ES2194744T3 - Derivados de quinocardina, su procedimiento de preparacion y su aplicacion como antifungicos. - Google Patents
Derivados de quinocardina, su procedimiento de preparacion y su aplicacion como antifungicos.Info
- Publication number
- ES2194744T3 ES2194744T3 ES00940456T ES00940456T ES2194744T3 ES 2194744 T3 ES2194744 T3 ES 2194744T3 ES 00940456 T ES00940456 T ES 00940456T ES 00940456 T ES00940456 T ES 00940456T ES 2194744 T3 ES2194744 T3 ES 2194744T3
- Authority
- ES
- Spain
- Prior art keywords
- derivatives
- application
- preparation procedure
- quinocardine
- antifungicos
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 150000001875 compounds Chemical class 0.000 abstract 3
- 229940121375 antifungal agent Drugs 0.000 abstract 2
- 239000003429 antifungal agent Substances 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- SYSQUGFVNFXIIT-UHFFFAOYSA-N n-[4-(1,3-benzoxazol-2-yl)phenyl]-4-nitrobenzenesulfonamide Chemical class C1=CC([N+](=O)[O-])=CC=C1S(=O)(=O)NC1=CC=C(C=2OC3=CC=CC=C3N=2)C=C1 SYSQUGFVNFXIIT-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Biochemistry (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Derivados de equinocardina, su procedimiento de preparación y su aplicación como antifúngicos. En el estado de la técnica ya fue descrita la utilización de compuestos ciclohexapeptídicos como agentes antifúngicos. Igualmente, ciertos compuestos ciclohexapeptídicos se pueden utilizar como agentes antimicrobianos. La invención tiene como objeto, en todas las formas posibles de isómeros así como sus mezclas, compuestos de fórmula (I).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9907252A FR2794747B1 (fr) | 1999-06-09 | 1999-06-09 | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2194744T3 true ES2194744T3 (es) | 2003-12-01 |
Family
ID=9546549
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES00940456T Expired - Lifetime ES2194744T3 (es) | 1999-06-09 | 2000-06-08 | Derivados de quinocardina, su procedimiento de preparacion y su aplicacion como antifungicos. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7005417B1 (es) |
| EP (1) | EP1189932B1 (es) |
| JP (1) | JP4619592B2 (es) |
| AR (1) | AR024315A1 (es) |
| AT (1) | ATE240971T1 (es) |
| AU (1) | AU5539100A (es) |
| CA (1) | CA2376490A1 (es) |
| CO (1) | CO5200761A1 (es) |
| DE (1) | DE60002866T2 (es) |
| DK (1) | DK1189932T3 (es) |
| ES (1) | ES2194744T3 (es) |
| FR (1) | FR2794747B1 (es) |
| GT (1) | GT200000090A (es) |
| PE (1) | PE20010234A1 (es) |
| PT (1) | PT1189932E (es) |
| TN (1) | TNSN00127A1 (es) |
| UY (1) | UY26195A1 (es) |
| WO (1) | WO2000075178A1 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA72200C2 (uk) * | 1997-12-10 | 2005-02-15 | Авентіс Фарма С.А. | Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція |
| FR2794746B1 (fr) * | 1999-06-09 | 2002-12-06 | Hoechst Marion Roussel Inc | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
| FR2833596B1 (fr) * | 2001-12-14 | 2005-02-18 | Aventis Pharma Sa | Procede de preparation de derives d'echinocandine |
| DE102004060750A1 (de) | 2004-12-15 | 2006-07-13 | Sanofi-Aventis Deutschland Gmbh | Verfahren zur Deacylierung von Lipopeptiden |
| US8853392B2 (en) | 2007-06-03 | 2014-10-07 | Vanderbilt University | Benzamide mGluR5 positive allosteric modulators and methods of making and using same |
| US8034806B2 (en) | 2007-11-02 | 2011-10-11 | Vanderbilt University | Bicyclic mGluR5 positive allosteric modulators and methods of making and using same |
| HUE029720T2 (en) * | 2011-09-09 | 2017-03-28 | Sandoz Ag | Preparation of micafungin intermediates |
| WO2016056023A2 (en) * | 2014-10-07 | 2016-04-14 | Alaparthi Lakshmi Prasad | Intermediates and processes to prepare micafungin |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL109615A (en) * | 1993-05-17 | 2000-12-06 | Fujisawa Pharmaceutical Co | Cyclic polypeptide derivatives processes for the preparation thereof and pharmaceutical compositions containing the same |
| US5516756A (en) * | 1994-10-31 | 1996-05-14 | Merck & Co., Inc. | Aza cyclohexapeptide compounds |
| US5646111A (en) * | 1995-04-07 | 1997-07-08 | Eli Lilly And Company | Cyclic peptide antifungal Agents |
| AUPO381496A0 (en) * | 1996-11-25 | 1996-12-19 | Fujisawa Pharmaceutical Co., Ltd. | New compound |
| UA72200C2 (uk) * | 1997-12-10 | 2005-02-15 | Авентіс Фарма С.А. | Похідні ехінокандину, спосіб їх одержання, їх застосування, проміжні сполуки та фармацевтична композиція |
