ES2570385T3 - N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación - Google Patents

N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación

Info

Publication number
ES2570385T3
ES2570385T3 ES12795740T ES12795740T ES2570385T3 ES 2570385 T3 ES2570385 T3 ES 2570385T3 ES 12795740 T ES12795740 T ES 12795740T ES 12795740 T ES12795740 T ES 12795740T ES 2570385 T3 ES2570385 T3 ES 2570385T3
Authority
ES
Spain
Prior art keywords
formamides
pyrazolyl
methyl
production
nitrification inhibitors
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
ES12795740T
Other languages
English (en)
Inventor
Ute Radics
Hans-Joachim Niclas
Christoph Bender
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SKW Stickstoffwerke Piesteritz GmbH
Original Assignee
SKW Stickstoffwerke Piesteritz GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SKW Stickstoffwerke Piesteritz GmbH filed Critical SKW Stickstoffwerke Piesteritz GmbH
Application granted granted Critical
Publication of ES2570385T3 publication Critical patent/ES2570385T3/es
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C05—FERTILISERS; MANUFACTURE THEREOF
    • C05G—MIXTURES OF FERTILISERS COVERED INDIVIDUALLY BY DIFFERENT SUBCLASSES OF CLASS C05; MIXTURES OF ONE OR MORE FERTILISERS WITH MATERIALS NOT HAVING A SPECIFIC FERTILISING ACTIVITY, e.g. PESTICIDES, SOIL-CONDITIONERS, WETTING AGENTS; FERTILISERS CHARACTERISED BY THEIR FORM
    • C05G3/00—Mixtures of one or more fertilisers with additives not having a specially fertilising activity
    • C05G3/90—Mixtures of one or more fertilisers with additives not having a specially fertilising activity for affecting the nitrification of ammonium compounds or urea in the soil
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P60/00—Technologies relating to agriculture, livestock or agroalimentary industries
    • Y02P60/20—Reduction of greenhouse gas [GHG] emissions in agriculture, e.g. CO2
    • Y02P60/21—Dinitrogen oxide [N2O], e.g. using aquaponics, hydroponics or efficiency measures

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Soil Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fertilizers (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

N-(1H-Pirazolil-metil)-formamidas de fórmula general I:**Fórmula** caracterizadas porque R4 es >= H, halógeno, alquilo C1-C4 o cicloalquilo C3-C8, R1 y R2 independientemente entre sí representan H, alquilo C1-C4 o cicloalquilo C3-C8, R3 representa alquilo C1-C4, cicloalquilo C3-C8 o arilo C6-C10 o H.
ES12795740T 2011-12-02 2012-11-28 N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación Active ES2570385T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102011120098.7A DE102011120098B4 (de) 2011-12-02 2011-12-02 N-(1H-Pyrazolyl-methyl)formamide, Verfahren zu ihrer Herstellung und ihre Verwendung als Nitrifikationsinhibitoren
PCT/EP2012/004918 WO2013079197A1 (de) 2011-12-02 2012-11-28 N-(1h-pyrazolyl-methyl)formamide, verfahren zu ihrer herstellung und ihre verwendung als nitrifikationsinhibitoren

Publications (1)

Publication Number Publication Date
ES2570385T3 true ES2570385T3 (es) 2016-05-18

Family

ID=47294835

Family Applications (1)

Application Number Title Priority Date Filing Date
ES12795740T Active ES2570385T3 (es) 2011-12-02 2012-11-28 N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación

Country Status (4)

Country Link
EP (1) EP2785697B1 (es)
DE (1) DE102011120098B4 (es)
ES (1) ES2570385T3 (es)
WO (1) WO2013079197A1 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102013021933A1 (de) 2013-12-20 2015-06-25 Skw Stickstoffwerke Piesteritz Gmbh Verwendung von Pyrazol-Derivaten als Mittel zur Verbesserung der Trockenstresstoleranz
KR102486616B1 (ko) 2014-11-14 2023-01-09 바스프 에스이 질화작용 억제제로서의 벤질프로파르길에테르
EP3233761B1 (en) 2014-12-18 2019-02-06 Basf Se Alkynylpyrazoles as nitrification inhibitors
EP3253209A1 (en) 2015-02-06 2017-12-13 Basf Se Pyrazole compounds as nitrification inhibitors
AR104596A1 (es) 2015-05-12 2017-08-02 Basf Se Compuestos de tioéter como inhibidores de la nitrificación
US10945994B2 (en) 2015-05-14 2021-03-16 Pfizer Inc. Combinations comprising a pyrrolidine-2,5-dione IDO1 inhibitor and an anti-body
DE102016106592A1 (de) 2016-04-11 2017-10-12 Skw Stickstoffwerke Piesteritz Gmbh Verfahren zur Herstellung von N-((3(5)-Methyl-1H-pyrazol-1-yl)methyl)acetamid (MPA)
EP3458433A1 (en) 2016-05-18 2019-03-27 Basf Se Capsules comprising benzylpropargylethers for use as nitrification inhibitors
WO2019012382A1 (en) 2017-07-10 2019-01-17 Basf Se MIXTURES COMPRISING A UREASE INHIBITOR (UI) AND A NITRIFICATION INHIBITOR SUCH AS 2- (3,4-DIMETHYL-1H-PYRAZOL-1-YL) SUCCINIC ACID (DMPSA) OR 3,4-DIMETHYL PYRAZOLIUM GLYCOLATE (DMPG)
WO2019166560A1 (en) 2018-02-28 2019-09-06 Basf Se Use of n-functionalized alkoxy pyrazole compounds as nitrification inhibitors
EP3758491A1 (en) * 2018-02-28 2021-01-06 Basf Se Use of pyrazole propargyl ethers as nitrification inhibitors
EP4090158A1 (en) 2020-01-16 2022-11-23 Basf Se Mixtures comprising nitrification inhibitors and carriers
CN114981230A (zh) 2020-01-16 2022-08-30 巴斯夫欧洲公司 包含含有脲酶抑制剂的固体载体和含有硝化抑制剂的另一固体载体的混合物
AR125955A1 (es) 2021-05-21 2023-08-30 Basf Se Uso de un compuesto de alcoxi pirazol n-funcionalizado como inhibidor de nitrificación

