EE9800309A - Uued asendatud tsüklilised aminohapped kui farmatseutilised toimeained - Google Patents

Uued asendatud tsüklilised aminohapped kui farmatseutilised toimeained

Info

Publication number
EE9800309A
EE9800309A EE9800309A EE9800309A EE9800309A EE 9800309 A EE9800309 A EE 9800309A EE 9800309 A EE9800309 A EE 9800309A EE 9800309 A EE9800309 A EE 9800309A EE 9800309 A EE9800309 A EE 9800309A
Authority
EE
Estonia
Prior art keywords
amino acids
cyclic amino
pct
active agents
pharmaceutically active
Prior art date
Application number
EE9800309A
Other languages
English (en)
Inventor
Stephen Bryans Justin
Octavia Kneen Clare
Stuart Ratcliffe Giles
Christopher Horwell David
Ian Morrell Andrew
Hartenstein Johannes
Original Assignee
Warner-Lambert Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner-Lambert Company filed Critical Warner-Lambert Company
Publication of EE9800309A publication Critical patent/EE9800309A/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/47—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A61P25/12—Antiepileptics; Anticonvulsants for grand-mal
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/28—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and containing rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Peptides Or Proteins (AREA)
EE9800309A 1996-03-14 1997-02-18 Uued asendatud tsüklilised aminohapped kui farmatseutilised toimeained EE9800309A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1343296P 1996-03-14 1996-03-14
PCT/US1997/002295 WO1997033858A1 (en) 1996-03-14 1997-02-18 Novel substituted cyclic amino acids as pharmaceutical agents

Publications (1)

Publication Number Publication Date
EE9800309A true EE9800309A (et) 1999-02-15

Family

ID=21759938

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9800309A EE9800309A (et) 1996-03-14 1997-02-18 Uued asendatud tsüklilised aminohapped kui farmatseutilised toimeained

Country Status (29)

Country Link
US (1) US6103932A (et)
EP (1) EP0888286B1 (et)
JP (1) JP2000506861A (et)
KR (1) KR100512506B1 (et)
AT (1) ATE207878T1 (et)
AU (1) AU734173B2 (et)
BG (1) BG63662B1 (et)
BR (1) BR9708200A (et)
CA (1) CA2244912C (et)
CZ (1) CZ293759B6 (et)
DE (1) DE69707842T2 (et)
DK (2) DK0888286T3 (et)
EA (1) EA002765B1 (et)
EE (1) EE9800309A (et)
ES (1) ES2167717T3 (et)
GE (1) GEP20012413B (et)
HU (1) HU224720B1 (et)
IL (1) IL125544A (et)
IS (1) IS1990B (et)
MX (1) MX9806069A (et)
NO (1) NO984205L (et)
NZ (1) NZ331143A (et)
PL (1) PL185991B1 (et)
PT (1) PT888286E (et)
SK (1) SK283295B6 (et)
TR (1) TR199801807T2 (et)
UA (1) UA49011C2 (et)
WO (1) WO1997033858A1 (et)
ZA (1) ZA972200B (et)

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US6984659B2 (en) 1997-11-18 2006-01-10 Klinikum Der Albert-Ludwigs Universitaet 2-pyrrolidinone derivatives substituted at position 4 for reducing the extracellular glutamate level
DE19751062A1 (de) 1997-11-18 1999-07-08 Univ Ludwigs Albert An 4-Stellung substituierte 2-Pyrrolidinon-Derivate zur Verringerung des extrazellulären Glutamat-Spiegels
WO1999031075A1 (en) * 1997-12-16 1999-06-24 Warner-Lambert Company 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
JP2002520286A (ja) * 1998-07-09 2002-07-09 ワーナー−ランバート・カンパニー Ｇａｂａ類縁体及びカフェインを含んでなる組成物
EP1031350A1 (en) * 1999-02-23 2000-08-30 Warner-Lambert Company Use of a gabapentin-analog for the manufacture of a medicament for preventing and treating visceral pain
US6992109B1 (en) * 1999-04-08 2006-01-31 Segal Catherine A Method for the treatment of incontinence
CZ20012758A3 (cs) * 1999-12-08 2002-09-11 Warner-Lambert Company Větvené aminokyselinově dependentní aminotransferasové inhibitory a jejich použití při léčení diabetické retinopatie
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GB2362646A (en) * 2000-05-26 2001-11-28 Warner Lambert Co Cyclic amino acid derivatives useful as pharmaceutical agents
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Also Published As

Publication number Publication date
BG63662B1 (bg) 2002-08-30
EP0888286B1 (en) 2001-10-31
IS4819A (is) 1998-08-10
DK0888285T3 (da) 2002-04-08
AU734173B2 (en) 2001-06-07
BR9708200A (pt) 1999-07-27
IS1990B (is) 2005-02-15
HUP9902136A3 (en) 2000-03-28
WO1997033858A1 (en) 1997-09-18
PL328816A1 (en) 1999-02-15
ZA972200B (en) 1997-09-17
CA2244912C (en) 2005-07-12
SK283295B6 (sk) 2003-05-02
UA49011C2 (uk) 2002-09-16
MX9806069A (es) 1998-11-30
AU2051197A (en) 1997-10-01
IL125544A0 (en) 1999-03-12
EP0888286A1 (en) 1999-01-07
NZ331143A (en) 2001-06-29
DE69707842T2 (de) 2002-05-16
KR19990087756A (ko) 1999-12-27
US6103932A (en) 2000-08-15
HU224720B1 (en) 2006-01-30
JP2000506861A (ja) 2000-06-06
BG102733A (en) 1999-04-30
PT888286E (pt) 2002-04-29
NO984205L (no) 1998-09-14
KR100512506B1 (ko) 2005-12-21
ATE207878T1 (de) 2001-11-15
TR199801807T2 (xx) 1998-12-21
EA199800798A1 (ru) 1999-04-29
CA2244912A1 (en) 1997-09-18
HUP9902136A2 (hu) 1999-10-28
ES2167717T3 (es) 2002-05-16
PL185991B1 (pl) 2003-09-30
EA002765B1 (ru) 2002-08-29
DE69707842D1 (de) 2001-12-06
SK123898A3 (en) 2000-04-10
GEP20012413B (en) 2001-04-25
CZ293759B6 (cs) 2004-07-14
CZ286398A3 (cs) 1999-03-17
DK0888286T3 (da) 2002-02-18
IL125544A (en) 2002-03-10
NO984205D0 (no) 1998-09-11

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