ES2688577T3 - Composiciones de buprenorfina en dosis altas y uso como analgésico - Google Patents

Composiciones de buprenorfina en dosis altas y uso como analgésico Download PDF

Info

Publication number: ES2688577T3
Authority: ES; Spain
Prior art keywords: buprenorphine; body weight; per kilogram; mammalian body; hours
Prior art date: 2010-09-03
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Active

Application number

ES11758027.4T

Other languages

English (en)

Spanish (es)

Inventor

Rachel A. Richardson

Carmela H. Luangdilok

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Zoetis Belgium SA

Original Assignee

Zoetis Belgium SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2010-09-03

Filing date

2011-09-02

Publication date

2018-11-05

2011-09-02 Application filed by Zoetis Belgium SA filed Critical Zoetis Belgium SA

2018-11-05 Application granted granted Critical

2018-11-05 Publication of ES2688577T3 publication Critical patent/ES2688577T3/es

Status Active legal-status Critical Current

2031-09-02 Anticipated expiration legal-status Critical

Links

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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Epidemiology (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Emergency Medicine (AREA)
Oil, Petroleum & Natural Gas (AREA)
Dermatology (AREA)
Biomedical Technology (AREA)
Pain & Pain Management (AREA)
Neurosurgery (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

ES11758027.4T 2010-09-03 2011-09-02 Composiciones de buprenorfina en dosis altas y uso como analgésico Active ES2688577T3 (es)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US37999610P	2010-09-03	2010-09-03
US379996P		2010-09-03
PCT/US2011/050413 WO2012031252A1 (en)	2010-09-03	2011-09-02	High dose buprenorphine compositions and use as analgesic

Publications (1)

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ES2688577T3 true ES2688577T3 (es)	2018-11-05

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Country	Link
US (1)	US9168251B2 (pl)
EP (1)	EP2611445B1 (pl)
JP (1)	JP5938409B2 (pl)
AU (1)	AU2011295694B2 (pl)
CA (1)	CA2808237C (pl)
CY (1)	CY1120920T1 (pl)
DK (1)	DK2611445T3 (pl)
ES (1)	ES2688577T3 (pl)
PL (1)	PL2611445T3 (pl)
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WO2014016428A1 (en)	2012-07-26	2014-01-30	Camurus Ab	Opioid formulations
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WO2019144079A1 (en) *	2018-01-22	2019-07-25	Yuhua Li	Pharmaceutical composition for sustained release delivery of buprenorphine
US11471475B1 (en)	2022-03-08	2022-10-18	Ralph P. Stone	Ophthalmic suspension vehicles and related methods for pharmaceutical ingredient delivery

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US5240711A (en) *	1989-11-29	1993-08-31	Lts Lohmann Therapie-Systeme Gmbh & Co. Kg	Transdermal therapeutic system comprising as active component buprenorphine
JP3701693B2 (ja) *	1993-12-28	2005-10-05	日本製薬株式会社	鎮痛薬含有注射用徐放性脂肪乳剤
US5968547A (en) *	1997-02-24	1999-10-19	Euro-Celtique, S.A.	Method of providing sustained analgesia with buprenorphine
WO1999012606A1 (en) *	1997-09-08	1999-03-18	Becton Dickinson And Company	Iontophoretic delivery of buprenorphine
GB0201367D0 (en) *	2002-01-22	2002-03-13	Ml Lab Plc	Composition
DE602004011055T2 (de) *	2003-07-25	2008-12-18	Euro-Celtique S.A.	Präoperative behandlung von postoperativen schmerzen
AU2006316607A1 (en) *	2005-11-21	2007-05-31	Schering-Plough Pty. Limited	Pharmaceutical compositions comprising buprenorphine
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BRPI0916761A2 (pt) *	2008-07-17	2018-02-14	Ap Pharma	formulações analgésicas injetáveis de ação prolongada para animais

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Publication number	Publication date
AU2011295694B2 (en)	2015-02-05
JP5938409B2 (ja)	2016-06-22
WO2012031252A1 (en)	2012-03-08
PL2611445T3 (pl)	2018-12-31
EP2611445A1 (en)	2013-07-10
CY1120920T1 (el)	2019-12-11
PT2611445T (pt)	2018-10-24
US9168251B2 (en)	2015-10-27
DK2611445T3 (en)	2018-10-22
CA2808237A1 (en)	2012-03-08
AU2011295694A1 (en)	2013-03-14
JP2013536872A (ja)	2013-09-26
EP2611445B1 (en)	2018-08-15
US20140329843A1 (en)	2014-11-06
CA2808237C (en)	2019-08-06

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