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Pharmaceuticals Containing Other Organic And Inorganic Compounds
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Medicinal Preparation
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Abstract
Se describen composiciones farmacéuticas que contienen 8-cloro-6,11-dihidro-11-(4-piperidiliden)-5H-benzo[5,6]-ciclohepta[1,2-b]piridina ("DCL") y una cantidad protectora de DCL de una sal básica farmacéuticamente aceptable como ser fosfato dibásico de calcio y una cantidad de por lo menos un desintegrante, preferentemente dos desintegrantes como ser celulosa microcristalina y almidón suficiente para proveer una disolución de por lo menos 80% en peso de la composición farmacéutica en aproximadamente 45 minutos y describe el uso de DCL para preparar una composición farmacéutica para tratar reacciones alérgicas en mamíferos como ser el hombre.Pharmaceutical compositions are described containing 8-chloro-6,11-dihydro-11- (4-piperidiliden) -5H-benzo [5,6] -cyclohepta [1,2-b] pyridine ("DCL") and an amount DCL protector of a pharmaceutically acceptable basic salt such as calcium dibasic phosphate and an amount of at least one disintegrant, preferably two disintegrants such as microcrystalline cellulose and starch sufficient to provide a solution of at least 80% by weight of the composition pharmaceutical in about 45 minutes and describes the use of DCL to prepare a pharmaceutical composition to treat allergic reactions in mammals such as man.
Azabicycloalkanes as CCR5 Modulators, Pharmaceutical Compositions Containing the Same and Their Use for Treatment and Prevention of Diseases Caused by CCR5 Activity
Piperidines as CCR5 Modulators, Pharmaceutical Compositions Containing the Same and Their Use for Treatment and Prevention of Diseases Caused by CCR5 Modulators
Indolylpiperidine derivatives and their use as antihistaminic and antiallergic agents, process for their preparation, pharmaceutical compositions containing them