ES2106682B1 - Nuevos derivados azo del acido 5-aminosalicilico. - Google Patents
Nuevos derivados azo del acido 5-aminosalicilico.Info
- Publication number
- ES2106682B1 ES2106682B1 ES9501752A ES9501752A ES2106682B1 ES 2106682 B1 ES2106682 B1 ES 2106682B1 ES 9501752 A ES9501752 A ES 9501752A ES 9501752 A ES9501752 A ES 9501752A ES 2106682 B1 ES2106682 B1 ES 2106682B1
- Authority
- ES
- Spain
- Prior art keywords
- alkyl
- cyclloalkyl
- aminosalicylic acid
- aryl
- new azo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- KBOPZPXVLCULAV-UHFFFAOYSA-N mesalamine Chemical class NC1=CC=C(O)C(C(O)=O)=C1 KBOPZPXVLCULAV-UHFFFAOYSA-N 0.000 title 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical group [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 4
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 239000001257 hydrogen Substances 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
COMPUESTOS DE FORMULA I, EN DONDE M REPRESENTA 1 O 2; R1 REPRESENTA C1-4 ALQUILO O C3-7 CICLOALQUILO; A, B Y C REPRESENTAN CR2, DONDE CADA R2 REPRESENTA HIDROGENO O C1-4 ALQUILO; A REPRESENTA -CO-, -SO2-, -NHCO- O -OCO-; B REPRESENTA UN GRUPO (I), (II), (III), (IV) O (V); N REPRESENTA 0-3; P REPRESENTA 0 O 1; R3 REPRESENTA HIDROGENO, C1-4 ALQUILO, C1-4 HALOALQUILO, C3-7 CICLOALQUILO, C1-4 ALCOXI-C1-4 ALQUILO O ARILO; R4 REPRESENTA HIDROGENO, C1-4 ALQUILO, -COOR5 O -CONR5R6, -NR5R6, -NR7C (=O) OR5, -NR7C (=O) R5, -NR7C (=O) NR5R6 O -NR7SO2R5; R5 REPRESENTA C1-4 ALQUILO, ARILO O ARIL C1-4 ALQUILO; R6 Y R7 REPRESENTAN HIDROGENO O C1-4 ALQUILO; Z REPRESENTA -OC(=O)-, -C(=O)-, -NR6C (=O)- O -SO2-; R8 REPRESENTA ARILO; R9 REPRESENTA C1-4 ALQUILO, C3-7 CICLOALQUILO, -C (=O) OR5, -C(=O)R5, -C(=O) NR5R6, O -SO2R5; Y R10 REPRESENTA C1-4 ALQUILO, C3-7 CICLOALQUILO, ARILO, O ARIL-C1-4 ALQUILO.
Priority Applications (18)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES9501752A ES2106682B1 (es) | 1995-09-08 | 1995-09-08 | Nuevos derivados azo del acido 5-aminosalicilico. |
| AU69875/96A AU6987596A (en) | 1995-09-08 | 1996-09-06 | Azo derivatives of 5-aminosalicylic acid for treatment of inflammatory bowel disease |
| PT96931039T PT790998E (pt) | 1995-09-08 | 1996-09-06 | Derivados azo do acido 5-aminosalicilico para o tratamento da doenca inflamatoria dos intestinos |
| CA002204747A CA2204747C (en) | 1995-09-08 | 1996-09-06 | New azo derivatives of 5-aminosalicylic acid |
| DK96931039T DK0790998T3 (da) | 1995-09-08 | 1996-09-06 | Azo-derivater af 5-aminosalicylsyre til behandling af inflammatorisk tarmsygdom |
| PCT/EP1996/003921 WO1997009329A1 (en) | 1995-09-08 | 1996-09-06 | Azo derivatives of 5-aminosalicylic acid for treatment of inflammatory bowel disease |
| US08/836,125 US5747477A (en) | 1995-09-08 | 1996-09-06 | Azo derivatives of 5-aminosalicylic acid |
| EP96931039A EP0790998B1 (en) | 1995-09-08 | 1996-09-06 | Azo derivatives of 5-aminosalicylic acid for treatment of inflammatory bowel disease |
| DE69611598T DE69611598T2 (de) | 1995-09-08 | 1996-09-06 | Azoderivate von 5-aminosalicylsäure zur behandlung von enzündlichen darmerkrankungen |
| ARP960104275A AR004198A1 (es) | 1995-09-08 | 1996-09-06 | Un compuesto azo del acido 5-aminosalicilico y procedimiento para preparar el mismo |
| AT96931039T ATE198751T1 (de) | 1995-09-08 | 1996-09-06 | Azoderivate von 5-aminosalicylsäure zur behandlung von enzündlichen darmerkrankungen |
| KR1019970703002A KR100481300B1 (ko) | 1995-09-08 | 1996-09-06 | 염증성장질환치료용의5-아미노살리실산의아조유도체 |
| MX9702919A MX9702919A (es) | 1995-09-08 | 1996-09-06 | Derivados azo del acido 5-aminosalicilico para el tratameitno de la enfermedad inflamatoria intestinal. |
| JP51087597A JP4115522B2 (ja) | 1995-09-08 | 1996-09-06 | 新規な５−アミノサリチル酸のアゾ誘導体 |
| ES96931039T ES2155621T3 (es) | 1995-09-08 | 1996-09-06 | Derivados azo del acido 5-aminosalicilico para el tratamiento de la enfermedad inflamatoria intestinal. |
| BR9606628A BR9606628A (pt) | 1995-09-08 | 1996-09-06 | Novos derivados azo de ácido 5-aminosalicílico |
| NO972113A NO308850B1 (no) | 1995-09-08 | 1997-05-07 | Nye azoderivater av 5-aminosalicylsyre, anvendelse av disse og farmasøytisk preparat inneholdende dem |
