(=O)O)=C(O)C(C(O)=O)=CC2=C1 IUDQMMSLVSVGDZ-UHFFFAOYSA-N 0.000 abstract 1
- 235000012000 cholesterol Nutrition 0.000 abstract 1
- 239000004005 microsphere Substances 0.000 abstract 1
- 229960001072 olanzapine pamoate Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La invención proporciona una formulación de olanzapina o pamoato de olanzapina, o de sus solvatos, en forma de microesferas oleaginosas o de colesterol farmacéuticamente aceptables. La invención también proporciona además nuevas sales pamoato de olanzapina o sus solvatos.The invention provides a formulation of olanzapine or olanzapine pamoate, or its solvates, in the form of pharmaceutically acceptable cholesterol or oil microspheres. The invention also further provides novel pamoate salts of olanzapine or its solvates.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992901 ECSP992901A (en) | 1999-03-30 | 1999-03-30 | 2- METHYL-THYENE BENZODIAZEPINE FORMULATION |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992901 ECSP992901A (en) | 1999-03-30 | 1999-03-30 | 2- METHYL-THYENE BENZODIAZEPINE FORMULATION |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP992901A true ECSP992901A (en) | 1999-10-29 |
Family
ID=42043889
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP992901 ECSP992901A (en) | 1999-03-30 | 1999-03-30 | 2- METHYL-THYENE BENZODIAZEPINE FORMULATION |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP992901A (en) |
-
1999
- 1999-03-30 EC ECSP992901 patent/ECSP992901A/en unknown
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