ES2170259T3 - Empleo de lipidos como agentes auxiliares en la obtencion de formas farmaceuticas solidas segun el procedimiento de extrusion en fusion. - Google Patents
Empleo de lipidos como agentes auxiliares en la obtencion de formas farmaceuticas solidas segun el procedimiento de extrusion en fusion.Info
- Publication number
- ES2170259T3 ES2170259T3 ES96929292T ES96929292T ES2170259T3 ES 2170259 T3 ES2170259 T3 ES 2170259T3 ES 96929292 T ES96929292 T ES 96929292T ES 96929292 T ES96929292 T ES 96929292T ES 2170259 T3 ES2170259 T3 ES 2170259T3
- Authority
- ES
- Spain
- Prior art keywords
- lipids
- employment
- forms according
- auxiliary agents
- solid pharmaceutical
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
USO DE LIPIDOS COMO ADYUVANTES EN LA PRODUCCION DE FORMAS MEDICAMENTOSAS SOLIDAS SEGUN EL PROCEDIMIENTO DE EXTRUSION DE LA MASA FUNDIDA.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19531277A DE19531277A1 (de) | 1995-08-25 | 1995-08-25 | Verwendung von Lipiden als Hilfsmittel bei der Herstellung von festen Arzneiformen nach dem Schmelzextrusionsverfahren |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2170259T3 true ES2170259T3 (es) | 2002-08-01 |
Family
ID=7770352
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES96929292T Expired - Lifetime ES2170259T3 (es) | 1995-08-25 | 1996-08-21 | Empleo de lipidos como agentes auxiliares en la obtencion de formas farmaceuticas solidas segun el procedimiento de extrusion en fusion. |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US6387401B2 (es) |
| EP (1) | EP0845982B1 (es) |
| AR (1) | AR003345A1 (es) |
| AT (1) | ATE210970T1 (es) |
| AU (1) | AU6875396A (es) |
| BR (1) | BR9610234A (es) |
| CA (1) | CA2227272C (es) |
| DE (2) | DE19531277A1 (es) |
| DK (1) | DK0845982T3 (es) |
| ES (1) | ES2170259T3 (es) |
| HR (1) | HRP960381A2 (es) |
| WO (1) | WO1997007786A2 (es) |
| ZA (1) | ZA967170B (es) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU1787800A (en) * | 1998-12-08 | 2000-06-26 | Phares Pharmaceutical Research N.V. | Phospholipid compositions |
| DE19916383A1 (de) * | 1999-03-31 | 2000-10-05 | Schering Ag | Pharmazeutische Zusammensetzung mit einem Extrusionsstoff |
| NZ516733A (en) * | 1999-07-30 | 2004-03-26 | Smithkline Beecham Plc | Pharmaceutical formulations for oral dosing that are dosage forms comprising two or more connected sub-units |
| US7364752B1 (en) | 1999-11-12 | 2008-04-29 | Abbott Laboratories | Solid dispersion pharamaceutical formulations |
| WO2001034119A2 (en) * | 1999-11-12 | 2001-05-17 | Abbott Laboratories | Inhibitors of crystallization in a solid dispersion |
| DE10026698A1 (de) * | 2000-05-30 | 2001-12-06 | Basf Ag | Selbstemulgierende Wirkstoffformulierung und Verwendung dieser Formulierung |
| DE10026699A1 (de) * | 2000-05-30 | 2001-12-06 | Basf Ag | Formulierung auf Heparin-, Glycosaminoglycan- oder Heparinoidbasis und Verwendung der Formulierung sowie der Formulierungsgrundlage |
| US7883721B2 (en) | 2001-01-30 | 2011-02-08 | Smithkline Beecham Limited | Pharmaceutical formulation |
| GB0102342D0 (en) | 2001-01-30 | 2001-03-14 | Smithkline Beecham Plc | Pharmaceutical formulation |
| US7842308B2 (en) | 2001-01-30 | 2010-11-30 | Smithkline Beecham Limited | Pharmaceutical formulation |
| US20050175687A1 (en) * | 2001-01-30 | 2005-08-11 | Mcallister Stephen M. | Pharmaceutical formulations |
| TW200526274A (en) | 2003-07-21 | 2005-08-16 | Smithkline Beecham Plc | Pharmaceutical formulations |
| US8377952B2 (en) * | 2003-08-28 | 2013-02-19 | Abbott Laboratories | Solid pharmaceutical dosage formulation |
| US8025899B2 (en) | 2003-08-28 | 2011-09-27 | Abbott Laboratories | Solid pharmaceutical dosage form |
| CA2549225A1 (en) * | 2003-12-04 | 2005-06-16 | Pfizer Products Inc. | Spray-congeal process using an extruder for preparing multiparticulate crystalline drug compositions containing preferably a poloxamer and a glyceride |
