ECSP992964A - PYROLEUM COMPOUND (2,3 -d) PIRIMIDE - Google Patents
PYROLEUM COMPOUND (2,3 -d) PIRIMIDEInfo
- Publication number
- ECSP992964A ECSP992964A ECSP992964A ECSP992964A EC SP992964 A ECSP992964 A EC SP992964A EC SP992964 A ECSP992964 A EC SP992964A EC SP992964 A ECSP992964 A EC SP992964A
- Authority
- EC
- Ecuador
- Prior art keywords
- compound
- diabetes
- disease
- pyroleum
- pirimide
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 208000024827 Alzheimer disease Diseases 0.000 abstract 1
- 206010009900 Colitis ulcerative Diseases 0.000 abstract 1
- 208000011231 Crohn disease Diseases 0.000 abstract 1
- 206010012438 Dermatitis atopic Diseases 0.000 abstract 1
- 102000006500 Janus Kinase 3 Human genes 0.000 abstract 1
- 108010019421 Janus Kinase 3 Proteins 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000004022 Protein-Tyrosine Kinases Human genes 0.000 abstract 1
- 108090000412 Protein-Tyrosine Kinases Proteins 0.000 abstract 1
- 201000004681 Psoriasis Diseases 0.000 abstract 1
- 208000024799 Thyroid disease Diseases 0.000 abstract 1
- 206010067584 Type 1 diabetes mellitus Diseases 0.000 abstract 1
- 201000006704 Ulcerative Colitis Diseases 0.000 abstract 1
- 208000006673 asthma Diseases 0.000 abstract 1
- 201000008937 atopic dermatitis Diseases 0.000 abstract 1
- 230000001363 autoimmune Effects 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 229940125721 immunosuppressive agent Drugs 0.000 abstract 1
- 239000003018 immunosuppressive agent Substances 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 208000032839 leukemia Diseases 0.000 abstract 1
- 206010025135 lupus erythematosus Diseases 0.000 abstract 1
- 201000006417 multiple sclerosis Diseases 0.000 abstract 1
- 210000000056 organ Anatomy 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
- 238000002054 transplantation Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Un compuesto de fórmula (gráfico), en la que R1, R2 y R3 son como se han definido antes, que son inhibidores de las enzimas proteínas tirosina quinasas, como Janus Quinasa 3 y, como tales, son una terapia útil como agentes inmunosupresores para el transplante de órganos, lupus, esclerosis múltiple, artritis reumatoide, psoriasis, diabetes tipo I y complicaciones de la diabetes, cáncer, asma, dermatitis atópica, trastornos autinmunes de tiroides, colitis ulcerosa, enfermedad de Crohn, enfermedad de Alzheimer, leucemia y otras enfermedades outoinmunes.A compound of formula (graph), in which R1, R2 and R3 are as defined above, that they are inhibitors of protein tyrosine kinase enzymes, such as Janus Kinase 3 and, as such, are useful therapy as immunosuppressive agents for organ transplantation, lupus, multiple sclerosis, rheumatoid arthritis, psoriasis, type I diabetes and complications of diabetes, cancer, asthma, atopic dermatitis, autoimmune thyroid disorders, ulcerative colitis, Crohn's disease, Alzheimer's disease, leukemia and others outoimmune diseases.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992964 ECSP992964A (en) | 1999-05-26 | 1999-05-26 | PYROLEUM COMPOUND (2,3 -d) PIRIMIDE |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992964 ECSP992964A (en) | 1999-05-26 | 1999-05-26 | PYROLEUM COMPOUND (2,3 -d) PIRIMIDE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP992964A true ECSP992964A (en) | 1999-07-08 |
Family
ID=42043953
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP992964 ECSP992964A (en) | 1999-05-26 | 1999-05-26 | PYROLEUM COMPOUND (2,3 -d) PIRIMIDE |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP992964A (en) |
-
1999
- 1999-05-26 EC ECSP992964 patent/ECSP992964A/en unknown
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