EE03090B1 - Kinoliin-3-karboksamiidühendite kasutamine kompositsiooni valmistamiseks I tüüpi suhkurtõve raviks - Google Patents

Kinoliin-3-karboksamiidühendite kasutamine kompositsiooni valmistamiseks I tüüpi suhkurtõve raviks

Info

Publication number
EE03090B1
EE03090B1 EE9400269A EE9400269A EE03090B1 EE 03090 B1 EE03090 B1 EE 03090B1 EE 9400269 A EE9400269 A EE 9400269A EE 9400269 A EE9400269 A EE 9400269A EE 03090 B1 EE03090 B1 EE 03090B1
Authority
EE
Estonia
Prior art keywords
quinoline
diabetes
preparation
treatment
composition
Prior art date
Application number
EE9400269A
Other languages
English (en)
Inventor
Slavin Shimon
Weiss Lola
Gross David
Original Assignee
Pharmacia & Upjohn Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Ab filed Critical Pharmacia & Upjohn Ab
Publication of EE03090B1 publication Critical patent/EE03090B1/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
EE9400269A 1992-04-06 1994-11-17 Kinoliin-3-karboksamiidühendite kasutamine kompositsiooni valmistamiseks I tüüpi suhkurtõve raviks EE03090B1 (et)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9201076A SE9201076L (sv) 1992-04-06 1992-04-06 Användningen av gamla läkemedel för behandling av diabetes

Publications (1)

Publication Number Publication Date
EE03090B1 true EE03090B1 (et) 1998-06-15

Family

ID=20385863

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9400269A EE03090B1 (et) 1992-04-06 1994-11-17 Kinoliin-3-karboksamiidühendite kasutamine kompositsiooni valmistamiseks I tüüpi suhkurtõve raviks

Country Status (16)

Country Link
US (1) US5594005A (et)
EP (1) EP0634931A1 (et)
JP (1) JPH07506568A (et)
KR (1) KR950700738A (et)
CN (1) CN1081671A (et)
AU (1) AU667362B2 (et)
CA (1) CA2131831C (et)
EE (1) EE03090B1 (et)
HU (1) HUT69710A (et)
IL (1) IL105285A0 (et)
NO (1) NO943723L (et)
NZ (1) NZ251494A (et)
PH (1) PH30820A (et)
SE (1) SE9201076L (et)
WO (1) WO1993019756A1 (et)
ZA (1) ZA932450B (et)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6133285A (en) * 1998-07-15 2000-10-17 Active Biotech Ab Quinoline derivatives
SE9802550D0 (sv) * 1998-07-15 1998-07-15 Active Biotech Ab Quinoline derivatives
SE9802549D0 (sv) * 1998-07-15 1998-07-15 Active Biotech Ab Quinoline derivatives
FR2827600A1 (fr) * 2001-07-20 2003-01-24 Lipha Derives acides de quinolone et leurs applications en therapeutique
US8124582B2 (en) * 2002-12-06 2012-02-28 Fibrogen, Inc. Treatment of diabetes
JP5619752B2 (ja) * 2008-10-09 2014-11-05 ニュートゥリー カンパニーリミテッド パンドラチン誘導体またはボエセンベルギアパンドラタ抽出物の新規な用途
WO2012050500A1 (en) 2010-10-14 2012-04-19 Lars Pettersson 1,2-dihydro-4-hydroxy-2-oxo-quinoline-3-carboxanilides as ahr activators.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1034124A (en) * 1973-05-11 1978-07-04 Ciba-Geigy Ag Process for the manufacture of new quinolines
FR2340735A1 (fr) * 1976-02-11 1977-09-09 Roussel Uclaf Nouveaux derives de l'acide 3-quinoleine carboxylique, leur procede de preparation et leur application comme medicament
IE52670B1 (en) * 1981-03-03 1988-01-20 Leo Ab Heterocyclic carboxamides,compositions containing such compounds,and processes for their preparation
DE3134780A1 (de) * 1981-09-02 1983-03-10 Hoechst Ag, 6000 Frankfurt "sulfonylharnstoffe, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen und ihre verwendung"
US5310913A (en) * 1989-06-09 1994-05-10 Kabi Pharmacia Aktiebolag Derivatives of quinoline-3-carboxanilide
SE9000624D0 (sv) * 1990-02-22 1990-02-22 Pharmacia Ab New use
SE9001111D0 (sv) * 1990-03-27 1990-03-27 Pharmacia Ab Supportive use

