ECSP992984A - ISOTIAZOLE DERIVATIVES USEFUL AS ANTI-CANCER AGENTS - Google Patents
ISOTIAZOLE DERIVATIVES USEFUL AS ANTI-CANCER AGENTSInfo
- Publication number
- ECSP992984A ECSP992984A ECSP992984A ECSP992984A EC SP992984 A ECSP992984 A EC SP992984A EC SP992984 A ECSP992984 A EC SP992984A EC SP992984 A ECSP992984 A EC SP992984A
- Authority
- EC
- Ecuador
- Prior art keywords
- isotiazole
- cancer agents
- derivatives useful
- relates
- compounds
- Prior art date
Links
- 239000002246 antineoplastic agent Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 241000124008 Mammalia Species 0.000 abstract 1
- 230000003463 hyperproliferative effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere a compuestos de fórmula I, (gráfico), y a sales farmacéuticamente aceptables, profármacos y solvatos de los mismos, en los que X1, R1, R2 y R3 son como se han definido en la presente. La invención también se refiere a composiciones farmacéuticas que contienen los compuestos anteriores y a procedimientos de tratamiento de trastornos hiperproliferativos en mamíferos mediante la administarción de los compuestos anteriores.The present invention relates to compounds of formula I, (graph), and to pharmaceutically acceptable salts, prodrugs, and solvates thereof, wherein X1, R1, R2, and R3 are as defined herein. The invention also relates to pharmaceutical compositions containing the above compounds and to methods of treating hyperproliferative disorders in mammals by administering the above compounds.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992984 ECSP992984A (en) | 1999-06-04 | 1999-06-04 | ISOTIAZOLE DERIVATIVES USEFUL AS ANTI-CANCER AGENTS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP992984 ECSP992984A (en) | 1999-06-04 | 1999-06-04 | ISOTIAZOLE DERIVATIVES USEFUL AS ANTI-CANCER AGENTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP992984A true ECSP992984A (en) | 1999-08-12 |
Family
ID=42043973
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP992984 ECSP992984A (en) | 1999-06-04 | 1999-06-04 | ISOTIAZOLE DERIVATIVES USEFUL AS ANTI-CANCER AGENTS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP992984A (en) |
-
1999
- 1999-06-04 EC ECSP992984 patent/ECSP992984A/en unknown
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