EP4136056A4 - Formulations topiques non aqueuses - Google Patents

Formulations topiques non aqueuses Download PDF

Info

Publication number
EP4136056A4
EP4136056A4 EP21788324.8A EP21788324A EP4136056A4 EP 4136056 A4 EP4136056 A4 EP 4136056A4 EP 21788324 A EP21788324 A EP 21788324A EP 4136056 A4 EP4136056 A4 EP 4136056A4
Authority
EP
European Patent Office
Prior art keywords
topical formulations
aqueous topical
aqueous
formulations
topical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
EP21788324.8A
Other languages
German (de)
English (en)
Other versions
EP4136056A2 (fr
Inventor
Jihoon P. BAEK
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Baek Clinical Inc
Original Assignee
Baek Clinical Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Baek Clinical Inc filed Critical Baek Clinical Inc
Publication of EP4136056A2 publication Critical patent/EP4136056A2/fr
Publication of EP4136056A4 publication Critical patent/EP4136056A4/fr
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/02—Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/04—Dispersions; Emulsions
    • A61K8/06—Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A61K31/375—Ascorbic acid, i.e. vitamin C; Salts thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/34—Alcohols
    • A61K8/345—Alcohols containing more than one hydroxy group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/36—Carboxylic acids; Salts or anhydrides thereof
    • A61K8/365—Hydroxycarboxylic acids; Ketocarboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/36—Carboxylic acids; Salts or anhydrides thereof
    • A61K8/368—Carboxylic acids; Salts or anhydrides thereof with carboxyl groups directly bound to carbon atoms of aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A61K8/42—Amides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67—Vitamins
    • A61K8/676—Ascorbic acid, i.e. vitamin C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
    • A61K8/84—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
    • A61K8/89—Polysiloxanes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/08—Anti-ageing preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/20—Chemical, physico-chemical or functional or structural properties of the composition as a whole
    • A61K2800/30—Characterized by the absence of a particular group of ingredients
    • A61K2800/31—Anhydrous

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Dispersion Chemistry (AREA)
  • Gerontology & Geriatric Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Cosmetics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EP21788324.8A 2020-04-16 2021-04-16 Formulations topiques non aqueuses Pending EP4136056A4 (fr)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US202063010884P 2020-04-16 2020-04-16
US202063010878P 2020-04-16 2020-04-16
US202063010889P 2020-04-16 2020-04-16
US202063010881P 2020-04-16 2020-04-16
US202063010888P 2020-04-16 2020-04-16
PCT/US2021/027832 WO2021212077A2 (fr) 2020-04-16 2021-04-16 Formulations topiques non aqueuses

Publications (2)

Publication Number Publication Date
EP4136056A2 EP4136056A2 (fr) 2023-02-22
EP4136056A4 true EP4136056A4 (fr) 2024-09-04

Family

ID=78084516

Family Applications (1)

Application Number Title Priority Date Filing Date
EP21788324.8A Pending EP4136056A4 (fr) 2020-04-16 2021-04-16 Formulations topiques non aqueuses

Country Status (7)

