ES2100706T3 - Compuestos heterociclicos con actividad antiparasitaria. - Google Patents

Compuestos heterociclicos con actividad antiparasitaria.

Info

Publication number
ES2100706T3
ES2100706T3 ES94910243T ES94910243T ES2100706T3 ES 2100706 T3 ES2100706 T3 ES 2100706T3 ES 94910243 T ES94910243 T ES 94910243T ES 94910243 T ES94910243 T ES 94910243T ES 2100706 T3 ES2100706 T3 ES 2100706T3
Authority
ES
Spain
Prior art keywords
optionally substituted
haloalkynyl
haloalkenyl
haloalkyl
alkynyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94910243T
Other languages
English (en)
Inventor
Steven Fitzjohn
Michael Peter Robinson
Michael Drysdale Turnbull
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Syngenta Ltd
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Application granted granted Critical
Publication of ES2100706T3 publication Critical patent/ES2100706T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/07—Preparation of halogenated hydrocarbons by addition of hydrogen halides
    • C07C17/087—Preparation of halogenated hydrocarbons by addition of hydrogen halides to unsaturated halogenated hydrocarbons
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/64—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
    • C07C309/65—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton
    • C07C309/66—Methanesulfonates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/30—Isothioureas
    • C07C335/32—Isothioureas having sulfur atoms of isothiourea groups bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56—One oxygen atom and one sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/58—Two sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

LA INVENCION PROPORCIONA NUEVOS COMPUESTOS DE FORMULA (I) QUE TIENEN PROPIEDADES NEMATICIDAS, INSECTICIDAS, ACARICIDAS Y FUNGICIDAS, COMPOSICIONES QUE LOS COMPRENDEN Y PROCESOS Y PRODUCTOS INTERMEDIOS PARA SU PREPARACION; EN DONDE R1 ES -S(O)NCH2CH2CH=CF2; N SE SELECCIONA DE 0, 1 Y 2; R2, R3, Y R4 SON SELECCIONADOS INDEPENDIENTEMENTE DE HIDROGENO, ALQUILO, ALQUENILO, ALQUINILO, CICLOALQUILO, ALQUILCICLOALQUILO, ARILO OPCIONALMENTE SUSTITUIDO, ARILALQUILO OPCIONALMENTE SUSTITUIDO, ARILOXILO OPCIONALMENTE SUSTITUIDO, ARILALCOXILO OPCIONALMENTE SUSTITUIDO, ALCOXILO, ALQUENILOXILO, ALQUINILOXILO, HIDROXIALQUILO, ALCOXIALQUILO, ALQUILTIO, ALQUENILTIO, ALQUINILTIO, HALOALQUILO, HALOALQUENILO, HALOALQUINILO, HALOALCOXILO, HALOALQUENILOXILO, HALOALQUINILOXILO, HALOALQUILTIO, HALOALQUENILTIO, HALOALQUINILTIO, HALOGENO, HIDROXILO, CIANO, NITRO, -NR5R6, -NR7COR8, -NR9SO2R10, -N(SO2-R11)(SO2-R12), -COR13, -CONR14R15, -COOR16, -OCOR17, -OSO2R18, -SO2NR19R20, -SO2R21, -SOR22, -CSNR23R24, -SIR25R26R27, -OCH2CO2R28, -OCH2CH2CO2R29, -CONR30SO2R31, -SO2Z, O UN PAR ADYACENTE DE R2, R3 Y R4 CUANDO SE TOMAN JUNTOS FORMAN UN ANILLO HETEROCICLICO O CARBOCICLICO DE 5- O 6-MIEMBROS; R5, R6, R7, R8, R9, R10, R11, R12, R13, R14, R15, R16, R17, R18, R19, R20, R21, R22, R23, R24, R25, R26, R27, R28, R29, R30 Y R31 SON SELECCIONADOS INDEPENDIENTEMENTE DE HIDROGENO, ALQUILO, ALQUENILO, ALQUINILO, HALOALQUILO, HALOALQUENILO, HALOALQUINILO, ARILO OPCIONALMENTE SUSTITUIDO Y ARILALQUILO OPCIONALMENTE SUSTITUIDO; Y Z ES HALOGENO.
ES94910243T 1992-09-16 1993-09-10 Compuestos heterociclicos con actividad antiparasitaria. Expired - Lifetime ES2100706T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929219635A GB9219635D0 (en) 1992-09-16 1992-09-16 Heterocyclic compounds

Publications (1)

Publication Number Publication Date
ES2100706T3 true ES2100706T3 (es) 1997-06-16

Family

ID=10722036

Family Applications (1)

Application Number Title Priority Date Filing Date
ES94910243T Expired - Lifetime ES2100706T3 (es) 1992-09-16 1993-09-10 Compuestos heterociclicos con actividad antiparasitaria.

