ES2193380T3 - Dihidropiranos condesados en el anillo, procedimiento para su preparacion, asi como su utilizacion. - Google Patents
Dihidropiranos condesados en el anillo, procedimiento para su preparacion, asi como su utilizacion.Info
- Publication number
- ES2193380T3 ES2193380T3 ES97928221T ES97928221T ES2193380T3 ES 2193380 T3 ES2193380 T3 ES 2193380T3 ES 97928221 T ES97928221 T ES 97928221T ES 97928221 T ES97928221 T ES 97928221T ES 2193380 T3 ES2193380 T3 ES 2193380T3
- Authority
- ES
- Spain
- Prior art keywords
- preparation
- dihydropirans
- condesated
- procedure
- ring
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 238000000034 method Methods 0.000 title abstract 2
- 238000002360 preparation method Methods 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 1
- 238000010532 solid phase synthesis reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Vascular Medicine (AREA)
- Oncology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Communicable Diseases (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyrane Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Processing And Handling Of Plastics And Other Materials For Molding In General (AREA)
Abstract
EL OBJETO DE LA INVENCION SON COMPUESTOS DE FORMULA (I), EN LA CUAL LOS RADICALES R 1 , R 2 , R 3 Y A TIENEN LOS SIGNIFICADOS INDICADOS EN LA DESCRIPCION. LA INVENCION TAMBIEN TRATA DE UN PROCEDIMIENTO PARA LA OBTENCION DE LOS COMPUESTOS DE FORMULA (I) MEDIANTE SINTESIS EN FASE SOLIDA ASI COMO SU UTILIZACION COMO MEDICAMENTOS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19624154A DE19624154A1 (de) | 1996-06-18 | 1996-06-18 | Ringannelierte Dihydropyrane, Verfahren zur Herstellung sowie deren Verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2193380T3 true ES2193380T3 (es) | 2003-11-01 |
Family
ID=7797180
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES97928221T Expired - Lifetime ES2193380T3 (es) | 1996-06-18 | 1997-06-18 | Dihidropiranos condesados en el anillo, procedimiento para su preparacion, asi como su utilizacion. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US6399653B1 (es) |
| EP (1) | EP0906303B1 (es) |
| JP (1) | JP4181219B2 (es) |
| AT (1) | ATE236895T1 (es) |
| AU (1) | AU3259997A (es) |
| CA (1) | CA2258539C (es) |
| DE (2) | DE19624154A1 (es) |
| DK (1) | DK0906303T3 (es) |
| ES (1) | ES2193380T3 (es) |
| PT (1) | PT906303E (es) |
| WO (1) | WO1997048691A1 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6137560A (en) | 1995-10-23 | 2000-10-24 | Hitachi, Ltd. | Active matrix type liquid crystal display apparatus with light source color compensation |
| CN1329493A (zh) * | 1998-12-02 | 2002-01-02 | 辉瑞产品公司 | 恢复p53家族蛋白质的构象稳定性的方法和组合物 |
| CN1929833A (zh) * | 2004-02-20 | 2007-03-14 | 安万特药物公司 | Hm74的氧杂十氢萘调节剂 |
| US7737155B2 (en) * | 2005-05-17 | 2010-06-15 | Schering Corporation | Nitrogen-containing heterocyclic compounds and methods of use thereof |
| US7750015B2 (en) * | 2005-05-17 | 2010-07-06 | Schering Corporation | Nitrogen-containing heterocyclic compounds and methods of use thereof |
| US7723342B2 (en) * | 2005-05-17 | 2010-05-25 | Schering Corporation | Heterocycles as nicotinic acid receptor agonists for the treatment of dyslipidemia |
| CA2637717A1 (en) * | 2006-01-20 | 2007-08-02 | Schering Corporation | Heterocycles as nicotinic acid receptor agonists for the treatment of dyyslipidemia |
| US11932655B1 (en) | 2023-10-17 | 2024-03-19 | King Faisal University | 12-bromo-2,16-dioxapentacyclo[7.7.5.01,21.03,8.010,15]henicosa3(8),10,12,14-tetraene-7,20-dione as an antimicrobial compound |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3775435A (en) * | 1971-08-26 | 1973-11-27 | American Home Prod | 5,6,7,8-tetrahydro-2,5(and 4,5)-dioxo-1-benzopyrans |
| GB9318431D0 (en) | 1993-09-06 | 1993-10-20 | Boots Co Plc | Therapeutic agents |
-
1996