Country Link
EP (1) EP4136056A4 (fr)
JP (1) JP2023522328A (fr)
KR (1) KR20230005221A (fr)
CN (1) CN115697903A (fr)
BR (1) BR112022020994A2 (fr)
TW (1) TW202203912A (fr)
WO (1) WO2021212077A2 (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021212073A1 (fr) 2020-04-16 2021-10-21 Baek Clinical Inc. Formulations topiques à haute puissance de vitamine c et d'alcool-sucre
AU2021255734A1 (en) 2020-04-16 2022-11-24 Mf Beauty Partners Llc Stabilizing vitamin C application formulations
JP7623822B2 (ja) * 2020-11-17 2025-01-29 ロート製薬株式会社 外用組成物
WO2022141384A1 (fr) * 2020-12-31 2022-07-07 L'oreal Composition pour le soin de matières kératiniques
US20250228756A1 (en) * 2021-10-20 2025-07-17 Baek Clinical Inc. Anhydrous Urea Emulsions with a Retinoid Agent
KR20240117121A (ko) * 2021-11-30 2024-07-31 로레알 피부 치료 키트 및 방법
CN115887289B (zh) * 2022-10-27 2024-03-08 广州百孚润化工有限公司 一种保湿组合物、含有该保湿组合物的化妆品及其制备方法
KR102671775B1 (ko) * 2023-08-30 2024-06-03 한국콜마주식회사 활성화 성분의 역가 유지율과 제형 안정성이 우수한 화장료 조성물 및 상기 화장료 조성물의 제조방법
CN117530874B (zh) * 2023-11-15 2025-04-15 无锡知妍生物科技有限公司 一种水溶性壬二酸体系及其制备方法
FR3157147A1 (fr) * 2023-12-20 2025-06-27 L'oreal Composition cosmétique comprenant une huile polaire, un alcanol, un polyol, de l’acide azélaïque, et une faible teneur en eau.
WO2025132572A1 (fr) 2023-12-20 2025-06-26 L'oreal Composition cosmétique comprenant une huile, un alcanol, un polyol, de l'acide azélaïque et une faible teneur en eau
FR3157146A1 (fr) 2023-12-20 2025-06-27 L'oreal Composition cosmétique comprenant une huile, un alcanol, un polyol, de l’acide azélaïque, et une faible teneur en eau.

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH05229927A (ja) * 1992-02-21 1993-09-07 Kao Corp 美白化粧料
WO1996039119A1 (fr) * 1995-06-06 1996-12-12 Neutrogena Corporation Excipients topiques contenant de l'acide azelaique solubilise et stabilise
US6361783B2 (en) * 1997-06-27 2002-03-26 Reulon Consumer Products Corporation Compositions containing stabilized ascorbic acid and related methods
WO2005070380A1 (fr) * 2004-01-13 2005-08-04 Skinceuticals, Inc. Compositions d'acide ascorbique stabilisees et methodes associees
US20070172436A1 (en) * 2006-01-23 2007-07-26 Jerry Zhang Nonaqueous ascorbic acid compositions and methods for preparing same
US10149808B2 (en) * 2016-03-31 2018-12-11 L'oreal Cosmetic compositions and methods for providing full spectrum photo protection

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6020367A (en) * 1997-12-02 2000-02-01 Avon Products, Inc. Supersaturated ascorbic acid solutions
US8568749B2 (en) * 2009-04-02 2013-10-29 Sesvalia Usa, Llc Systems and methods for skin rejuvenation
WO2017117099A1 (fr) * 2015-12-29 2017-07-06 L'oreal Compositions antioxydantes stables
EP4299077A3 (fr) * 2016-10-31 2024-04-17 Sytheon Limited Compositions et procédés d'amélioration de la peau
CN111372595A (zh) * 2017-11-21 2020-07-03 塔普克斯制药公司 治疗皮肤的方法和组合物
EP3866771A4 (fr) * 2018-10-18 2022-07-27 Baek Clinical Inc. Formulations topiques de vitamine c à dosage élevé

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH05229927A (ja) * 1992-02-21 1993-09-07 Kao Corp 美白化粧料
WO1996039119A1 (fr) * 1995-06-06 1996-12-12 Neutrogena Corporation Excipients topiques contenant de l'acide azelaique solubilise et stabilise
US6361783B2 (en) * 1997-06-27 2002-03-26 Reulon Consumer Products Corporation Compositions containing stabilized ascorbic acid and related methods
WO2005070380A1 (fr) * 2004-01-13 2005-08-04 Skinceuticals, Inc. Compositions d'acide ascorbique stabilisees et methodes associees
US20070172436A1 (en) * 2006-01-23 2007-07-26 Jerry Zhang Nonaqueous ascorbic acid compositions and methods for preparing same
US10149808B2 (en) * 2016-03-31 2018-12-11 L'oreal Cosmetic compositions and methods for providing full spectrum photo protection

