ES2064229B1 - Nuevas 1,2-dihidro-2-oxopiridinas de formula i. - Google Patents
Nuevas 1,2-dihidro-2-oxopiridinas de formula i.Info
- Publication number
- ES2064229B1 ES2064229B1 ES9202251A ES9202251A ES2064229B1 ES 2064229 B1 ES2064229 B1 ES 2064229B1 ES 9202251 A ES9202251 A ES 9202251A ES 9202251 A ES9202251 A ES 9202251A ES 2064229 B1 ES2064229 B1 ES 2064229B1
- Authority
- ES
- Spain
- Prior art keywords
- oxopyridines
- dihydro
- formula
- new
- aldosteronism
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 102000005862 Angiotensin II Human genes 0.000 abstract 1
- 101800000733 Angiotensin-2 Proteins 0.000 abstract 1
- 206010019280 Heart failures Diseases 0.000 abstract 1
- 206010020571 Hyperaldosteronism Diseases 0.000 abstract 1
- 206010020772 Hypertension Diseases 0.000 abstract 1
- CZGUSIXMZVURDU-JZXHSEFVSA-N Ile(5)-angiotensin II Chemical compound C([C@@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC=1NC=NC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC=1C=CC=CC=1)C([O-])=O)NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=[NH2+])NC(=O)[C@@H]([NH3+])CC([O-])=O)C(C)C)C1=CC=C(O)C=C1 CZGUSIXMZVURDU-JZXHSEFVSA-N 0.000 abstract 1
- 229950006323 angiotensin ii Drugs 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
NUEVAS 1,2-DIHIDRO-2-OXOPIRIDINAS DE FORMULA I *FIG* EN LAS QUE: R ES EL RADICAL Y R1 A R6 Y X SON COMO SE DEFINE LA REIVINDICACION 1, Y SUS SALES, TIENEN PROPIEDADES ANTAGONISTAS HACIA LA ANGIOTENSINA II Y PUEDEN USARSE PARA EL TRATAMIENTO DE HIPERTENSION, ALDOSTERONISMO E INSUFICIENCIA CARDIACA.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES9202251A ES2064229B1 (es) | 1992-11-06 | 1992-11-06 | Nuevas 1,2-dihidro-2-oxopiridinas de formula i. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES9202251A ES2064229B1 (es) | 1992-11-06 | 1992-11-06 | Nuevas 1,2-dihidro-2-oxopiridinas de formula i. |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES2064229A1 ES2064229A1 (es) | 1995-01-16 |
| ES2064229B1 true ES2064229B1 (es) | 1996-03-01 |
Family
ID=8278715
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES9202251A Expired - Lifetime ES2064229B1 (es) | 1992-11-06 | 1992-11-06 | Nuevas 1,2-dihidro-2-oxopiridinas de formula i. |
Country Status (1)
| Country | Link |
|---|---|
| ES (1) | ES2064229B1 (es) |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4880804A (en) * | 1988-01-07 | 1989-11-14 | E. I. Du Pont De Nemours And Company | Angiotensin II receptor blocking benzimidazoles |
| CA2037630C (en) * | 1990-03-07 | 2001-07-03 | Akira Morimoto | Nitrogen-containing heterocylic compounds, their production and use |
| CA2051705A1 (en) * | 1990-06-19 | 1991-12-20 | Kiyoaki Katano | Pyridine derivatives having angiotensin ii antagonism |
| IL100917A0 (en) * | 1991-02-16 | 1992-11-15 | Fisons Plc | Pyridinone and pyrimidinone derivatives,their preparation and pharmaceutical compositions containing them |
-
1992
- 1992-11-06 ES ES9202251A patent/ES2064229B1/es not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| ES2064229A1 (es) | 1995-01-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA2A | Application withdrawn |
Effective date: 19970218 |