Also Published As

Publication number Publication date
ZA932450B (en) 1993-10-20
SE9201076L (sv) 1993-10-07
AU3913193A (en) 1993-11-08
IL105285A0 (en) 1993-08-18
CA2131831C (en) 1999-03-09
WO1993019756A1 (en) 1993-10-14
CA2131831A1 (en) 1993-10-14
NO943723D0 (no) 1994-10-05
AU667362B2 (en) 1996-03-21
HUT69710A (en) 1995-09-28
EP0634931A1 (en) 1995-01-25
PH30820A (en) 1997-10-17
KR950700738A (ko) 1995-02-20
HU9402854D0 (en) 1995-01-30
JPH07506568A (ja) 1995-07-20
NO943723L (no) 1994-10-05
SE9201076D0 (sv) 1992-04-06
NZ251494A (en) 1997-07-27
CN1081671A (zh) 1994-02-09
US5594005A (en) 1997-01-14

Similar Documents

Publication Publication Date Title
FI951413A7 (fi) Pintakäsittelykoostumus
FI930747A7 (fi) Heterosyklisiä yhdisteitä ja niiden valmistus ja käyttö
FI903215A7 (fi) Heteroaryyliamino- ja heteroaryylioksipyridiiniamiineja ja niihin liittyviä yhdisteitä, menetelmä niiden valmistamiseksi sekä niiden käyttö lääkkeinä
FI931901A7 (fi) Atsoliyhdisteet, niiden valmistus ja käyttö
FI945281A7 (fi) Heterosykliset yhdisteet, niiden valmistus ja käyttö
FI925661L (fi) Injicerbar farmaceutisk komposition
FI914419A7 (fi) Uusia insuliiniyhdisteitä
FI930656A7 (fi) Nasaalihoitoon tarkoitettu koostumus
FI910310A7 (fi) Asesulfaami-K:ta sisältävä koostumus
FI935887L (fi) Tiatzolidiinidionijohdannaiset, niiden valmistus ja käyttö
DK90089A (da) Hudbehandlingspraeparat
FI930746A7 (fi) Heterosyklisiä yhdisteitä ja niiden valmistus ja käyttö
FI943313A7 (fi) Heterosykliset yhdisteet ja niiden valmistus ja käyttö
FI942963A7 (fi) Imidatsokinatsoliiniyhdisteitä ja niiden valmistus ja käyttö
EE9400257A (et) Kinoliin-3-karboksamiidi ühendi kasutamine ravimkompositsiooni valmistamiseks
EE03090B1 (et) Kinoliin-3-karboksamiidühendite kasutamine kompositsiooni valmistamiseks I tüüpi suhkurtõve raviks
UA26064A1 (uk) Фармацевтичhа композиція
FI946057L (fi) Paikalliseen käyttöön tarkoitettu valmiste
DE69323607D1 (de) Flüssige korrekturzusammensetzung
FI935654A7 (fi) Kondensoituneet heterosykliset yhdisteet, niiden valmistus ja käyttö
FI911644A7 (fi) Terapeuttinen yhdiste ja koostumus
KR930702465A (ko) 카르복시에스테르 복합체를 함유하는 액체 조성물
FI915979A7 (fi) Fenyylialkyyliaminoalkyyliyhdisteet sekä menetelmät niiden valmistamiseksi ja näitä yhdisteitä sisältävät lääkeaineet
FI914525A7 (fi) Yhdiste, käyttö ja valmistus
FI950050L (fi) (S)-timololihemihydraattia sisältävä oftalminen tooppinen koostumus