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
ANONYMOUS: "24hr moisturizing anti-fatigue concentrate", GNPD, MINTEL, 31 March 2010 (2010-03-31), XP002762818 *

Also Published As

Publication number Publication date
WO2021212077A3 (fr) 2022-06-16
KR20230005221A (ko) 2023-01-09
WO2021212077A2 (fr) 2021-10-21
CN115697903A (zh) 2023-02-03
JP2023522328A (ja) 2023-05-30
BR112022020994A2 (pt) 2022-12-06
EP4136056A2 (fr) 2023-02-22
TW202203912A (zh) 2022-02-01

Similar Documents

Publication Publication Date Title
EP4136056A4 (fr) Formulations topiques non aqueuses
EP4225284C0 (fr) Compositions ophtalmologiques topiques
SI3927315T1 (sl) Okusne formulacije
EP3746043A4 (fr) Compositions topiques
EP4171537A4 (fr) Composition de vitamine c topique
EP4288151A4 (fr) Compositions ophtalmologiques topiques
IL280533A (en) Topical composition
EP3856128C0 (fr) Formulation d'écran solaire topique
EP4125430A4 (fr) Formulations d'édulcorant
EP4100987A4 (fr) Amélioration de gravure
EP4566770A4 (fr) Main
DK3911298T3 (da) Formuleringer
EP4284362A4 (fr) Préparations
EP3804734A4 (fr) Composition topique
DK3958835T5 (da) Topisk formulering
IL310652A (en) Formulations of radiprodil
EP4188088A4 (fr) Formulations
EP4277592A4 (fr) Composition topique
EP4175676A4 (fr) Formulations muco-pénétrantes
JP1762087S (ja) フィールドスコープ
EP4168116A4 (fr) Formulations topiques de (1s)-1-phényl-2-pyridin-2-yléthanamine
EP4171583A4 (fr) Formulations virucides améliorées
DE112021007890A5 (de) Kurzschließer
EP4021413A4 (fr) Formulations liposomales de composés troponoïdes
EP3941442A4 (fr) Formulations de supraparticules

Legal Events

Date Code Title Description
STAA Information on the status of an ep patent application or granted ep patent

Free format text: STATUS: THE INTERNATIONAL PUBLICATION HAS BEEN MADE

PUAI Public reference made under article 153(3) epc to a published international application that has entered the european phase

Free format text: ORIGINAL CODE: 0009012

STAA Information on the status of an ep patent application or granted ep patent

Free format text: STATUS: REQUEST FOR EXAMINATION WAS MADE

17P Request for examination filed

Effective date: 20221116

AK Designated contracting states

Kind code of ref document: A2

Designated state(s): AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

REG Reference to a national code

Ref country code: HK

Ref legal event code: DE

Ref document number: 40080948

Country of ref document: HK

DAV Request for validation of the european patent (deleted)
DAX Request for extension of the european patent (deleted)
REG Reference to a national code

Ref country code: DE

Ref legal event code: R079

Free format text: PREVIOUS MAIN CLASS: C01B0032336000

Ipc: A61K0008340000

RIC1 Information provided on ipc code assigned before grant

Ipc: A61Q 19/00 20060101ALI20240511BHEP

Ipc: A61K 8/42 20060101ALI20240511BHEP

Ipc: A61K 8/67 20060101ALI20240511BHEP

Ipc: A61K 8/36 20060101ALI20240511BHEP

Ipc: A61K 8/34 20060101AFI20240511BHEP

A4 Supplementary search report drawn up and despatched

Effective date: 20240806

RIC1 Information provided on ipc code assigned before grant

Ipc: A61Q 19/00 20060101ALI20240731BHEP

Ipc: A61K 8/42 20060101ALI20240731BHEP

Ipc: A61K 8/67 20060101ALI20240731BHEP

Ipc: A61K 8/36 20060101ALI20240731BHEP

Ipc: A61K 8/34 20060101AFI20240731BHEP