EP0784627A4 - METHOD FOR PRODUCING 17-BETA-SUBSTITUTED ANDROSTA-3,5-DIEN-3-CARBONIC ACID - Google Patents

METHOD FOR PRODUCING 17-BETA-SUBSTITUTED ANDROSTA-3,5-DIEN-3-CARBONIC ACID

Info

Publication number
EP0784627A4
EP0784627A4 EP95936242A EP95936242A EP0784627A4 EP 0784627 A4 EP0784627 A4 EP 0784627A4 EP 95936242 A EP95936242 A EP 95936242A EP 95936242 A EP95936242 A EP 95936242A EP 0784627 A4 EP0784627 A4 EP 0784627A4
Authority
EP
European Patent Office
Prior art keywords
dien
beta
producing
carbonic acid
substituted androsta
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP95936242A
Other languages
German (de)
French (fr)
Other versions
EP0784627A1 (en
Inventor
Neil Howard Baine
Michael Anthony Mcguire
Marvin Sungwhan Yu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
SmithKline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB9420063A external-priority patent/GB9420063D0/en
Priority claimed from GBGB9515925.7A external-priority patent/GB9515925D0/en
Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp
Publication of EP0784627A1 publication Critical patent/EP0784627A1/en
Publication of EP0784627A4 publication Critical patent/EP0784627A4/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
EP95936242A 1994-10-05 1995-10-04 METHOD FOR PRODUCING 17-BETA-SUBSTITUTED ANDROSTA-3,5-DIEN-3-CARBONIC ACID Withdrawn EP0784627A4 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB9420063A GB9420063D0 (en) 1994-10-05 1994-10-05 Process
GB9420063 1994-10-05
GBGB9515925.7A GB9515925D0 (en) 1995-08-03 1995-08-03 Process
GB9515925 1995-08-03
PCT/US1995/012710 WO1996011206A1 (en) 1994-10-05 1995-10-04 Process for preparing 17-beta-substituted-androsta-3,5-dien-3-carboxylic acids

Publications (2)

Publication Number Publication Date
EP0784627A1 EP0784627A1 (en) 1997-07-23
EP0784627A4 true EP0784627A4 (en) 1998-05-06

Family

ID=26305742

Family Applications (1)

Application Number Title Priority Date Filing Date
EP95936242A Withdrawn EP0784627A4 (en) 1994-10-05 1995-10-04 METHOD FOR PRODUCING 17-BETA-SUBSTITUTED ANDROSTA-3,5-DIEN-3-CARBONIC ACID

Country Status (4)

Country Link
EP (1) EP0784627A4 (en)
JP (1) JPH10507176A (en)
AU (1) AU3826095A (en)
WO (1) WO1996011206A1 (en)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994011386A1 (en) * 1992-11-18 1994-05-26 Smithkline Beecham Corporation 17-alpha and 17-beta substituted acyl-3-carboxy-3,5-dienes and use in inhibiting 5-alpha-reductase

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4910226A (en) * 1987-04-29 1990-03-20 Smithkline Beckman Corporation Steroid 5-alpha-reductase inhibitors
US5032586A (en) * 1989-08-24 1991-07-16 Smithkline Beecham Corporation 7-keto or hydroxy 3,5-diene steroids as inhibitors of steroid 5-alpha reductase

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994011386A1 (en) * 1992-11-18 1994-05-26 Smithkline Beecham Corporation 17-alpha and 17-beta substituted acyl-3-carboxy-3,5-dienes and use in inhibiting 5-alpha-reductase

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
See also references of WO9611206A1 *

Also Published As

Publication number Publication date
WO1996011206A1 (en) 1996-04-18
EP0784627A1 (en) 1997-07-23
AU3826095A (en) 1996-05-02
JPH10507176A (en) 1998-07-14

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