ES2003200A6 - Un procedimiento para la preparacion de esteroides aminoglicosidicos. - Google Patents

Un procedimiento para la preparacion de esteroides aminoglicosidicos.

Info

Publication number
ES2003200A6
ES2003200A6 ES8700042A ES8700042A ES2003200A6 ES 2003200 A6 ES2003200 A6 ES 2003200A6 ES 8700042 A ES8700042 A ES 8700042A ES 8700042 A ES8700042 A ES 8700042A ES 2003200 A6 ES2003200 A6 ES 2003200A6
Authority
ES
Spain
Prior art keywords
preparation
aminoglycosidic
steroids
procedure
aminotrideoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES8700042A
Other languages
English (en)
Inventor
Laura Chiodini
Mauro Gobbini
Sergio Mantegani
Daniela Ruggieri
Aldemio Temperilli
Gabriella Traquandi
Patrizi Ferrari
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of ES2003200A6 publication Critical patent/ES2003200A6/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

LOS COMPUESTOS I (DONDE O BIEN R1 F OH, ALXOCI C1-4 Y R2 F, ALQUILO C1-4, O R1 B R2 F UN ENLACE QUIMICO; R3 F UN RESTO AMINODESOXI O AMINODIDESOXI O AMINOTRIDESOXI AZUCAR DE LAS SERIES D O L, SIENDO EL ENLACE GLICOSIDICO A O B) Y SUS SALES FARMACEUTICAMENTE ACEPTABLES, SE PREPARAN POR REACCION DE LOS PRECURSORES 3-HIDROXI CORRESPONDIENTES CON UN DERIVADO 1-HALO PROTEGIDO DE UN AZUCAR ADECUADO. LOS COMPUESTOS RESULTANTES DE FORMULA I SON AGENTES ANTIHIPERTENSIVOS UTILES. 1. UN PROCEDIMIENTO PARA LA PREPARACION DE UN COMPUESTO DE FORMULA GENERAL IARMACEUTICAMENTE ACEPTABLE; CUYO PROCEDIMIENTO ESTA CARACTERIZADO PORQUE COMPRENDE CONDENSAR UN ESTEROIDE DE FORMULA GENERAL II.
ES8700042A 1986-01-09 1987-01-08 Un procedimiento para la preparacion de esteroides aminoglicosidicos. Expired ES2003200A6 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868600489A GB8600489D0 (en) 1986-01-09 1986-01-09 Aminoglycoside steroids

Publications (1)

Publication Number Publication Date
ES2003200A6 true ES2003200A6 (es) 1988-10-16

Family

ID=10591134

Family Applications (1)

Application Number Title Priority Date Filing Date
ES8700042A Expired ES2003200A6 (es) 1986-01-09 1987-01-08 Un procedimiento para la preparacion de esteroides aminoglicosidicos.

Country Status (15)

Country Link
US (1) US4882315A (es)
EP (1) EP0254744B1 (es)
JP (1) JPS63502436A (es)
KR (1) KR880700814A (es)
AU (1) AU590409B2 (es)
DK (1) DK468387A (es)
ES (1) ES2003200A6 (es)
FI (1) FI873798A0 (es)
GB (1) GB8600489D0 (es)
GR (1) GR870014B (es)
HU (1) HU198740B (es)
IL (1) IL81164A (es)
NZ (1) NZ218856A (es)
PT (1) PT84072B (es)
ZA (1) ZA87114B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8600490D0 (en) * 1986-01-09 1986-02-12 Erba Farmitalia Aminoglycoside norcholanic acid lactams
US5104856A (en) * 1990-11-09 1992-04-14 Uab Research Foundation Heparan sulfate biosynthesis primers
US5270457A (en) * 1992-06-12 1993-12-14 University Of Manitoba Cardiac steriod glycosides
CZ171095A3 (en) * 1993-01-08 1996-01-17 Astra Ab Novel steroidal derivatives specific for colon or ilium
SK141899A3 (en) * 1997-04-15 2000-09-12 Csir Corporate Building Pharmaceutical compositions having appetite suppressant activity
US6372712B1 (en) 1998-05-22 2002-04-16 The Board Of Trustees Of The Leland Stanford Jr. University Synthetic bifunctional molecules containing a drug moiety and presenter protein ligand
GB2396815B (en) * 1999-10-27 2004-09-08 Phytopharm Plc A composition comprising a pregnenone derivative and an NSAID
GB2363985B (en) * 2000-06-30 2004-09-29 Phytopharm Plc Extracts,compounds & pharmaceutical compositions having anti-diabetic activity and their use
US20040064050A1 (en) * 2002-09-20 2004-04-01 Jun Liu System and method for screening tissue
EP2671508B1 (en) 2005-04-28 2020-09-16 Proteus Digital Health, Inc. Pharma-informatics system
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
ES2919563T3 (es) 2009-02-20 2022-07-27 Enhanx Biopharm Inc Sistema de administración de medicamentos a base de glutatión
KR20180114970A (ko) 2009-05-06 2018-10-19 라보라토리 스킨 케어, 인크. 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법

Also Published As

Publication number Publication date
WO1987004167A2 (en) 1987-07-16
FI873798A7 (fi) 1987-09-01
ZA87114B (en) 1987-09-30
DK468387D0 (da) 1987-09-08
WO1987004167A3 (en) 1987-08-13
IL81164A (en) 1990-12-23
AU7161187A (en) 1987-07-28
GB8600489D0 (en) 1986-02-12
GR870014B (en) 1987-05-08
IL81164A0 (en) 1987-08-31
HUT46930A (en) 1988-12-28
JPS63502436A (ja) 1988-09-14
FI873798L (fi) 1987-09-01
AU590409B2 (en) 1989-11-02
DK468387A (da) 1987-09-08
EP0254744B1 (en) 1990-09-19
KR880700814A (ko) 1988-04-12
US4882315A (en) 1989-11-21
PT84072A (en) 1987-02-01
HU198740B (en) 1989-11-28
FI873798A0 (fi) 1987-09-01
PT84072B (pt) 1989-07-31
EP0254744A1 (en) 1988-02-03
NZ218856A (en) 1989-05-29

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19950109