EP0738155A4 - Structure et synthese modulaire de molecules derivees de l'oxazolone - Google Patents
Structure et synthese modulaire de molecules derivees de l'oxazoloneInfo
- Publication number
- EP0738155A4 EP0738155A4 EP94907107A EP94907107A EP0738155A4 EP 0738155 A4 EP0738155 A4 EP 0738155A4 EP 94907107 A EP94907107 A EP 94907107A EP 94907107 A EP94907107 A EP 94907107A EP 0738155 A4 EP0738155 A4 EP 0738155A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- oxazolone
- synthesis
- modular structure
- derived molecules
- molecules
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
- C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids
- C07H13/04—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals attached to acyclic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/36—One oxygen atom
- C07D263/42—One oxygen atom attached in position 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
- C07K1/047—Simultaneous synthesis of different peptide species; Peptide libraries
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/005—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from viruses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12N—MICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
- C12N2740/00—Reverse transcribing RNA viruses
- C12N2740/00011—Details
- C12N2740/10011—Retroviridae
- C12N2740/16011—Human Immunodeficiency Virus, HIV
- C12N2740/16111—Human Immunodeficiency Virus, HIV concerning HIV env
- C12N2740/16122—New viral proteins or individual genes, new structural or functional aspects of known viral proteins or genes
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Engineering & Computer Science (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Biophysics (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Psychiatry (AREA)
- Biotechnology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Gastroenterology & Hepatology (AREA)
- Pain & Pain Management (AREA)
- Analytical Chemistry (AREA)
- Saccharide Compounds (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Furan Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/US1993/012591 WO1995017903A1 (fr) | 1993-12-28 | 1993-12-28 | Structure et synthese modulaire de molecules derivees de l'oxazolone |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EP0738155A1 EP0738155A1 (fr) | 1996-10-23 |
| EP0738155A4 true EP0738155A4 (fr) | 1997-03-19 |
Family
ID=22237332
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP94907107A Withdrawn EP0738155A4 (fr) | 1993-12-28 | 1993-12-28 | Structure et synthese modulaire de molecules derivees de l'oxazolone |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP0738155A4 (fr) |
| JP (1) | JPH09511225A (fr) |
| AU (1) | AU6049994A (fr) |
| WO (1) | WO1995017903A1 (fr) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU704878B2 (en) * | 1994-01-05 | 1999-05-06 | Arqule, Inc. | Method of making polymers having specific properties |
| US5712171A (en) | 1995-01-20 | 1998-01-27 | Arqule, Inc. | Method of generating a plurality of chemical compounds in a spatially arranged array |
| US6355641B1 (en) | 1999-03-17 | 2002-03-12 | Syntex (U.S.A.) Llc | Oxazolone derivatives and uses thereof |
| US7074961B2 (en) | 2000-09-26 | 2006-07-11 | The Brigham And Women's Hospital, Inc. | Antidepressants and their analogues as long-acting local anesthetics and analgesics |
| WO2002026020A2 (fr) | 2000-09-26 | 2002-04-04 | The Brigham And Women's Hospital, Inc. | Antidepresseurs tricycliques et leurs analogues comme anesthesiques et analgesiques locaux de longue duree |
| JP4556473B2 (ja) * | 2003-10-17 | 2010-10-06 | 株式会社島津製作所 | タンパク質又はペプチドのc末端を修飾する方法 |
| EP4301765A4 (fr) * | 2021-03-03 | 2025-03-12 | Emergent Product Development Gaithersburg Inc. | Dérivés de valiolamine en tant qu'inhibiteurs de la glucosidase |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0433034A2 (fr) * | 1989-12-12 | 1991-06-19 | Minnesota Mining And Manufacturing Company | Méthode impliquant liaisons alpha-amidoacétyles ou béta-amidopropionyles thermosensibles |
| EP0449488A1 (fr) * | 1990-03-28 | 1991-10-02 | Minnesota Mining And Manufacturing Company | Produits d'addition Michael des azlactones |