Country Status (13)

Country Link
US (1) US5684011A (es)
EP (1) EP0660827B1 (es)
JP (1) JPH08503932A (es)
CN (1) CN1041922C (es)
AT (1) ATE151757T1 (es)
AU (1) AU4977793A (es)
DE (1) DE69309941T2 (es)
DK (1) DK0660827T3 (es)
ES (1) ES2100706T3 (es)
GB (2) GB9219635D0 (es)
IL (1) IL106970A0 (es)
WO (1) WO1994006777A1 (es)
ZA (1) ZA936708B (es)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5125957A (en) * 1989-11-01 1992-06-30 Sumitomo Chemical Company, Limited Pyrimidine derivatives
KR100234555B1 (ko) * 1993-08-05 1999-12-15 돈 리사 로얄 플루오로아테닐티오 복소환식 유도체의 제조방법
IL112721A0 (en) * 1994-03-10 1995-05-26 Zeneca Ltd Azole derivatives
GB9404942D0 (en) * 1994-03-15 1994-04-27 Zeneca Ltd Heterocyclic compound
GB9518111D0 (en) * 1995-09-06 1995-11-08 Zeneca Ltd Chemical process
JPH1120619A (ja) * 1997-07-02 1999-01-26 Mitsuba Corp ワイパ装置
JP2000001481A (ja) * 1998-04-13 2000-01-07 Nippon Nohyaku Co Ltd １，２，３―チアジアゾ―ル誘導体又はその塩類及び有害生物防除剤並びにその使用方法
JP2001322988A (ja) 2000-03-09 2001-11-20 Nippon Bayer Agrochem Co Ltd 殺センチュウ性トリフルオロブテン類
AU2001241195A1 (en) * 2000-03-17 2001-09-24 Nissan Chemical Industries Ltd. Pyrimidinone derivatives and herbicides
DE10034131A1 (de) * 2000-07-13 2002-01-24 Bayer Ag Heterocyclische Fluoralkenylthioether (II)
US7138404B2 (en) * 2001-05-23 2006-11-21 Hoffmann-La Roche Inc. 4-aminopyrimidine derivatives
DE10238725A1 (de) * 2002-08-23 2004-03-04 Bayer Cropscience Ag Substituierte Heterocyclypyrimidine
AU2003275242B2 (en) * 2002-09-27 2010-03-04 Merck Sharp & Dohme Corp. Substituted pyrimidines
AU2002953128A0 (en) * 2002-12-05 2002-12-19 Osmose (Australia) Pty Ltd Surface treatment for wood and wood products
EP1654249A1 (en) * 2003-08-07 2006-05-10 Pharmacia & Upjohn Company LLC Anthelmintic and insecticide pyrimidine derivatives
JP2007524694A (ja) * 2004-02-18 2007-08-30 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 殺虫および殺線虫性ジフルオロアルケン誘導体
JP5287033B2 (ja) * 2007-08-23 2013-09-11 住友化学株式会社 含フッ素有機硫黄化合物およびその有害節足動物防除剤
WO2010119879A1 (en) * 2009-04-16 2010-10-21 Sumitomo Chemical Company, Limited Pyrimidine compound and its use for pest control
WO2010119878A1 (en) * 2009-04-16 2010-10-21 Sumitomo Chemical Company, Limited Pyrimidine compound and its use for pest control
EP3728204A1 (en) 2017-12-20 2020-10-28 PI Industries Ltd. Fluoralkenyl compounds, process for preparation and use thereof
CN108314656B (zh) * 2018-02-27 2020-10-27 浙江工业大学 不饱和烃嘧啶硫醚类化合物及其制备方法与应用
CN115385862B (zh) * 2022-09-07 2023-03-28 贵州大学 一种含磺酸酯结构的嘧啶硫醚类化合物及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3223707A (en) * 1963-12-23 1965-12-14 Stauffer Chemical Co 2-(trifluorobutenylmercapto)-pyrimidines
AU549117B2 (en) * 1980-01-10 1986-01-16 Nyegaard & Co. A/S Pyrimidine-2-sulphides and their 5-oxides
EP0036839A2 (de) * 1980-03-20 1981-09-30 Ciba-Geigy Ag 4-N,N-Dimethylcarbamoyloxy-5-methyl-pyrimidine, Verfahren zu ihrer Herstellung und ihre Verwendung in der Schädlingsbekämpfung, sowie die als Zwischenprodukte verwendeten 4-Hydroxy-5-methyl-pyrimidine
EP0388838B1 (de) * 1989-03-22 1996-01-10 Ciba-Geigy Ag Schädlingsbekämpfungsmittel
EP0506270A1 (en) * 1991-03-28 1992-09-30 Zeneca Limited Nematocide pyrimidine derivatives
EP0506269A1 (en) * 1991-03-28 1992-09-30 Zeneca Limited Nematicide pyrimidine derivatives
GB9106609D0 (en) * 1991-03-28 1991-05-15 Ici Plc Heterocyclic compounds
GB9122098D0 (en) * 1991-10-17 1991-11-27 Ici Plc Fungicides

Also Published As

Publication number Publication date
EP0660827B1 (en) 1997-04-16
ZA936708B (en) 1994-05-19
GB2270688A (en) 1994-03-23
US5684011A (en) 1997-11-04
CN1098718A (zh) 1995-02-15
ATE151757T1 (de) 1997-05-15
GB9219635D0 (en) 1992-10-28
EP0660827A1 (en) 1995-07-05
WO1994006777A1 (en) 1994-03-31
JPH08503932A (ja) 1996-04-30
IL106970A0 (en) 1993-12-28
GB9318737D0 (en) 1993-10-27
AU4977793A (en) 1994-04-12
DK0660827T3 (da) 1997-10-27
DE69309941D1 (de) 1997-05-22
CN1041922C (zh) 1999-02-03
DE69309941T2 (de) 1997-09-04

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