- 1996-06-18 DE DE19624154A patent/DE19624154A1/de not_active Withdrawn
-
1997
- 1997-06-18 AT AT97928221T patent/ATE236895T1/de active
- 1997-06-18 CA CA002258539A patent/CA2258539C/en not_active Expired - Fee Related
- 1997-06-18 JP JP50225198A patent/JP4181219B2/ja not_active Expired - Fee Related
- 1997-06-18 ES ES97928221T patent/ES2193380T3/es not_active Expired - Lifetime
- 1997-06-18 DK DK97928221T patent/DK0906303T3/da active
- 1997-06-18 DE DE59709792T patent/DE59709792D1/de not_active Expired - Lifetime
- 1997-06-18 WO PCT/EP1997/003146 patent/WO1997048691A1/de not_active Ceased
- 1997-06-18 AU AU32599/97A patent/AU3259997A/en not_active Abandoned
- 1997-06-18 EP EP97928221A patent/EP0906303B1/de not_active Expired - Lifetime
- 1997-06-18 PT PT97928221T patent/PT906303E/pt unknown
-
2000
- 2000-06-30 US US09/609,594 patent/US6399653B1/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| AU3259997A (en) | 1998-01-07 |
| WO1997048691A1 (de) | 1997-12-24 |
| DK0906303T3 (da) | 2003-07-28 |
| EP0906303B1 (de) | 2003-04-09 |
| DE19624154A1 (de) | 1998-01-08 |
| JP2000512305A (ja) | 2000-09-19 |
| PT906303E (pt) | 2003-08-29 |
| ATE236895T1 (de) | 2003-04-15 |
| JP4181219B2 (ja) | 2008-11-12 |
| US6399653B1 (en) | 2002-06-04 |
| EP0906303A1 (de) | 1999-04-07 |
| DE59709792D1 (de) | 2003-05-15 |
| CA2258539C (en) | 2009-06-02 |
| CA2258539A1 (en) | 1997-12-24 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK0640592T3 (da) | N-acylerede tricycliske azaheteroringe anvendelige som vasopressin-antagonister | |
| ATE469892T1 (de) | Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung | |
| SV2002000249A (es) | Derivados de tiazolilamida ref, lea 34082-sv | |
| SV2003001172A (es) | 2-tio-3,5-diciano-4-fenil-6-aminopiridinas substituidas y su uso ref. lea 35510-sv | |
| SV1999000047A (es) | Nuevas dihidropirimidinas fef. lea 32792-sv | |
| AR025739A1 (es) | Nuevos derivados de bencimidazolonas que tienen afinidad para receptores mezclados de serotonina y dopamina | |
| TNSN05007A1 (en) | Novel thiophenylglycoside derivatives, methods for production thereof, medicaments comprising said compounds and use thereof. | |
| ES2178055T3 (es) | Derivados aminicos substituidos, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. | |
| ES2172937T3 (es) | 21-hidroxi-6,19-oxidoprogesterona(21oh-6op) como medicamento para tratar el exceso de glucocorticoides. | |
| CR9182A (es) | Derivado de quinolina, su uso, preparacion y medicamento que lo contiene | |
| UY26133A1 (es) | Derivado sustituido de pirazol. | |
| ES2193380T3 (es) | Dihidropiranos condesados en el anillo, procedimiento para su preparacion, asi como su utilizacion. | |
| AR006058A1 (es) | Procedimientos para preparar compuestos de dicianoacetato y de 1,2-pirazol-5-amino-3-substituido | |
| EA200100040A1 (ru) | Химический синтез морфолиновых производных | |
| AP2001002188A0 (en) | 5HT1 antagonists for antidepressant therapy. | |
| AR017997A3 (es) | Procedimiento para preparar compuestos aza ciclohexapeptidos y compuestos para su exclusivo uso en dicho procedimiento | |
| PA8571401A1 (es) | Imidazolinilmetil aralquilsulfonamidas | |
| ES2057322T3 (es) | Derivados de amida de aminoacido substituidos, su fabricacion y uso. | |
| AR028947A1 (es) | Compuestos novedosos | |
| ES2179864T3 (es) | 4-benzoil-isoxazoles y su uso como herbicidas. | |
| ES2185196T3 (es) | Un procedimiento para la preparacion de tetraazamacrociclos. | |
| AR003977A1 (es) | Composiciones endoparasiticidas a base de didepsipeptidos, nuevos didepsipeptidos y procedimientos para su produccion. | |
| ES2145480T3 (es) | Amidas de acido carbamoilcarboxilico. | |
| DE69808922D1 (de) | Thiazolobenzoheterocyclen, ihre herstellung und diese enthaltende phatrmazeutische zubereitungen | |
| YU100202A (sh) | Bifunkcionalni agensi koji poseduju antioksidantnu i antiaritmičku aktivnost |