| WO1994000509A1 (fr) * | 1992-06-30 | 1994-01-06 | Legomer Partners, L.P. | Matieres derivees d'oxazolone |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5182366A (en) * | 1990-05-15 | 1993-01-26 | Huebner Verena D | Controlled synthesis of peptide mixtures using mixed resins |
| US5219731A (en) * | 1991-11-01 | 1993-06-15 | Wisconsin Alumni Research Foundation | Method for preparing optically-active amino acid derivatives |
-
1993
- 1993-12-28 WO PCT/US1993/012591 patent/WO1995017903A1/fr not_active Ceased
- 1993-12-28 AU AU60499/94A patent/AU6049994A/en not_active Abandoned
- 1993-12-28 EP EP94907107A patent/EP0738155A4/fr not_active Withdrawn
- 1993-12-28 JP JP7517993A patent/JPH09511225A/ja active Pending
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0433034A2 (fr) * | 1989-12-12 | 1991-06-19 | Minnesota Mining And Manufacturing Company | Méthode impliquant liaisons alpha-amidoacétyles ou béta-amidopropionyles thermosensibles |
| EP0449488A1 (fr) * | 1990-03-28 | 1991-10-02 | Minnesota Mining And Manufacturing Company | Produits d'addition Michael des azlactones |
| WO1994000509A1 (fr) * | 1992-06-30 | 1994-01-06 | Legomer Partners, L.P. | Matieres derivees d'oxazolone |
Non-Patent Citations (1)
| Title |
|---|
| See also references of WO9517903A1 * |
Also Published As
| Publication number | Publication date |
|---|---|
| WO1995017903A1 (fr) | 1995-07-06 |
| JPH09511225A (ja) | 1997-11-11 |
| AU6049994A (en) | 1995-07-17 |
| EP0738155A1 (fr) | 1996-10-23 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EP0868403A4 (fr) | Synthese de phases "312" et leurs composites | |
| EP0854878A4 (fr) | Synthese de glycoconjugues de l'epitope y de lewis et leurs utilisations | |
| EP0746301A4 (fr) | Compositions cosmetiques autobronzantes et procede d'utilisation desdites compositions | |
| NO933198D0 (no) | Forbindelser anvendelige som hypoglycemiske midler og forbehandling av Alzheimer's sykdom | |
| FI951356A7 (fi) | N-substituoitujen oligomeerien synteesi | |
| NO933240L (no) | Anordning ved og fremstilling av tannbörste | |
| DE69416220D1 (de) | Synthese von festen Lösungen von Chinacridonpigmenten | |
| FI954541L (fi) | Keratinosyyttikasvutekijän terapeuttisia käyttöjä | |
| FI923911A7 (fi) | DNA-molekyylien in vitro-synteesi | |
| FI945705A7 (fi) | Bisindolyylimaleimidien parannettu synteesi | |
| ATA178394A (de) | Verbindungs- und befestigungsorgan | |
| PT744437E (pt) | Misturas de compostos de organossilano e sua utilizacao | |
| EP0826033A4 (fr) | Gene de l'ataxie-telangiectasie | |
| EP0737232A4 (fr) | Structure et synthese modulaire de molecules contenant l'aminimide | |
| FR2731885B1 (fr) | Installation d'etageres demontables | |
| EP0727959A4 (fr) | Utilisations diagnostiques d'hydrozinoadenosines | |
| EP0738155A4 (fr) | Structure et synthese modulaire de molecules derivees de l'oxazolone | |
| DE69410814D1 (de) | Synthese von sphingosinen | |
| DE69603578D1 (de) | Synthese von tetrafluorethylen | |
| FI953736A0 (fi) | I en bastugn anvaendbar foeraongnings och befuktingsanordning | |
| FR2767824B1 (fr) | Synthese d'acides carboxyalkylthiosucciniques | |
| FR2672591B1 (fr) | Synthese d'hydrogeno-perfluoroalcanes. | |
| ITRM940763A0 (it) | Disposizione e metodo di sintesi vocale | |
| FR2741216B1 (fr) | Blindage d'une membrane | |
| AU4341193A (en) | Analysis and synthesis of rhythm |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
| 17P | Request for examination filed |
Effective date: 19960719 |
|
| AK | Designated contracting states |
Kind code of ref document: A1 Designated state(s): AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE |
|
| A4 | Supplementary search report drawn up and despatched |
Effective date: 19970131 |
|
| AK | Designated contracting states |
Kind code of ref document: A4 Designated state(s): AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE |
|
| RAP1 | Party data changed (applicant data changed or rights of an application transferred) |
Owner name: ARQULE, INC. |
|
| STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION HAS BEEN WITHDRAWN |
|
| 18W | Application withdrawn |
Withdrawal date: 20011011 |