ECSP993018A - NEW PROTEASE INHIBITORS, PARTICULARLY CYSTEINE AND SERINE PROTEASE INHIBITORS - Google Patents
NEW PROTEASE INHIBITORS, PARTICULARLY CYSTEINE AND SERINE PROTEASE INHIBITORSInfo
- Publication number
- ECSP993018A ECSP993018A ECSP993018A ECSP993018A EC SP993018 A ECSP993018 A EC SP993018A EC SP993018 A ECSP993018 A EC SP993018A EC SP993018 A ECSP993018 A EC SP993018A
- Authority
- EC
- Ecuador
- Prior art keywords
- protease inhibitors
- new
- particularly cysteine
- serine protease
- serine
- Prior art date
Links
- 239000002852 cysteine proteinase inhibitor Substances 0.000 title abstract 2
- XUJNEKJLAYXESH-UHFFFAOYSA-N cysteine Natural products SCC(N)C(O)=O XUJNEKJLAYXESH-UHFFFAOYSA-N 0.000 title 1
- 235000018417 cysteine Nutrition 0.000 title 1
- 229940042399 direct acting antivirals protease inhibitors Drugs 0.000 title 1
- 239000000137 peptide hydrolase inhibitor Substances 0.000 title 1
- 239000003001 serine protease inhibitor Substances 0.000 title 1
- 206010065687 Bone loss Diseases 0.000 abstract 1
- 102000004171 Cathepsin K Human genes 0.000 abstract 1
- 108090000625 Cathepsin K Proteins 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Esta invención se refiere a compuestos de fórmula (I), (gráfico), o una sal farmacéuticamente aceptable de los mismos, que son inhibidores de cisteína-proteasas, particularmente catepsina K, y son útiles en el tratamiento de enfermedades en las que la inhibición de pérdida de hueso es un factor.This invention relates to compounds of formula (I), (graph), or a pharmaceutically acceptable salt thereof, which are cysteine protease inhibitors, particularly cathepsin K, and are useful in the treatment of diseases in which inhibition bone loss is a factor.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP993018 ECSP993018A (en) | 1999-06-10 | 1999-06-10 | NEW PROTEASE INHIBITORS, PARTICULARLY CYSTEINE AND SERINE PROTEASE INHIBITORS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP993018 ECSP993018A (en) | 1999-06-10 | 1999-06-10 | NEW PROTEASE INHIBITORS, PARTICULARLY CYSTEINE AND SERINE PROTEASE INHIBITORS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP993018A true ECSP993018A (en) | 1999-11-29 |
Family
ID=42044007
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP993018 ECSP993018A (en) | 1999-06-10 | 1999-06-10 | NEW PROTEASE INHIBITORS, PARTICULARLY CYSTEINE AND SERINE PROTEASE INHIBITORS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP993018A (en) |
-
1999
- 1999-06-10 EC ECSP993018 patent/ECSP993018A/en unknown
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