ECSP992927A - SUBSTITUTED TRICYCLIC COMPOUNDS (CASE X-12143A) - Google Patents
SUBSTITUTED TRICYCLIC COMPOUNDS (CASE X-12143A)Info
- Publication number
- ECSP992927A ECSP992927A ECSP992927A ECSP992927A EC SP992927 A ECSP992927 A EC SP992927A EC SP992927 A ECSP992927 A EC SP992927A EC SP992927 A ECSP992927 A EC SP992927A
- Authority
- EC
- Ecuador
- Prior art keywords
- case
- tricyclic compounds
- substituted tricyclic
- compounds
- substituted
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- UUZURPUIMYJOIL-JNRWAQIZSA-N (2s)-n-[(2s)-1-[[(2s)-1-[(2s)-2-[[(2s)-1-[[(2s)-1-amino-4-methylsulfanyl-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-5-oxopyrrolidine-2-carboxamide Chemical compound CSCC[C@@H](C(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CC=1C=CC=CC=1)NC(=O)[C@H]1NC(=O)CC1)CC1=CC=CC=C1 UUZURPUIMYJOIL-JNRWAQIZSA-N 0.000 abstract 1
- 102000005473 Secretory Phospholipases A2 Human genes 0.000 abstract 1
- 108010031873 Secretory Phospholipases A2 Proteins 0.000 abstract 1
- 235000014113 dietary fatty acids Nutrition 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 229930195729 fatty acid Natural products 0.000 abstract 1
- 239000000194 fatty acid Substances 0.000 abstract 1
- 150000004665 fatty acids Chemical class 0.000 abstract 1
- 108010052031 septide Proteins 0.000 abstract 1
- 230000035939 shock Effects 0.000 abstract 1
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Se describen nuevos compuestos triciclicos junto con el uso de tales compuestos para inhibir la liberación de ácidos grasos inducida por sPLA2 para el tratamiento de trastornos como el choque séptido.Novel tricyclic compounds are described in conjunction with the use of such compounds to inhibit sPLA2-induced fatty acid release for the treatment of disorders such as septide shock.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992927 ECSP992927A (en) | 1999-04-16 | 1999-04-16 | SUBSTITUTED TRICYCLIC COMPOUNDS (CASE X-12143A) |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992927 ECSP992927A (en) | 1999-04-16 | 1999-04-16 | SUBSTITUTED TRICYCLIC COMPOUNDS (CASE X-12143A) |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP992927A true ECSP992927A (en) | 2000-01-27 |
Family
ID=42043917
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP992927 ECSP992927A (en) | 1999-04-16 | 1999-04-16 | SUBSTITUTED TRICYCLIC COMPOUNDS (CASE X-12143A) |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP992927A (en) |
-
1999
- 1999-04-16 EC ECSP992927 patent/ECSP992927A/en unknown
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