| GR20010400467T GR3035622T3 (en) | 1995-09-08 | 2001-03-23 | Azo derivatives of 5-aminosalicylic acid for treatment of inflammatory bowel disease |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES9501752A ES2106682B1 (es) | 1995-09-08 | 1995-09-08 | Nuevos derivados azo del acido 5-aminosalicilico. |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES2106682A1 ES2106682A1 (es) | 1997-11-01 |
| ES2106682B1 true ES2106682B1 (es) | 1998-07-01 |
Family
ID=8291526
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES9501752A Expired - Fee Related ES2106682B1 (es) | 1995-09-08 | 1995-09-08 | Nuevos derivados azo del acido 5-aminosalicilico. |
Country Status (1)
| Country | Link |
|---|---|
| ES (1) | ES2106682B1 (es) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4312806A (en) * | 1981-03-02 | 1982-01-26 | G. D. Searle & Co. | Method and compounds for treating inflammatory bowel disease |
| PT98673B (pt) * | 1990-08-15 | 1999-01-29 | British Bio Technology | Processo para a preparacao de compostos que sao antagonistas do factor de activacao de plaquetas por exemplo derivados de benzimidazole e de seus intermediarios |
-
1995
- 1995-09-08 ES ES9501752A patent/ES2106682B1/es not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| ES2106682A1 (es) | 1997-11-01 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| YU20094A (sh) | Hidrazidi 1-h-indol-3-sirćetne kisleine kao inhibitori spla2 | |
| ES8801193A1 (es) | Procedimiento para la preparacion de carbamatos de fenilo | |
| ATE147067T1 (de) | Selektive n-acylation von aminoalkoholen | |
| SE8302172D0 (sv) | Forfarande for framstellning av nya acetohydroxamsyror | |
| NO951543L (no) | Polyenforbindelser, farmasöytiske og kosmetiske preparater inneholdende disse, og deres anvendelser | |
| ES2045481T3 (es) | Procedimiento para la preparacion de sulfatos ciclicos. | |
| CO4700469A1 (es) | 3-[4-(4(4-cianofenil)-1-piperazinanil)butil]-5]ciannoindol y su proceso de obtencion . | |
| AR247732A1 (es) | Procedimiento para obtener amidas de acido piridin-2, 4- y -2, 5-dicarboxilico | |
| ES8507112A1 (es) | Un procedimiento para la prpeparacion de compuestos de 1,4-dihidropiridina. | |
| IS4133A (is) | Aðferð við framleiðslu á nýjum afleiðum af 3-hýdroxýantraniliksýru og milliefni við framleiðslu þeirra | |
| ATE224872T1 (de) | Azetidinonderivate zur behandlung von hcmv entzündungen | |
| DK0677042T3 (da) | Selektive ligander af 5HT1D-5HT1B-receptorer, der er afledt af indolpiperazin og er nyttige som lægemidler | |
| ES8702343A1 (es) | Un procedimiento para la produccion de un derivado de diami-das de n-acilaminoacidos | |
| KR850000755B1 (en) | Process for preparing 3,1-benzoxazin-2-ones and acid addition salts thereof | |
| FI830810A0 (fi) | Pyridinkarboxylsyraestrar, foerfarande foer deras framstaellning och deras anvaendning som laekemed | |
| ES2106682B1 (es) | Nuevos derivados azo del acido 5-aminosalicilico. | |
| ES2058177T3 (es) | Nuevos derivados de alcanosulfonanilida, procedimientos para su preparacion y composiciones farmaceuticas que los contienen. | |
| TW324007B (en) | N-substituted diazabicycloheptane derivative and its pharmaceutical use | |
| NO995289D0 (no) | Benzimidazol-derivater | |
| ES8505369A1 (es) | Un procedimiento para la preparacion de derivados de pirimidona | |
| YU46193B (sh) | Postupak za dobijanje derivata benzimidazol-2-sulfonamida i imidazopiridin-2-sulfonamida | |
| ATE3803T1 (de) | Verfahren und mittel zum schutz von pflanzenkulturen vor der phytotoxischen wirkung starker herbizide; oximaetherderivate. | |
| DK1205476T3 (da) | Fremgangsmåde til syntese af N-(mercaptoacyl)-aminosyrederivater ud fra alfa-substituerede acrylsyrer | |
| DE69303721D1 (de) | Herbizide pyranolyloxy-picolinamide | |
| ES2190781T3 (es) | Derivados de 1-trifluorometil-4-hidroxi-7-piperidinil-aminometilcromano. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EC2A | Search report published |
Date of ref document: 19971101 Kind code of ref document: A1 Effective date: 19971101 |
|
| FD1A | Patent lapsed |
Effective date: 20100623 |