Family Cites Families (21)

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Publication number Priority date Publication date Assignee Title
US3635690A (en) 1968-05-16 1972-01-18 Dow Chemical Co Soil treating method and composition for conserving nitrogen in soil by addition of a pyrazole thereto
US3697244A (en) 1968-10-15 1972-10-10 Dow Chemical Co Crop culture with 4h-1,2,4-triazoles
DE2745833C2 (de) 1977-10-12 1986-10-16 VEB Fahlberg-List Chemische und pharmazeutische Fabriken, DDR 3013 Magdeburg Mittel zur Hemmung bzw. Regelung der Nitrifikation von Ammoniumstickstoff in Kulturböden
DE3409317A1 (de) 1984-03-14 1985-09-19 Basf Ag, 6700 Ludwigshafen Nitrifikationsinhibierende 1-hydroxipyrazol-derivate
AU4348285A (en) 1984-06-25 1986-01-02 Dow Chemical Company, The Pyrazole growth enhancer
US4523940A (en) 1984-06-25 1985-06-18 The Dow Chemical Company Soil treating method and composition for conserving nitrogen in soil
US4969946A (en) 1986-01-29 1990-11-13 The Dow Chemical Company Soil treating method and composition for conserving nitrogen in naturally alkaline soil
SU1470737A1 (ru) 1986-09-19 1989-04-07 Предприятие П/Я Г-4302 Способ ингибировани нитрификации карбамида в почве
DE3704359A1 (de) 1987-02-12 1988-08-25 Basf Ag Azolhalbaminal-derivate und ihre verwendung als nitrifikationsinhibitoren
DD292232A5 (de) 1988-10-17 1991-07-25 Stickstoffwerke Ag Wittenberg-Piesteritz,De Mittel zur hemmung bzw. regelung der nitrifikation von ammoniumstickstoff in kulturboeden
DE4018395A1 (de) 1990-06-08 1992-02-20 Wittenberg Stickstoff Ag Mittel zur hemmung bzw. regelung der nitrifikation von ammoniumstickstoff in kulturboeden
DE4111922A1 (de) 1991-04-12 1992-10-15 Basf Ag Verfahren zur herstellung von 1-carbamoyl-pyrazolen
DE4128828A1 (de) 1991-08-30 1993-03-04 Basf Ag Ammonium- oder harnstoffhaltige duengemittel und verfahren zu ihrer herstellung
JPH07104135A (ja) 1993-10-06 1995-04-21 Sanyo Electric Co Ltd 立体画像表示装置
DE4446194A1 (de) 1994-12-23 1996-06-27 Basf Ag Verwendung von Pyrazolderivaten mit hydrophoben Resten als Nitrifikationsinhibitoren
DE19503827A1 (de) 1995-02-06 1996-08-08 Basf Ag Verwendung von schwerflüchtigen Pyrazolderivaten mit hydrophilen Gruppen als Nitrifikationsinhibitoren
DE19631764A1 (de) 1996-08-06 1998-02-12 Basf Ag Neue Nitrifikationsinhibitoren sowie die Verwendung von Polysäuren zur Behandlung von Mineraldüngemitteln die einen Nitrifikationsinhibitor enthalten
DE19822340B4 (de) 1998-05-19 2008-02-28 Skw Stickstoffwerke Piesteritz Gmbh Thermostabile schwerflüchtige Alkyl-1H-1-pyrazolylmethanamin-Derivate und deren Verwendung als Nitrifikationsinhibitoren
DE50105621D1 (de) 2000-04-14 2005-04-21 Piesteritz Stickstoff 1h-pyrazol-derivate, verfahren zu ihrer herstellung und deren verwendung zur hemmung und steuerung der nitrifikation
DE10135423A1 (de) 2000-08-08 2002-02-21 Piesteritz Stickstoff 1H-Pyrazol-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Nitrifikationsinhibitoren
DE10343277A1 (de) 2003-09-18 2005-04-21 Piesteritz Stickstoff N-(1H-Azolyl-methyl)amide, Verfahren zu ihrer Herstellung und ihre Verwendung als Nitrifikationsinhibitoren

Also Published As

Publication number Publication date
DE102011120098A1 (de) 2013-06-06
EP2785697B1 (de) 2016-02-03
EP2785697A1 (de) 2014-10-08
DE102011120098B4 (de) 2021-02-11
WO2013079197A1 (de) 2013-06-06

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