ES2061445T3 - Un procedimiento para la preparacion de una omega-alquil-amino-tetrahidro-6h-1,3-tiazin-6-ona aromatica. - Google Patents

Un procedimiento para la preparacion de una omega-alquil-amino-tetrahidro-6h-1,3-tiazin-6-ona aromatica.

Info

Publication number
ES2061445T3
ES2061445T3 ES87103078T ES87103078T ES2061445T3 ES 2061445 T3 ES2061445 T3 ES 2061445T3 ES 87103078 T ES87103078 T ES 87103078T ES 87103078 T ES87103078 T ES 87103078T ES 2061445 T3 ES2061445 T3 ES 2061445T3
Authority
ES
Spain
Prior art keywords
procedure
preparation
tiazin
aromatica
ona
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87103078T
Other languages
English (en)
Inventor
Marcel Hibert
Maurice W Gittos
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Merrell Dow Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharmaceuticals Inc filed Critical Merrell Dow Pharmaceuticals Inc
Application granted granted Critical
Publication of ES2061445T3 publication Critical patent/ES2061445T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Anesthesiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

ESTA INVENCION SE REFIERE A DERIVADOS AROMATICOS DE W-ALQUILIMINO-TETRAHIDRO - 6H-1,3-TIAZINONA-6, A UN PROCEDIMIENTO PARA SU PREPARACION Y A SU EMPLEO COMO AGENTES ANSIOLITICOS Y ANTIHIPERTENSORES.
ES87103078T 1986-03-05 1987-03-04 Un procedimiento para la preparacion de una omega-alquil-amino-tetrahidro-6h-1,3-tiazin-6-ona aromatica. Expired - Lifetime ES2061445T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US83627586A 1986-03-05 1986-03-05

Publications (1)

Publication Number Publication Date
ES2061445T3 true ES2061445T3 (es) 1994-12-16

Family

ID=25271603

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87103078T Expired - Lifetime ES2061445T3 (es) 1986-03-05 1987-03-04 Un procedimiento para la preparacion de una omega-alquil-amino-tetrahidro-6h-1,3-tiazin-6-ona aromatica.

Country Status (18)

Country Link
EP (1) EP0236931B1 (es)
JP (1) JPH0667933B2 (es)
KR (1) KR900000676B1 (es)
CN (1) CN1021825C (es)
AR (1) AR241162A2 (es)
AT (1) ATE99309T1 (es)
AU (1) AU589256B2 (es)
CA (1) CA1288101C (es)
DE (1) DE3788581T2 (es)
DK (1) DK111887A (es)
ES (1) ES2061445T3 (es)
FI (1) FI89919C (es)
HU (1) HU201546B (es)
IL (2) IL81718A0 (es)
NO (1) NO166182C (es)
PH (1) PH25227A (es)
PT (1) PT84406B (es)
ZA (1) ZA871449B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5116970A (en) * 1988-02-18 1992-05-26 New James S Psychotropic heterobicycloalkylpiperazine derivatives: 2. fused pyridazinones
US5001130A (en) * 1988-02-18 1991-03-19 Bristol-Myers Company Psychotropic heterobicycloalkylpiperazine derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3398151A (en) * 1966-02-01 1968-08-20 Mead Johnson & Co Azaspirodecanediones and azaspiroundecanediones
BE759371A (fr) * 1969-11-24 1971-05-24 Bristol Myers Co Azaspirodecanediones heterocycliques et procedes pour leur preparation
DE2727469A1 (de) * 1977-06-18 1978-12-21 Hoechst Ag Neue hexahydropyrimidine, verfahren zu ihrer herstellung und arzneimittel, die diese verbindungen enthalten
ZA855563B (en) * 1984-07-30 1986-05-28 Merrell Dow Pharma Glutarimide antianxiety and antihypertensive agents

Also Published As

Publication number Publication date
ATE99309T1 (de) 1994-01-15
DK111887D0 (da) 1987-03-04
NO166182C (no) 1991-06-12
PT84406B (pt) 1989-10-04
KR900000676B1 (ko) 1990-02-02
CN87101690A (zh) 1987-12-30
JPS62221683A (ja) 1987-09-29
ZA871449B (en) 1987-08-20
PT84406A (en) 1987-04-01
PH25227A (en) 1991-03-27
CN1021825C (zh) 1993-08-18
FI870924A7 (fi) 1987-09-06
DE3788581D1 (de) 1994-02-10
NO166182B (no) 1991-03-04
NO870889L (no) 1987-09-07
NO870889D0 (no) 1987-03-04
FI870924A0 (fi) 1987-03-03
FI89919C (fi) 1993-12-10
HUT47105A (en) 1989-01-30
EP0236931B1 (en) 1993-12-29
HU201546B (en) 1990-11-28
IL81718A0 (en) 1987-10-20
AU6960587A (en) 1987-09-10
DK111887A (da) 1987-09-06
DE3788581T2 (de) 1994-04-28
AR241162A2 (en) 1991-12-30
EP0236931A2 (en) 1987-09-16
FI89919B (fi) 1993-08-31
KR870008887A (ko) 1987-10-21
IL81738A0 (en) 1987-10-20
CA1288101C (en) 1991-08-27
EP0236931A3 (en) 1990-01-17
AU589256B2 (en) 1989-10-05
JPH0667933B2 (ja) 1994-08-31

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