ES2003200A6 - Un procedimiento para la preparacion de esteroides aminoglicosidicos. - Google Patents

Un procedimiento para la preparacion de esteroides aminoglicosidicos.

Info

Publication number
ES2003200A6
ES2003200A6 ES8700042A ES8700042A ES2003200A6 ES 2003200 A6 ES2003200 A6 ES 2003200A6 ES 8700042 A ES8700042 A ES 8700042A ES 8700042 A ES8700042 A ES 8700042A ES 2003200 A6 ES2003200 A6 ES 2003200A6
Authority
ES
Spain
Prior art keywords
preparation
aminoglycosidic
steroids
procedure
aminotrideoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES8700042A
Other languages
English (en)
Inventor
Laura Chiodini
Mauro Gobbini
Sergio Mantegani
Daniela Ruggieri
Aldemio Temperilli
Gabriella Traquandi
Patrizi Ferrari
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of ES2003200A6 publication Critical patent/ES2003200A6/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

LOS COMPUESTOS I (DONDE O BIEN R1 F OH, ALXOCI C1-4 Y R2 F, ALQUILO C1-4, O R1 B R2 F UN ENLACE QUIMICO; R3 F UN RESTO AMINODESOXI O AMINODIDESOXI O AMINOTRIDESOXI AZUCAR DE LAS SERIES D O L, SIENDO EL ENLACE GLICOSIDICO A O B) Y SUS SALES FARMACEUTICAMENTE ACEPTABLES, SE PREPARAN POR REACCION DE LOS PRECURSORES 3-HIDROXI CORRESPONDIENTES CON UN DERIVADO 1-HALO PROTEGIDO DE UN AZUCAR ADECUADO. LOS COMPUESTOS RESULTANTES DE FORMULA I SON AGENTES ANTIHIPERTENSIVOS UTILES. 1. UN PROCEDIMIENTO PARA LA PREPARACION DE UN COMPUESTO DE FORMULA GENERAL IARMACEUTICAMENTE ACEPTABLE; CUYO PROCEDIMIENTO ESTA CARACTERIZADO PORQUE COMPRENDE CONDENSAR UN ESTEROIDE DE FORMULA GENERAL II.
ES8700042A 1986-01-09 1987-01-08 Un procedimiento para la preparacion de esteroides aminoglicosidicos. Expired ES2003200A6 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868600489A GB8600489D0 (en) 1986-01-09 1986-01-09 Aminoglycoside steroids

Publications (1)

Publication Number Publication Date
ES2003200A6 true ES2003200A6 (es) 1988-10-16

Family

ID=10591134

Family Applications (1)

Application Number Title Priority Date Filing Date
ES8700042A Expired ES2003200A6 (es) 1986-01-09 1987-01-08 Un procedimiento para la preparacion de esteroides aminoglicosidicos.

Country Status (16)

Country Link
US (1) US4882315A (es)
EP (1) EP0254744B1 (es)
JP (1) JPS63502436A (es)
KR (1) KR880700814A (es)
AU (1) AU590409B2 (es)
DK (1) DK468387A (es)
ES (1) ES2003200A6 (es)
FI (1) FI873798A7 (es)
GB (1) GB8600489D0 (es)
GR (1) GR870014B (es)
HU (1) HU198740B (es)
IL (1) IL81164A (es)
NZ (1) NZ218856A (es)
PT (1) PT84072B (es)
WO (1) WO1987004167A2 (es)
ZA (1) ZA87114B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8600490D0 (en) * 1986-01-09 1986-02-12 Erba Farmitalia Aminoglycoside norcholanic acid lactams
US5104856A (en) * 1990-11-09 1992-04-14 Uab Research Foundation Heparan sulfate biosynthesis primers
US5270457A (en) * 1992-06-12 1993-12-14 University Of Manitoba Cardiac steriod glycosides
ATE183192T1 (de) * 1993-01-08 1999-08-15 Astra Ab Neue colon-oder ilean-spezifische steroid derivate
BR9407612A (pt) * 1993-09-24 1997-01-14 Procter & Gamble Novos compostos de 14-aminoesteróides contendo oligossacarideos e nova química de processo de aminoesteróide diastereosseletivo
US5922703A (en) * 1993-09-24 1999-07-13 The Procter & Gamble Company Urethane-containing aminosteroid compounds
ATE422359T1 (de) 1997-04-15 2009-02-15 Csir Verbindungen und pharmazeutische zusammensetzungen mit appetitunterdrückender aktivität
ATE473759T1 (de) 1998-05-22 2010-07-15 Univ Leland Stanford Junior Bifunktionelle moleküle sowie darauf basierende therapien.
GB2396815B (en) * 1999-10-27 2004-09-08 Phytopharm Plc A composition comprising a pregnenone derivative and an NSAID
GB2363985B (en) * 2000-06-30 2004-09-29 Phytopharm Plc Extracts,compounds & pharmaceutical compositions having anti-diabetic activity and their use
US20040064050A1 (en) * 2002-09-20 2004-04-01 Jun Liu System and method for screening tissue
CN102379684B (zh) 2005-04-28 2014-11-19 普罗透斯数字保健公司 药物信息系统
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
EP2398500B1 (en) 2009-02-20 2019-03-13 2-BBB Medicines B.V. Glutathione-based drug delivery system
ES2942923T3 (es) 2009-05-06 2023-06-07 Laboratory Skin Care Inc Composiciones de administración dérmica que comprenden complejos de agente activo-partículas de fosfato de calcio y métodos de uso de las mismas
EP2468253A1 (en) * 2010-12-14 2012-06-27 InterMed Discovery GmbH Terpenoid spiro ketal compounds with LXR agonists activity, their use and formulations with them

Also Published As

Publication number Publication date
IL81164A (en) 1990-12-23
HU198740B (en) 1989-11-28
HUT46930A (en) 1988-12-28
DK468387D0 (da) 1987-09-08
US4882315A (en) 1989-11-21
EP0254744A1 (en) 1988-02-03
AU590409B2 (en) 1989-11-02
NZ218856A (en) 1989-05-29
JPS63502436A (ja) 1988-09-14
FI873798L (fi) 1987-09-01
GB8600489D0 (en) 1986-02-12
FI873798A0 (fi) 1987-09-01
ZA87114B (en) 1987-09-30
WO1987004167A3 (en) 1987-08-13
WO1987004167A2 (en) 1987-07-16
DK468387A (da) 1987-09-08
IL81164A0 (en) 1987-08-31
GR870014B (en) 1987-05-08
PT84072A (en) 1987-02-01
PT84072B (pt) 1989-07-31
FI873798A7 (fi) 1987-09-01
KR880700814A (ko) 1988-04-12
EP0254744B1 (en) 1990-09-19
AU7161187A (en) 1987-07-28

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19950109