-
1999
- 1999-06-09 FR FR9907252A patent/FR2794747B1/fr not_active Expired - Fee Related
-
2000
- 2000-06-06 TN TNTNSN00127A patent/TNSN00127A1/fr unknown
- 2000-06-07 UY UY26195A patent/UY26195A1/es not_active Application Discontinuation
- 2000-06-07 AR ARP000102834A patent/AR024315A1/es unknown
- 2000-06-07 PE PE2000000567A patent/PE20010234A1/es not_active Application Discontinuation
- 2000-06-08 DK DK00940456T patent/DK1189932T3/da active
- 2000-06-08 CA CA002376490A patent/CA2376490A1/fr not_active Abandoned
- 2000-06-08 AU AU55391/00A patent/AU5539100A/en not_active Abandoned
- 2000-06-08 GT GT200000090A patent/GT200000090A/es unknown
- 2000-06-08 WO PCT/FR2000/001569 patent/WO2000075178A1/fr not_active Ceased
- 2000-06-08 PT PT00940456T patent/PT1189932E/pt unknown
- 2000-06-08 AT AT00940456T patent/ATE240971T1/de not_active IP Right Cessation
- 2000-06-08 ES ES00940456T patent/ES2194744T3/es not_active Expired - Lifetime
- 2000-06-08 DE DE60002866T patent/DE60002866T2/de not_active Expired - Lifetime
- 2000-06-08 EP EP00940456A patent/EP1189932B1/fr not_active Expired - Lifetime
- 2000-06-08 JP JP2001502459A patent/JP4619592B2/ja not_active Expired - Fee Related
- 2000-06-08 US US10/009,407 patent/US7005417B1/en not_active Expired - Fee Related
- 2000-06-09 CO CO00042902A patent/CO5200761A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ATE240971T1 (de) | 2003-06-15 |
| JP2003504309A (ja) | 2003-02-04 |
| PE20010234A1 (es) | 2001-02-24 |
| EP1189932B1 (fr) | 2003-05-21 |
| EP1189932A1 (fr) | 2002-03-27 |
| AR024315A1 (es) | 2002-09-25 |
| CO5200761A1 (es) | 2002-09-27 |
| TNSN00127A1 (fr) | 2005-11-10 |
| WO2000075178A1 (fr) | 2000-12-14 |
| JP4619592B2 (ja) | 2011-01-26 |
| GT200000090A (es) | 2001-11-30 |
| FR2794747A1 (fr) | 2000-12-15 |
| DE60002866T2 (de) | 2004-03-11 |
| PT1189932E (pt) | 2003-09-30 |
| DK1189932T3 (da) | 2003-09-15 |
| US7005417B1 (en) | 2006-02-28 |
| CA2376490A1 (fr) | 2000-12-14 |
| DE60002866D1 (de) | 2003-06-26 |
| AU5539100A (en) | 2000-12-28 |
| UY26195A1 (es) | 2001-01-31 |
| FR2794747B1 (fr) | 2004-04-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| PA8539901A1 (es) | Novedosa sal de succinato de o-desmetil-venlafaxina | |
| ECSP055813A (es) | Quinolin-, isoquinolin- y quinazolin-oxialquilamidas y su uso como fungicidas | |
| UY28513A1 (es) | Nuevos compuestos | |
| CY1108610T1 (el) | Πεπτιδια της il-2 και παραγωγα αυτων και χρηση αυτων ως θεραπευτικοι παραγοντες | |
| ECSP034444A (es) | Derivados de 4-amino-6-fenil-pirrolo(2,3-d)pirimidina | |
| UY28623A1 (es) | Derivados de pirazol y usos de los mismos | |
| UY27446A1 (es) | Nuevos compuestos | |
| MXPA03001785A (es) | Derivados de pirazol y su uso como inhibidores de proteina cinasa. | |
| AR023727A1 (es) | Compuestos empleados en el tratamiento de padecimientos inflamatorios | |
| ATE231872T1 (de) | Thiazolopyrimidinderivate | |
| BR0107691A (pt) | Sapogeninas substituìdas e seu uso | |
| BR0107770A (pt) | Derivados de 3-fenóxi-1-fenil acetileno e seu uso como herbicidas | |
| BRPI0412320A (pt) | uso de um agente modificador de reologia, e composições de revestimento | |
| CL2004001678A1 (es) | Compuestos derivados de oxazolidinona; composicion farmaceutica; y uso de los compuestos como agentes bacterianos. | |
| BR0115080A (pt) | Derivados de acila e sulfonila de 2-(trans-1,4-diaminocicloexil)-purinas 6,9-dissubstituìdas e o uso destes como agentes antiproliferativos | |
| DE60237003D1 (de) | Verwendung von 3-positions-cyclosporin-derivaten für haarwachstum | |
| ES2194744T3 (es) | Derivados de quinocardina, su procedimiento de preparacion y su aplicacion como antifungicos. | |
| BR0309923B1 (pt) | Formulação aquosa de poliuretano, e, uso da mesma | |
| UY28622A1 (es) | Agentes antibacterianos de quinolona | |
| ATE259813T1 (de) | Triazolopyrimidinderivate | |
| DE60335563D1 (de) | Verwendung von 3-positions-cyclosporin-derivaten für haarwachstum | |
| BR0208967B1 (pt) | Composto monoazocorante fibrorreativo, mistura deste, processos de formação do referido composto e da referida mistura e uso do corante fibrorreativo | |
| BR0316544A (pt) | Compostos calcilìticos | |
| BR0206917A (pt) | Uso de antagonistas de mglur5 para o tratamento de condições prurìticas | |
| SV2003001061A (es) | Nuevos heterociclos 3 ref.lea 35361-sv |