EP3355889A4 - Diaminopyrimidin-p2x3- und p2x2/3-rezeptor-modulatoren zur verwendung bei der behandlung von husten - Google Patents

Diaminopyrimidin-p2x3- und p2x2/3-rezeptor-modulatoren zur verwendung bei der behandlung von husten Download PDF

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Publication number
EP3355889A4
EP3355889A4 EP16852340.5A EP16852340A EP3355889A4 EP 3355889 A4 EP3355889 A4 EP 3355889A4 EP 16852340 A EP16852340 A EP 16852340A EP 3355889 A4 EP3355889 A4 EP 3355889A4
Authority
EP
European Patent Office
Prior art keywords
diaminopyrimidine
cough
modulators
receptors
treatment
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
EP16852340.5A
Other languages
English (en)
French (fr)
Other versions
EP3355889A1 (de
EP3355889B1 (de
Inventor
Anthony P. FORD
Kathleen Sereda GLAUB
Michael M. KITT
Steven Smith
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Afferent Pharmaceuticals Inc
Original Assignee
Afferent Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Afferent Pharmaceuticals Inc filed Critical Afferent Pharmaceuticals Inc
Priority to EP23155536.8A priority Critical patent/EP4215182A1/de
Priority to HRP20230445TT priority patent/HRP20230445T1/hr
Priority to SI201631686T priority patent/SI3355889T1/sl
Priority to RS20230321A priority patent/RS64155B1/sr
Publication of EP3355889A1 publication Critical patent/EP3355889A1/de
Publication of EP3355889A4 publication Critical patent/EP3355889A4/de
Application granted granted Critical
Publication of EP3355889B1 publication Critical patent/EP3355889B1/de
Priority to HUS2400004C priority patent/HUS2400004I1/hu
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0078Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a nebulizer such as a jet nebulizer, ultrasonic nebulizer, e.g. in the form of aqueous drug solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dispersion Chemistry (AREA)
  • Otolaryngology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Inorganic Chemistry (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
EP16852340.5A 2015-09-29 2016-09-23 Diaminopyrimidin-p2x3- und p2x2/3-rezeptor-modulatoren zur verwendung bei der behandlung von husten Active EP3355889B1 (de)

Priority Applications (5)

Application Number Priority Date Filing Date Title
EP23155536.8A EP4215182A1 (de) 2015-09-29 2016-09-23 Diaminopyrimidin-p2x3- und p2x2/3-rezeptormodulatoren zur verwendung bei der behandlung von husten
HRP20230445TT HRP20230445T1 (hr) 2015-09-29 2016-09-23 Modulatori diaminopirimidin p2x3 i p2x2/3 receptora za primjenu u liječenju kašlja
SI201631686T SI3355889T1 (sl) 2015-09-29 2016-09-23 Modulatorji receptorja diaminopirimidina P2X3 in P2X2/3 za uporabo pri zdravljenju kašlja
RS20230321A RS64155B1 (sr) 2015-09-29 2016-09-23 Diaminopirimidinski modulatori p2x3 i p2x2/3 receptora, za upotrebu u lečenju kašlja
HUS2400004C HUS2400004I1 (hu) 2015-09-29 2024-03-05 Diaminopirimidin-P2X3 és P2X2/3 receptor modulátorok felhasználásra köhögés kezelésében

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562234584P 2015-09-29 2015-09-29
US201662336381P 2016-05-13 2016-05-13
PCT/US2016/053223 WO2017058645A1 (en) 2015-09-29 2016-09-23 Diaminopyrimidine p2x3 and p2x2/3 receptor modulators for use in the treatment of cough

Related Child Applications (1)

Application Number Title Priority Date Filing Date
EP23155536.8A Division EP4215182A1 (de) 2015-09-29 2016-09-23 Diaminopyrimidin-p2x3- und p2x2/3-rezeptormodulatoren zur verwendung bei der behandlung von husten

Publications (3)

Publication Number Publication Date
EP3355889A1 EP3355889A1 (de) 2018-08-08
EP3355889A4 true EP3355889A4 (de) 2019-05-22
EP3355889B1 EP3355889B1 (de) 2023-02-15

