ES2062351T3 - Derivados de triazolo (4,5-c) piridina anticonvulsivos. - Google Patents
Derivados de triazolo (4,5-c) piridina anticonvulsivos.Info
- Publication number
- ES2062351T3 ES2062351T3 ES90304271T ES90304271T ES2062351T3 ES 2062351 T3 ES2062351 T3 ES 2062351T3 ES 90304271 T ES90304271 T ES 90304271T ES 90304271 T ES90304271 T ES 90304271T ES 2062351 T3 ES2062351 T3 ES 2062351T3
- Authority
- ES
- Spain
- Prior art keywords
- anticonvulsives
- piridine
- triazole derivatives
- disclosed
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 229940042055 systemic antimycotics triazole derivative Drugs 0.000 title 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 206010015037 epilepsy Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Chemical class 0.000 abstract 1
- YWBFPKPWMSWWEA-UHFFFAOYSA-O triazolopyrimidine Chemical class BrC1=CC=CC(C=2N=C3N=CN[N+]3=C(NCC=3C=CN=CC=3)C=2)=C1 YWBFPKPWMSWWEA-UHFFFAOYSA-O 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
SE PRESENTAN UNA SERIE DE COMPUESTOS DE TRIAZOLOPIRIMIDINA Y COMPUESTOS FARMACEUTICOS QUE LA CONTIENEN. LOS COMPUESTOS PRESENTADOS SON UTILES EN EL TRATAMIENTO DE DESORDENES NERVIOSOS CENTRALES, TALES COMO LA EPILEPSIA EN LOS MAMIFEROS. TAMBIEN SE PRESENTAN METODOS PARA LA PREPARACION DE ESTAS TRIAZOLOPIRIMIDINAS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB898909136A GB8909136D0 (en) | 1989-04-21 | 1989-04-21 | Anticonvulsant pyridines and analogues thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2062351T3 true ES2062351T3 (es) | 1994-12-16 |
Family
ID=10655494
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES90304271T Expired - Lifetime ES2062351T3 (es) | 1989-04-21 | 1990-04-20 | Derivados de triazolo (4,5-c) piridina anticonvulsivos. |
Country Status (21)
| Country | Link |
|---|---|
| EP (1) | EP0399653B1 (es) |
| JP (1) | JP2865367B2 (es) |
| KR (1) | KR0183972B1 (es) |
| AT (1) | ATE113046T1 (es) |
| CA (1) | CA2015047A1 (es) |
| CY (1) | CY2003B1 (es) |
| DD (1) | DD293823A5 (es) |
| DE (1) | DE69013396T2 (es) |
| DK (1) | DK0399653T3 (es) |
| ES (1) | ES2062351T3 (es) |
| FI (1) | FI93448C (es) |
| GB (1) | GB8909136D0 (es) |
| HK (1) | HK78397A (es) |
| HU (2) | HU206210B (es) |
| IE (1) | IE67335B1 (es) |
| IL (1) | IL94150A (es) |
| LV (1) | LV5780B4 (es) |
| NZ (1) | NZ233404A (es) |
| PH (1) | PH27118A (es) |
| PT (1) | PT93822B (es) |
| ZA (1) | ZA903021B (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002518391A (ja) | 1998-06-16 | 2002-06-25 | メルク シャープ エンド ドーム リミテッド | Ｇａｂａ受容体のリガンドとしてのトリアゾロ−ピリジン誘導体 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3929812A (en) * | 1974-05-20 | 1975-12-30 | Squibb & Sons Inc | Derivatives of 1H-triazolo {8 4,5-c{9 pyridine-7-carboxylic acids and esters |
| ES2051886T3 (es) * | 1987-04-07 | 1994-07-01 | Ciba Geigy Ag | Procedimiento para la obtencion de nuevos derivados de la 3h-1,2,3-triazolo(4,5-d)pirimidina. |