| PE20060003A1 (es) * | 2004-03-12 | 2006-03-01 | Smithkline Beecham Plc | Formulacion farmaceutica polimerica para moldear por inyeccion |
| CA2560165A1 (en) * | 2004-05-04 | 2005-11-10 | Boehringer Ingelheim International Gmbh | Solid pharmaceutical form comprising an ltb4 antagonist |
| EP1693045A1 (de) | 2005-02-17 | 2006-08-23 | Abbott GmbH & Co. KG | Herstellung von Dosierungsformen aus wirkstoffhaltigen Schmelzen |
| SI2200588T1 (sl) * | 2007-09-25 | 2019-08-30 | Solubest Ltd. | Sestavki, ki obsegajo lipofilne aktivne spojine, in postopek za njihovo pripravo |
| JP2011503048A (ja) | 2007-11-08 | 2011-01-27 | グラクソ グループ リミテッド | 医薬製剤 |
| WO2009150228A2 (en) * | 2008-06-13 | 2009-12-17 | Glaxo Group Limited | Pharmaceutical formulations |
| AU2011306065B2 (en) | 2010-09-22 | 2015-03-19 | Mcneil-Ppc, Inc. | Manufacture of tablets from energy-applied powder blend |
| AT511581A1 (de) * | 2011-05-26 | 2012-12-15 | G L Pharma Gmbh | Orale retardierende formulierung |
| US9511028B2 (en) | 2012-05-01 | 2016-12-06 | Johnson & Johnson Consumer Inc. | Orally disintegrating tablet |
| DE102017106216A1 (de) * | 2017-03-22 | 2018-09-27 | Amw Gmbh | Extrudierte Depotform zur anhaltenden Wirkstofffreisetzung |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2581541B1 (fr) | 1985-05-09 | 1988-05-20 | Rhone Poulenc Sante | Nouvelles compositions pharmaceutiques permettant la liberation prolongee d'un principe actif et leur procede de preparation |
| DE4226753A1 (de) | 1992-08-13 | 1994-02-17 | Basf Ag | Wirkstoffe enthaltende Zubereitungen in Form fester Teilchen |
| CA2182282C (en) | 1994-02-16 | 2006-04-18 | Jacqueline E. Briskin | Process for preparing fine particle pharmaceutical formulations |
| DE4413350A1 (de) * | 1994-04-18 | 1995-10-19 | Basf Ag | Retard-Matrixpellets und Verfahren zu ihrer Herstellung |
| US5965161A (en) * | 1994-11-04 | 1999-10-12 | Euro-Celtique, S.A. | Extruded multi-particulates |
| DE19504832A1 (de) * | 1995-02-14 | 1996-08-22 | Basf Ag | Feste Wirkstoff-Zubereitungen |
-
1995
- 1995-08-25 DE DE19531277A patent/DE19531277A1/de not_active Withdrawn
-
1996
- 1996-08-20 HR HR19531277.5A patent/HRP960381A2/hr not_active Application Discontinuation
- 1996-08-21 AT AT96929292T patent/ATE210970T1/de not_active IP Right Cessation
- 1996-08-21 AU AU68753/96A patent/AU6875396A/en not_active Abandoned
- 1996-08-21 DE DE59608516T patent/DE59608516D1/de not_active Expired - Lifetime
- 1996-08-21 BR BR9610234A patent/BR9610234A/pt not_active Application Discontinuation
- 1996-08-21 CA CA002227272A patent/CA2227272C/en not_active Expired - Lifetime
- 1996-08-21 DK DK96929292T patent/DK0845982T3/da active
- 1996-08-21 ES ES96929292T patent/ES2170259T3/es not_active Expired - Lifetime
- 1996-08-21 WO PCT/EP1996/003667 patent/WO1997007786A2/de not_active Ceased
- 1996-08-21 US US09/000,389 patent/US6387401B2/en not_active Expired - Lifetime
- 1996-08-21 EP EP96929292A patent/EP0845982B1/de not_active Expired - Lifetime
- 1996-08-23 ZA ZA9607170A patent/ZA967170B/xx unknown
- 1996-08-23 AR ARP960104102A patent/AR003345A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ATE210970T1 (de) | 2002-01-15 |
| DE19531277A1 (de) | 1997-02-27 |
| US20010007664A1 (en) | 2001-07-12 |
| WO1997007786A2 (de) | 1997-03-06 |
| DK0845982T3 (da) | 2002-03-25 |
| WO1997007786A3 (de) | 1997-04-03 |
| US6387401B2 (en) | 2002-05-14 |
| CA2227272A1 (en) | 1997-03-06 |
| EP0845982A2 (de) | 1998-06-10 |
| EP0845982B1 (de) | 2001-12-19 |
| HRP960381A2 (en) | 1998-02-28 |
| AR003345A1 (es) | 1998-07-08 |
| AU6875396A (en) | 1997-03-19 |
| ZA967170B (en) | 1998-03-02 |
| BR9610234A (pt) | 1999-06-29 |
| DE59608516D1 (de) | 2002-01-31 |
| CA2227272C (en) | 2007-12-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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