Family

ID=58424436

Family Applications (2)

Application Number Title Priority Date Filing Date
EP16852340.5A Active EP3355889B1 (de) 2015-09-29 2016-09-23 Diaminopyrimidin-p2x3- und p2x2/3-rezeptor-modulatoren zur verwendung bei der behandlung von husten
EP23155536.8A Pending EP4215182A1 (de) 2015-09-29 2016-09-23 Diaminopyrimidin-p2x3- und p2x2/3-rezeptormodulatoren zur verwendung bei der behandlung von husten

Family Applications After (1)

Application Number Title Priority Date Filing Date
EP23155536.8A Pending EP4215182A1 (de) 2015-09-29 2016-09-23 Diaminopyrimidin-p2x3- und p2x2/3-rezeptormodulatoren zur verwendung bei der behandlung von husten

Country Status (23)

Country Link
US (3) US11260056B2 (de)
EP (2) EP3355889B1 (de)
JP (1) JP6877441B2 (de)
KR (2) KR20260022473A (de)
AU (1) AU2016330466B2 (de)
CA (1) CA2998742C (de)
CY (2) CY1125963T1 (de)
DK (1) DK3355889T3 (de)
ES (1) ES2942711T3 (de)
FI (2) FI3355889T3 (de)
FR (1) FR24C1010I2 (de)
HR (1) HRP20230445T1 (de)
HU (2) HUE061764T2 (de)
LT (2) LT3355889T (de)
LU (1) LUC00332I2 (de)
MX (1) MX390084B (de)
NL (1) NL301260I2 (de)
NO (1) NO2024009I1 (de)
PL (1) PL3355889T3 (de)
PT (1) PT3355889T (de)
RS (1) RS64155B1 (de)
SI (1) SI3355889T1 (de)
WO (1) WO2017058645A1 (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10676444B2 (en) * 2016-12-20 2020-06-09 Afferent Pharmaceuticals, Inc. Crystalline salts and polymorphs of a P2X3 antagonist
US10111883B1 (en) * 2017-09-18 2018-10-30 Bellus Health Cough Inc. Selective P2X3 modulators
KR20210009341A (ko) * 2018-05-15 2021-01-26 바이엘 악티엔게젤샤프트 신경 섬유 감작과 연관된 질환의 치료를 위한 1,3-티아졸-2-일 치환된 벤즈아미드
PL3862000T3 (pl) 2018-10-05 2024-03-18 Shionogi & Co., Ltd Lek na przewlekły kaszel
WO2020174283A1 (en) 2019-02-25 2020-09-03 Bellus Health Cough Inc. Treatment with p2x3 modulators
SG11202111877TA (en) * 2019-04-30 2021-11-29 Beijing Tide Pharmaceutical Co Ltd Method for treating cough by using diaminopyrimidine compound
BR112021021738A2 (pt) 2019-05-31 2021-12-28 Chiesi Farm Spa Derivados de amino quinazolina como inibidores de p2x3
MX2021014116A (es) 2019-05-31 2021-12-10 Chiesi Farm Spa Derivados de piridopirimidinas como inhibidores del purinoreceptor 3 de p2x (p2x3).
US12312327B2 (en) 2019-09-19 2025-05-27 Shionogi & Co., Ltd. Crystal of 1,3,5-triazine derivative or solvate thereof and method for producing same
CN111635368B (zh) * 2020-06-12 2021-06-29 东莞市东阳光仿制药研发有限公司 一种胺化合物的制备方法
EP4251617B1 (de) 2020-11-27 2025-03-12 Chiesi Farmaceutici S.p.A. (aza)chinolin-4-aminderivate als p2x3-inhibitoren
AU2021386405A1 (en) 2020-11-27 2023-05-25 Chiesi Farmaceutici S.P.A. Phthalazine derivatives as p2x3 inhibitors
MX2023005803A (es) 2020-11-27 2023-05-29 Chiesi Farm Spa Derivados de amino-quinazolina como inhibidores del purinorreceptor 3 p2x (p2x3).
CN116396285A (zh) * 2022-01-04 2023-07-07 上海华汇拓医药科技有限公司 氘代四氢呋喃类化合物制备及其应用