-
1989
- 1989-04-21 GB GB898909136A patent/GB8909136D0/en active Pending
-
1990
- 1990-04-19 PH PH40399A patent/PH27118A/en unknown
- 1990-04-20 ZA ZA903021A patent/ZA903021B/xx unknown
- 1990-04-20 DD DD90339946A patent/DD293823A5/de not_active IP Right Cessation
- 1990-04-20 CA CA002015047A patent/CA2015047A1/en not_active Abandoned
- 1990-04-20 DK DK90304271.1T patent/DK0399653T3/da active
- 1990-04-20 IL IL9415090A patent/IL94150A/en not_active IP Right Cessation
- 1990-04-20 AT AT90304271T patent/ATE113046T1/de not_active IP Right Cessation
- 1990-04-20 HU HU902502A patent/HU206210B/hu not_active IP Right Cessation
- 1990-04-20 KR KR1019900005523A patent/KR0183972B1/ko not_active Expired - Fee Related
- 1990-04-20 FI FI901981A patent/FI93448C/fi not_active IP Right Cessation
- 1990-04-20 DE DE69013396T patent/DE69013396T2/de not_active Expired - Fee Related
- 1990-04-20 JP JP2105156A patent/JP2865367B2/ja not_active Expired - Lifetime
- 1990-04-20 EP EP90304271A patent/EP0399653B1/en not_active Expired - Lifetime
- 1990-04-20 ES ES90304271T patent/ES2062351T3/es not_active Expired - Lifetime
- 1990-04-20 IE IE140990A patent/IE67335B1/en not_active IP Right Cessation
- 1990-04-20 NZ NZ233404A patent/NZ233404A/en unknown
- 1990-04-20 PT PT93822A patent/PT93822B/pt not_active IP Right Cessation
-
1995
- 1995-05-11 HU HU95P/P00126P patent/HU211137A9/hu unknown
-
1996
- 1996-07-17 LV LV960252A patent/LV5780B4/xx unknown
-
1997
- 1997-06-12 HK HK78397A patent/HK78397A/en not_active IP Right Cessation
-
1998
- 1998-04-30 CY CY9802003A patent/CY2003B1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NZ233404A (en) | 1992-08-26 |
| HU902502D0 (en) | 1990-08-28 |
| DE69013396D1 (de) | 1994-11-24 |
| DD293823A5 (de) | 1991-09-12 |
| KR0183972B1 (ko) | 1999-05-01 |
| CY2003B1 (en) | 1998-04-30 |
| KR900016208A (ko) | 1990-11-12 |
| FI93448B (fi) | 1994-12-30 |
| ATE113046T1 (de) | 1994-11-15 |
| FI93448C (fi) | 1995-04-10 |
| FI901981A0 (fi) | 1990-04-20 |
| AU626409B2 (en) | 1992-07-30 |
| AU5372290A (en) | 1990-10-25 |
| LV5780A4 (lv) | 1996-12-20 |
| ZA903021B (en) | 1991-12-24 |
| PH27118A (en) | 1993-03-16 |
| PT93822A (pt) | 1990-11-20 |
| IL94150A (en) | 1994-02-27 |
| HUT53905A (en) | 1990-12-28 |
| GB8909136D0 (en) | 1989-06-07 |
| HU211137A9 (en) | 1995-10-30 |
| EP0399653A1 (en) | 1990-11-28 |
| DK0399653T3 (da) | 1994-11-14 |
| JPH02292286A (ja) | 1990-12-03 |
| CA2015047A1 (en) | 1990-10-21 |
| IE901409L (en) | 1990-10-21 |
| HU206210B (en) | 1992-09-28 |
| LV5780B4 (lv) | 1997-04-20 |
| JP2865367B2 (ja) | 1999-03-08 |
| IL94150A0 (en) | 1991-01-31 |
| DE69013396T2 (de) | 1995-05-04 |
| IE67335B1 (en) | 1996-03-20 |
| HK78397A (en) | 1997-06-20 |
| EP0399653B1 (en) | 1994-10-19 |
| PT93822B (pt) | 1996-09-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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