ES2007259A6 - Un procedimiento para preparar cis-4-amino-5-cloro-n-(1-(3-(4-fluorfenoxi)propil)-3-metoxi-4-piperidinil)-2-metoxibenzamina. - Google Patents
Un procedimiento para preparar cis-4-amino-5-cloro-n-(1-(3-(4-fluorfenoxi)propil)-3-metoxi-4-piperidinil)-2-metoxibenzamina.Info
- Publication number
- ES2007259A6 ES2007259A6 ES8802167A ES8802167A ES2007259A6 ES 2007259 A6 ES2007259 A6 ES 2007259A6 ES 8802167 A ES8802167 A ES 8802167A ES 8802167 A ES8802167 A ES 8802167A ES 2007259 A6 ES2007259 A6 ES 2007259A6
- Authority
- ES
- Spain
- Prior art keywords
- methoxy
- fluoro
- piperidinyl
- benzamide
- opt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- -1 phenoxy propyl methoxy-piperidinyl methoxy-benzamide Chemical compound 0.000 title abstract 2
- 125000001153 fluoro group Chemical group F* 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 2
- MNWSGMTUGXNYHJ-UHFFFAOYSA-N 2-methoxybenzamide Chemical compound COC1=CC=CC=C1C(N)=O MNWSGMTUGXNYHJ-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical group C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 abstract 1
- 239000002585 base Substances 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 239000012458 free base Substances 0.000 abstract 1
- 230000005176 gastrointestinal motility Effects 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 150000002500 ions Chemical class 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
- 239000003960 organic solvent Substances 0.000 abstract 1
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 abstract 1
- 230000004936 stimulating effect Effects 0.000 abstract 1
Landscapes
- Hydrogenated Pyridines (AREA)
Abstract
UN PROCEDIMIENTO PARA PREPARAR CIS-4-AMINO-5-CLORO-N-[1-[3-(4-FLUORFENOXI)PROPIL]-3-METOXI-4-PIPERIDINIL]-2-METOXIBENZAMIDA. EL COMPUESTO DE FORMULA (I) SE OBTIENE POR REDUCCION DE LA SAL DE PIRIDINIO CUATERNARIO DE FORMULA (II) EN LA QUE W- REPRESENTA UN ANION INORGANICO U ORGANICO CON UN CATALIZADOR METALICO, EN UN DISOLVENTE INERTE, EN PRESENCIA DE HIDROGENO, OPCIONALMENTE A TEMPERATURA Y PRESION ELEVADA Y, OPCIONALMENTE, EN PRESENCIA DE UNA BASE; Y SI SE DESEA, PREPARAR SALES FARMACEUTICAMENTE ACEPTABLES O TRANSFORMAR LAS SALES EN LA BASE LIBRE. EL COMPUESTO (I) TIENE UTILIDAD POR SUS BUENAS PROPIEDADES ESTIMULANTES EN LA MOTILIDAD GASTROINTESTINAL.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES8802167A ES2007259A6 (es) | 1988-07-08 | 1988-07-08 | Un procedimiento para preparar cis-4-amino-5-cloro-n-(1-(3-(4-fluorfenoxi)propil)-3-metoxi-4-piperidinil)-2-metoxibenzamina. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES8802167A ES2007259A6 (es) | 1988-07-08 | 1988-07-08 | Un procedimiento para preparar cis-4-amino-5-cloro-n-(1-(3-(4-fluorfenoxi)propil)-3-metoxi-4-piperidinil)-2-metoxibenzamina. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2007259A6 true ES2007259A6 (es) | 1989-06-01 |
Family
ID=8257244
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES8802167A Expired ES2007259A6 (es) | 1988-07-08 | 1988-07-08 | Un procedimiento para preparar cis-4-amino-5-cloro-n-(1-(3-(4-fluorfenoxi)propil)-3-metoxi-4-piperidinil)-2-metoxibenzamina. |
Country Status (1)
| Country | Link |
|---|---|
| ES (1) | ES2007259A6 (es) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2053394A1 (es) * | 1992-11-16 | 1994-07-16 | S A L V A T Lab Sa | "3-bromo-4-oxo-1-piperidincarboxilato de etilo, procedimiento para la obtencion del mismo y nuevos intermedios utilizados en su preparacion" |
-
1988
- 1988-07-08 ES ES8802167A patent/ES2007259A6/es not_active Expired
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2053394A1 (es) * | 1992-11-16 | 1994-07-16 | S A L V A T Lab Sa | "3-bromo-4-oxo-1-piperidincarboxilato de etilo, procedimiento para la obtencion del mismo y nuevos intermedios utilizados en su preparacion" |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 20050709 |