ES2193380T3 - Dihidropiranos condesados en el anillo, procedimiento para su preparacion, asi como su utilizacion. - Google Patents
Dihidropiranos condesados en el anillo, procedimiento para su preparacion, asi como su utilizacion.Info
- Publication number
- ES2193380T3 ES2193380T3 ES97928221T ES97928221T ES2193380T3 ES 2193380 T3 ES2193380 T3 ES 2193380T3 ES 97928221 T ES97928221 T ES 97928221T ES 97928221 T ES97928221 T ES 97928221T ES 2193380 T3 ES2193380 T3 ES 2193380T3
- Authority
- ES
- Spain
- Prior art keywords
- preparation
- dihydropirans
- condesated
- procedure
- ring
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 238000000034 method Methods 0.000 title abstract 2
- 238000002360 preparation method Methods 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 1
- 238000010532 solid phase synthesis reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Immunology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Biomedical Technology (AREA)
- Vascular Medicine (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyrane Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Epoxy Compounds (AREA)
Abstract
EL OBJETO DE LA INVENCION SON COMPUESTOS DE FORMULA (I), EN LA CUAL LOS RADICALES R 1 , R 2 , R 3 Y A TIENEN LOS SIGNIFICADOS INDICADOS EN LA DESCRIPCION. LA INVENCION TAMBIEN TRATA DE UN PROCEDIMIENTO PARA LA OBTENCION DE LOS COMPUESTOS DE FORMULA (I) MEDIANTE SINTESIS EN FASE SOLIDA ASI COMO SU UTILIZACION COMO MEDICAMENTOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19624154A DE19624154A1 (de) | 1996-06-18 | 1996-06-18 | Ringannelierte Dihydropyrane, Verfahren zur Herstellung sowie deren Verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2193380T3 true ES2193380T3 (es) | 2003-11-01 |
Family
ID=7797180
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES97928221T Expired - Lifetime ES2193380T3 (es) | 1996-06-18 | 1997-06-18 | Dihidropiranos condesados en el anillo, procedimiento para su preparacion, asi como su utilizacion. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US6399653B1 (es) |
| EP (1) | EP0906303B1 (es) |
| JP (1) | JP4181219B2 (es) |
| AT (1) | ATE236895T1 (es) |
| AU (1) | AU3259997A (es) |
| CA (1) | CA2258539C (es) |
| DE (2) | DE19624154A1 (es) |
| DK (1) | DK0906303T3 (es) |
| ES (1) | ES2193380T3 (es) |
| PT (1) | PT906303E (es) |
| WO (1) | WO1997048691A1 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100405893B1 (ko) | 1995-10-23 | 2004-10-06 | 가부시끼가이샤 히다치 세이사꾸쇼 | 액정표시장치 |
| HRP20010414A2 (en) * | 1998-12-02 | 2002-06-30 | Pfizer Prod Inc | METHODS AND COMPOSITIONS FOR RESTORING CONFORMATIONAL STABILITY OF A PROTEIN OF THE p53 FAMILY |
| ME00059B (me) * | 2004-02-20 | 2010-06-10 | Oksidekahidronaftalen modulatori hm74 | |
| US7723342B2 (en) * | 2005-05-17 | 2010-05-25 | Schering Corporation | Heterocycles as nicotinic acid receptor agonists for the treatment of dyslipidemia |
| US7737155B2 (en) * | 2005-05-17 | 2010-06-15 | Schering Corporation | Nitrogen-containing heterocyclic compounds and methods of use thereof |
| US7750015B2 (en) * | 2005-05-17 | 2010-07-06 | Schering Corporation | Nitrogen-containing heterocyclic compounds and methods of use thereof |
| KR20080091814A (ko) * | 2006-01-20 | 2008-10-14 | 쉐링 코포레이션 | 지질혈증장애의 치료를 위한 니코틴산 수용체 효능제로서의헤테로사이클 |
| US11932655B1 (en) | 2023-10-17 | 2024-03-19 | King Faisal University | 12-bromo-2,16-dioxapentacyclo[7.7.5.01,21.03,8.010,15]henicosa3(8),10,12,14-tetraene-7,20-dione as an antimicrobial compound |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3775435A (en) * | 1971-08-26 | 1973-11-27 | American Home Prod | 5,6,7,8-tetrahydro-2,5(and 4,5)-dioxo-1-benzopyrans |
| GB9318431D0 (en) | 1993-09-06 | 1993-10-20 | Boots Co Plc | Therapeutic agents |
-
1996
- 1996-06-18 DE DE19624154A patent/DE19624154A1/de not_active Withdrawn
-
1997
- 1997-06-18 AU AU32599/97A patent/AU3259997A/en not_active Abandoned
- 1997-06-18 CA CA002258539A patent/CA2258539C/en not_active Expired - Fee Related
- 1997-06-18 ES ES97928221T patent/ES2193380T3/es not_active Expired - Lifetime
- 1997-06-18 JP JP50225198A patent/JP4181219B2/ja not_active Expired - Fee Related
- 1997-06-18 PT PT97928221T patent/PT906303E/pt unknown
- 1997-06-18 WO PCT/EP1997/003146 patent/WO1997048691A1/de not_active Ceased
- 1997-06-18 AT AT97928221T patent/ATE236895T1/de active
- 1997-06-18 DE DE59709792T patent/DE59709792D1/de not_active Expired - Lifetime
- 1997-06-18 EP EP97928221A patent/EP0906303B1/de not_active Expired - Lifetime
- 1997-06-18 DK DK97928221T patent/DK0906303T3/da active
-
2000
- 2000-06-30 US US09/609,594 patent/US6399653B1/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP0906303B1 (de) | 2003-04-09 |
| CA2258539A1 (en) | 1997-12-24 |
| JP4181219B2 (ja) | 2008-11-12 |
| CA2258539C (en) | 2009-06-02 |
| PT906303E (pt) | 2003-08-29 |
| AU3259997A (en) | 1998-01-07 |
| US6399653B1 (en) | 2002-06-04 |
| EP0906303A1 (de) | 1999-04-07 |
| DE59709792D1 (de) | 2003-05-15 |
| DE19624154A1 (de) | 1998-01-08 |
| JP2000512305A (ja) | 2000-09-19 |
| WO1997048691A1 (de) | 1997-12-24 |
| DK0906303T3 (da) | 2003-07-28 |
| ATE236895T1 (de) | 2003-04-15 |
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