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007025925A1 (en) * 2005-09-01 2007-03-08 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
WO2008040652A1 (en) * 2006-10-04 2008-04-10 F. Hoffmann-La Roche Ag Process for synthesis of phenoxy diaminopyrimidine derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2391636T3 (es) 2004-03-05 2012-11-28 F. Hoffmann-La Roche Ag Diaminopirimidinas como antagonistas de P2X3 y P2X2/3
EP1773405A4 (de) 2004-07-22 2011-10-05 Duska Scient Co Verfahren zur diagnose, überwachung und behandlung von lungenerkrankungen
WO2007025901A1 (en) 2005-09-01 2007-03-08 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
CN101253158B (zh) 2005-09-01 2013-07-10 弗·哈夫曼-拉罗切有限公司 合成芳氧基二氨基嘧啶类化合物的方法
ES2612890T3 (es) 2005-09-01 2017-05-19 F. Hoffmann-La Roche Ag Diaminopirimidinas como moduladores de P2X3 y P2X2/3
WO2008104474A1 (en) * 2007-02-28 2008-09-04 F. Hoffmann-La Roche Ag Diaminopyrimidines
CR20160093A (es) * 2013-08-23 2016-08-26 Afferent Pharmaceuticals Inc Moduladores del receptor p2x3 y p2x2/3 de diaminopiridina para el tratamiento de la tos aguda, sub aguda o cronica

Patent Citations (2)

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Publication number Priority date Publication date Assignee Title
WO2007025925A1 (en) * 2005-09-01 2007-03-08 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
WO2008040652A1 (en) * 2006-10-04 2008-04-10 F. Hoffmann-La Roche Ag Process for synthesis of phenoxy diaminopyrimidine derivatives

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
FORD ANTHONY P: "In pursuit of P2X3 antagonists: novel therapeutics for chronic pain and afferent sensitization", vol. 8, no. Suppl 1, 1 February 2012 (2012-02-01), pages S3 - S26, XP002699076, ISSN: 1573-9546, Retrieved from the Internet <URL:http://rd.springer.com/article/10.1007%2Fs11302-011-9271-6> DOI: 10.1007/S11302-011-9271-6 *

Also Published As

Publication number Publication date
RS64155B1 (sr) 2023-05-31
FIC20240006I1 (fi) 2024-03-13
KR20260022473A (ko) 2026-02-19
LUC00332I2 (de) 2026-03-04
PL3355889T3 (pl) 2023-05-22
CY2024005I2 (el) 2024-09-20
NO2024009I1 (no) 2024-03-06
CY1125963T1 (el) 2024-09-20
MX390084B (es) 2025-03-20
PT3355889T (pt) 2023-04-26
LT3355889T (lt) 2023-05-10
FR24C1010I1 (fr) 2024-05-24
WO2017058645A1 (en) 2017-04-06
CA2998742A1 (en) 2017-04-06
EP3355889A1 (de) 2018-08-08
MX2018003893A (es) 2018-06-22
JP2018529776A (ja) 2018-10-11
FI3355889T3 (fi) 2023-05-15
US11260056B2 (en) 2022-03-01
US20220143015A1 (en) 2022-05-12
ES2942711T3 (es) 2023-06-06
EP3355889B1 (de) 2023-02-15
CY2024005I1 (el) 2024-09-20
KR20180054843A (ko) 2018-05-24
HUE061764T2 (hu) 2023-08-28
US20180280388A1 (en) 2018-10-04
AU2016330466B2 (en) 2021-01-28
AU2016330466A1 (en) 2018-03-29
FR24C1010I2 (fr) 2024-12-13
JP6877441B2 (ja) 2021-05-26
SI3355889T1 (sl) 2023-07-31
NL301260I2 (nl) 2024-03-25
EP4215182A1 (de) 2023-07-26
HRP20230445T1 (hr) 2023-07-21
DK3355889T3 (da) 2023-05-15
LTPA2024507I1 (de) 2024-04-10
HUS2400004I1 (hu) 2024-04-28
US20240285620A1 (en) 2024-08-29
CA2998742C (en) 2023-08-29

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